Potent Kv1.3 inhibitors from correolide—modification of the C18 position
Bao, Jianming, Miao, Shouwu, Kayser, Frank, Kotliar, Andrew J., Baker, Robert K., Doss, George A., Felix, John P., Bugianesi, Randal M., Slaughter, Robert S., Kaczorowski, Gregory J., Garcia, Maria L., Ha, Sookhee N., Castonguay, Laurie, Koo, Gloria C., Shah, Kashmira, Springer, Marty S., Staruch, Mary Jo, Parsons, William H., Rupprecht, Kathleen M.
Published in Bioorganic & medicinal chemistry letters (17.01.2005)
Published in Bioorganic & medicinal chemistry letters (17.01.2005)
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p38 MAP kinase inhibitors: Metabolically stabilized piperidine-substituted quinolinones and naphthyridinones
Bao, Jianming, Hunt, Julianne A., Miao, Shouwu, Rupprecht, Kathleen M., Stelmach, John E., Liu, Luping, Ruzek, Rowena D., Sinclair, Peter J., Pivnichny, James V., Hop, Cornelis E.C.A., Kumar, Sanjeev, Zaller, Dennis M., Shoop, Wesley L., O’Neill, Edward A., O’Keefe, Stephen J., Thompson, Chris M., Cubbon, Rose M., Wang, Ruixiu, Zhang, Wen Xiao, Thompson, James E., Doherty, James B.
Published in Bioorganic & medicinal chemistry letters (2006)
Published in Bioorganic & medicinal chemistry letters (2006)
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Benzamide derivatives as blockers of Kv1.3 ion channel
Miao, Shouwu, Bao, Jianming, Garcia, Maria L., Goulet, Joung L., Hong, Xingfang J., Kaczorowski, Gregory J., Kayser, Frank, Koo, Gloria C., Kotliar, Andrew, Schmalhofer, William A., Shah, Kashmira, Sinclair, Peter J., Slaughter, Robert S., Springer, Marty S., Staruch, Mary Jo, Tsou, Nancy N., Wong, Frederick, Parsons, William H., Rupprecht, Kathleen M.
Published in Bioorganic & medicinal chemistry letters (24.03.2003)
Published in Bioorganic & medicinal chemistry letters (24.03.2003)
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1,3,8-Triazaspiro[4.5]decane-2,4-diones as Efficacious Pan-Inhibitors of Hypoxia-Inducible Factor Prolyl Hydroxylase 1–3 (HIF PHD1–3) for the Treatment of Anemia
Vachal, Petr, Miao, Shouwu, Pierce, Joan M, Guiadeen, Deodial, Colandrea, Vincent J, Wyvratt, Matthew J, Salowe, Scott P, Sonatore, Lisa M, Milligan, James A, Hajdu, Richard, Gollapudi, Anantha, Keohane, Carol A, Lingham, Russell B, Mandala, Suzanne M, DeMartino, Julie A, Tong, Xinchun, Wolff, Michael, Steinhuebel, Dietrich, Kieczykowski, Gerard R, Fleitz, Fred J, Chapman, Kevin, Athanasopoulos, John, Adam, Gregory, Akyuz, Can D, Jena, Dhirendra K, Lusen, Jeffrey W, Meng, Juncai, Stein, Benjamin D, Xia, Lei, Sherer, Edward C, Hale, Jeffrey J
Published in Journal of medicinal chemistry (12.04.2012)
Published in Journal of medicinal chemistry (12.04.2012)
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Discovery of Chromane Propionic Acid Analogues as Selective Agonists of GPR120 with in Vivo Activity in Rodents
Adams, Gregory L, Velazquez, Francisco, Jayne, Charles, Shah, Unmesh, Miao, Shouwu, Ashley, Eric R, Madeira, Maria, Akiyama, Taro E, Di Salvo, Jerry, Suzuki, Takao, Wang, Nengxue, Truong, Quang, Gilbert, Eric, Zhou, Dan, Verras, Andreas, Kirkland, Melissa, Pachanski, Michele, Powles, Maryann, Yin, Wu, Ujjainwalla, Feroze, Venkatraman, Srikanth, Edmondson, Scott D
Published in ACS medicinal chemistry letters (12.01.2017)
Published in ACS medicinal chemistry letters (12.01.2017)
