Antimalarial pharmacology and therapeutics of atovaquone
Nixon, Gemma L, Moss, Darren M, Shone, Alison E, Lalloo, David G, Fisher, Nicholas, O'Neill, Paul M, Ward, Stephen A, Biagini, Giancarlo A
Published in Journal of antimicrobial chemotherapy (01.05.2013)
Published in Journal of antimicrobial chemotherapy (01.05.2013)
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Generation of quinolone antimalarials targeting the Plasmodium falciparum mitochondrial respiratory chain for the treatment and prophylaxis of malaria
Biagini, Giancarlo A, Fisher, Nicholas, Shone, Alison E, Mubaraki, Murad A, Srivastava, Abhishek, Hill, Alisdair, Antoine, Thomas, Warman, Ashley J, Davies, Jill, Pidathala, Chandrakala, Amewu, Richard K, Leung, Suet C, Sharma, Raman, Gibbons, Peter, Hong, David W, Pacorel, Bénédicte, Lawrenson, Alexandre S, Charoensutthivarakul, Sitthivut, Taylor, Lee, Berger, Olivier, Mbekeani, Alison, Stocks, Paul A, Nixon, Gemma L, Chadwick, James, Hemingway, Janet, Delves, Michael J, Sinden, Robert E, Zeeman, Anne-Marie, Kocken, Clemens H. M, Berry, Neil G, O’Neill, Paul M, Ward, Stephen A
Published in Proceedings of the National Academy of Sciences - PNAS (22.05.2012)
Published in Proceedings of the National Academy of Sciences - PNAS (22.05.2012)
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Development of a defined compost system for the study of plant-microbe interactions
Masters-Clark, E, Shone, E, Paradelo, M, Hirsch, P R, Clark, I M, Otten, W, Brennan, F, Mauchline, T H
Published in Scientific reports (05.05.2020)
Published in Scientific reports (05.05.2020)
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Identification, Design and Biological Evaluation of Bisaryl Quinolones Targeting Plasmodium falciparum Type II NADH:Quinone Oxidoreductase (PfNDH2)
Pidathala, Chandrakala, Amewu, Richard, Pacorel, Bénédicte, Nixon, Gemma L, Gibbons, Peter, Hong, W. David, Leung, Suet C, Berry, Neil G, Sharma, Raman, Stocks, Paul A, Srivastava, Abhishek, Shone, Alison E, Charoensutthivarakul, Sitthivut, Taylor, Lee, Berger, Olivier, Mbekeani, Alison, Hill, Alasdair, Fisher, Nicholas E, Warman, Ashley J, Biagini, Giancarlo A, Ward, Stephen A, O’Neill, Paul M
Published in Journal of medicinal chemistry (08.03.2012)
Published in Journal of medicinal chemistry (08.03.2012)
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Identification of a 1,2,4,5-Tetraoxane Antimalarial Drug-Development Candidate (RKA 182) with Superior Properties to the Semisynthetic Artemisinins
O'Neill, Paul M, Amewu, Richard K, Nixon, Gemma L, Bousejra ElGarah, Fatima, Mungthin, Mathirut, Chadwick, James, Shone, Alison E, Vivas, Livia, Lander, Hollie, Barton, Victoria, Muangnoicharoen, Sant, Bray, Patrick G, Davies, Jill, Park, B. Kevin, Wittlin, Sergio, Brun, Reto, Preschel, Michael, Zhang, Kesheng, Ward, Stephen A
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Published in Angewandte Chemie (International ed.) (02.08.2010)
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O’Neill, Paul M, Park, B. Kevin, Shone, Alison E, Maggs, James L, Roberts, Phillip, Stocks, Paul A, Biagini, Giancarlo A, Bray, Patrick G, Gibbons, Peter, Berry, Neil, Winstanley, Peter A, Mukhtar, Amira, Bonar-Law, Richard, Hindley, Stephen, Bambal, Ramesh B, Davis, Charles B, Bates, Martin, Hart, Timothy K, Gresham, Stephanie L, Lawrence, Ron M, Brigandi, Richard A, Gomez-delas-Heras, Federico M, Gargallo, Domingo V, Ward, Stephen A
Published in Journal of medicinal chemistry (12.03.2009)
Published in Journal of medicinal chemistry (12.03.2009)
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Discovery of Potent Small-Molecule Inhibitors of Multidrug-Resistant Plasmodium falciparum Using a Novel Miniaturized High-Throughput Luciferase-Based Assay
Lucumi, Edinson, Darling, Claire, Jo, Hyunil, Napper, Andrew D, Chandramohanadas, Rajesh, Fisher, Nicholas, Shone, Alison E, Jing, Huiyan, Ward, Stephen A, Biagini, Giancarlo A, DeGrado, William F, Diamond, Scott L, Greenbaum, Doron C
Published in Antimicrobial Agents and Chemotherapy (01.09.2010)
Published in Antimicrobial Agents and Chemotherapy (01.09.2010)
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Rational Design, Synthesis, and Biological Evaluation of Heterocyclic Quinolones Targeting the Respiratory Chain of Mycobacterium tuberculosis
Hong, W. David, Gibbons, Peter D, Leung, Suet C, Amewu, Richard, Stocks, Paul A, Stachulski, Andrew, Horta, Pedro, Cristiano, Maria L. S, Shone, Alison E, Moss, Darren, Ardrey, Alison, Sharma, Raman, Warman, Ashley J, Bedingfield, Paul T. P, Fisher, Nicholas E, Aljayyoussi, Ghaith, Mead, Sally, Caws, Maxine, Berry, Neil G, Ward, Stephen A, Biagini, Giancarlo A, O’Neill, Paul M, Nixon, Gemma L
Published in Journal of medicinal chemistry (11.05.2017)
Published in Journal of medicinal chemistry (11.05.2017)
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Targeting the mitochondrial electron transport chain of Plasmodium falciparum: new strategies towards the development of improved antimalarials for the elimination era
Nixon, Gemma L, Pidathala, Chandrakala, Shone, Alison E, Antoine, Thomas, Fisher, Nicholas, O'Neill, Paul M, Ward, Stephen A, Biagini, Giancarlo A
Published in Future medicinal chemistry (01.09.2013)
Published in Future medicinal chemistry (01.09.2013)
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Identification, Design and Biological Evaluation of Heterocyclic Quinolones Targeting Plasmodium falciparum Type II NADH:Quinone Oxidoreductase (PfNDH2)
Leung, Suet C, Gibbons, Peter, Amewu, Richard, Nixon, Gemma L, Pidathala, Chandrakala, Hong, W. David, Pacorel, Bénédicte, Berry, Neil G, Sharma, Raman, Stocks, Paul A, Srivastava, Abhishek, Shone, Alison E, Charoensutthivarakul, Sitthivut, Taylor, Lee, Berger, Olivier, Mbekeani, Alison, Hill, Alasdair, Fisher, Nicholas E, Warman, Ashley J, Biagini, Giancarlo A, Ward, Stephen A, O’Neill, Paul M
Published in Journal of medicinal chemistry (08.03.2012)
Published in Journal of medicinal