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Discovery of MK-8831, A Novel Spiro-Proline Macrocycle as a Pan-Genotypic HCV-NS3/4a Protease Inhibitor
Neelamkavil, Santhosh F, Agrawal, Sony, Bara, Thomas, Bennett, Chad, Bhat, Sathesh, Biswas, Dipshikha, Brockunier, Linda, Buist, Nicole, Burnette, Duane, Cartwright, Mark, Chackalamannil, Samuel, Chase, Robert, Chelliah, Mariappan, Chen, Austin, Clasby, Martin, Colandrea, Vincent J, Davies, Ian W, Eagen, Keith, Guo, Zhuyan, Han, Yongxin, Howe, John, Jayne, Charles, Josien, Hubert, Kargman, Stacia, Marcantonio, Karen, Miao, Shouwu, Miller, Randy, Nolting, Andrew, Pinto, Patrick, Rajagopalan, Murali, Ruck, Rebecca T, Shah, Unmesh, Soriano, Aileen, Sperbeck, Donald, Velazquez, Francisco, Wu, Jin, Xia, Yan, Venkatraman, Srikanth
Published in ACS medicinal chemistry letters (14.01.2016)
Published in ACS medicinal chemistry letters (14.01.2016)
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MK-7128, a novel CB1 receptor inverse agonist, improves scopolamine-induced learning and memory deficits in mice
Dillon, Gregory M, Lubbers, Laura S, Ferguson, Mitchell T, Lao, Julie Z, Huang, Ruey-Ruey C, Xiao, Jing C, Fong, Tung M, Hale, Jeffrey J, Rupprecht, Kathleen, Miao, Shouwu, Rowe, Blake A, Kornecook, Thomas J, Dodart, Jean-Cosme
Published in Behavioural pharmacology (01.04.2011)
Published in Behavioural pharmacology (01.04.2011)
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Identification of a New Class of Inhibitors of the Voltage-Gated Potassium Channel, Kv1.3, with Immunosuppressant Properties
Schmalhofer, William A, Bao, Jianming, McManus, Owen B, Green, Brian, Matyskiela, Mary, Wunderler, Denise, Bugianesi, Randal M, Felix, John P, Hanner, Markus, Linde-Arias, Ana-Rosa, Ponte, Cristiano G, Velasco, Lucia, Koo, Gloria, Staruch, Mary Jo, Miao, Shouwu, Parsons, William H, Rupprecht, Kathleen, Slaughter, Robert S, Kaczorowski, Gregory J, Garcia, Maria L
Published in Biochemistry (Easton) (18.06.2002)
Published in Biochemistry (Easton) (18.06.2002)
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Journal Article
Novel Fragmentation Reaction of Correolide
Bao, Jianming, Baker, Robert K, Doss, George A, Kayser, Frank, Kotliar, Andrew, Miao, Shouwu, Parsons, William H, Rupprecht, Kathleen M
Published in Organic letters (30.05.2002)
Published in Organic letters (30.05.2002)
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4-AMINO-2-(1HPYRAZOLO[3,4-B]PYRIDIN-3-YL)-6-OXO-6,7-DIHYDRO-5H-PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AND THE RESPECTIVE (1H-INDAZOL-3-YL) DERIVATIVES AS CGMP MODULATORS FOR TREATING CARDIOVASCULAR DISEASES
MIAO, SHOUWU, FU, JIANMIN, CHEN, YI-HENG, LI, HONG, WHITEHEAD, ALAN, SMITH, CAMERON, J, STELMACH, JOHN, ZHANG, YONG, GARFUNKLE, JOIE, LI, GUOQING, JI, GANG, BERGER, RAPHELLE, ZHANG, RUI, JIANG, FALONG, RAGHAVAN, SUBHAREKHA
Year of Publication 08.11.2022
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Year of Publication 08.11.2022
Patent
Identification of a New Class of Inhibitors of the Voltage-Gated Potassium Channel, K v 1.3, with Immunosuppressant Properties
Schmalhofer, William A., Bao, Jianming, McManus, Owen B., Green, Brian, Matyskiela, Mary, Wunderler, Denise, Bugianesi, Randal M., Felix, John P., Hanner, Markus, Linde-Arias, Ana-Rosa, Ponte, Cristiano G., Velasco, Lucia, Koo, Gloria, Staruch, Mary Jo, Miao, Shouwu, Parsons, William H., Rupprecht, Kathleen, Slaughter, Robert S., Kaczorowski, Gregory J., Garcia, Maria L.
Published in Biochemistry (Easton) (01.06.2002)
Published in Biochemistry (Easton) (01.06.2002)
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4-AMINO-2-(1H-PYRAZOLO[3,4-B]PYRIDIN-3-YL)-6-OXO-6,7-DIHYDRO-5H-PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AND THE RESPECTIVE (1H-INDAZOL-3-YL) DERIVATIVES AS CGMP MODULATORS FOR TREATING CARDIOVASCULAR DISEASES
CHEN, Yi-Heng, GARFUNKLE, Joie, ZHANG, Rui, JI, Gang, MIAO, Shouwu, BERGER, Raphelle, LI, Hong, SMITH, Cameron J, STELMACH, John, FU, Jianmin, JIANG, Falong, WHITEHEAD, Alan, ZHANG, Yong, RAGHAVAN, Subharekha, LI, Guoqing
Year of Publication 20.04.2021
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Year of Publication 20.04.2021
Patent
4-AMINO-2-(1H-PYRAZOLO[3,4-B]PYRIDIN-3-YL)-6-OXO-6,7-DIHYDRO-5H-PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AND THE RESPECTIVE (1H-INDAZOL-3-YL) DERIVATIVES AS CGMP MODULATORS FOR TREATING CARDIOVASCULAR DISEASES
CHEN, Yi-Heng, GARFUNKLE, Joie, ZHANG, Rui, JI, Gang, MIAO, Shouwu, SMITH, Cameron, BERGER, Raphelle, LI, Hong, STELMACH, John, FU, Jianmin, JIANG, Falong, WHITEHEAD, Alan, ZHANG, Yong, RAGHAVAN, Subharekha, LI, Guoqing
Year of Publication 30.11.2020
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Year of Publication 30.11.2020
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4-AMINO-2-(1H-PYRAZOLO[3,4-B]PYRIDIN-3-YL)-6-OXO-6,7-DIHYDRO-5H-PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AND THE RESPECTIVE (1H-INDAZOL-3-YL) DERIVATIVES AS CGMP MODULATORS FOR TREATING CARDIOVASCULAR DISEASES
Li, Guoqing, Zhang, Rui, Li, Hong, Whitehead, Alan, Ji, Gang, Jiang, Falong, Chen, Yi-Heng, Berger, Raphelle, Raghavan, Subharekha, Garfunkle, Joie, Stelmach, John, Fu, Jianmin, Miao, Shouwu, Zhang, Yong, Smith, Cameron J
Year of Publication 13.11.2020
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Year of Publication 13.11.2020
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4-AMINO-2-(1H-PYRAZOLO(3,4-B)PYRIDIN-3-YL)-6-OXO-6,7-DIHYDRO-5H-PYRROLO(2,3-D)PYRIMIDINE DERIVATIVES AND THE RESPECTIVE (1H-INDAZOL-3-YL) DERIVATIVES AS CGMP MODULATORS FOR TREATING CARDIOVASCULAR DISEASES
MIAO Shouwu, JI Gang, CHEN Yi-Heng, SMITH Cameron J, JIANG Falong, FU Jianmin, RAGHAVAN Subharekha, LI Hong, WHITEHEAD Alan, GARFUNKLE Joie, STELMACH John, BERGER Raphelle, LI Guoqing, ZHANG Rui, ZHANG Yong
Year of Publication 31.07.2020
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Year of Publication 31.07.2020
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4-AMINO-2-(1H-PYRAZOLO[3,4-B]PYRIDIN-3-YL)-6-OXO-6,7-DIHYDRO-5H-PYRROLO[2,3- D]PYRIMIDINDERIVATER OG TILSVARENDE (1H-INDAZOL-3-YL) DERIVATER SOM CGMP- MODULATORER TIL BEHANDLING AF KARDIOVASKULÆRE SYGDOMME
CHEN, Yi-Heng, GARFUNKLE, Joie, ZHANG, Rui, JI, Gang, MIAO, Shouwu, BERGER, Raphelle, LI, Hong, SMITH, Cameron, J, STELMACH, John, FU, Jianmin, JIANG, Falong, WHITEHEAD, Alan, ZHANG, Yong, RAGHAVAN, Subharekha, LI, Guoqing
Year of Publication 15.06.2020
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Year of Publication 15.06.2020
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4-AMINO-2-(1H-PYRAZOLO[3,4-B]PYRIDIN-3-YL)-6-OXO-6,7-DIHYDRO-5H-PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AND THE RESPECTIVE (1H-INDAZOL-3-YL) DERIVATIVES AS CGMP MODULATORS FOR TREATING CARDIOVASCULAR DISEASES
CHEN, Yi-Heng, GARFUNKLE, Joie, ZHANG, Rui, JI, Gang, MIAO, Shouwu, SMITH, Cameron, BERGER, Raphelle, LI, Hong, STELMACH, John, FU, Jianmin, JIANG, Falong, WHITEHEAD, Alan, ZHANG, Yong, RAGHAVAN, Subharekha, LI, Guoqing
Year of Publication 10.06.2020
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Year of Publication 10.06.2020
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4-AMINO-2-(1H-PYRAZOLO[3,4-B]PYRIDIN-3-YL)-6-OXO-6,7-DIHYDRO-5H-PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AND THE RESPECTIVE (1H-INDAZOL-3-YL) DERIVATIVES AS CGMP MODULATORS FOR TREATING CARDIOVASCULAR DISEASES
CHEN, Yi-Heng, GARFUNKLE, Joie, ZHANG, Rui, JI, Gang, MIAO, Shouwu, BERGER, Raphelle, LI, Hong, SMITH, Cameron, J, STELMACH, John, FU, Jianmin, JIANG, Falong, WHITEHEAD, Alan, ZHANG, Yong, RAGHAVAN, Subharekha, LI, Guoqing
Year of Publication 01.04.2020
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Year of Publication 01.04.2020
Patent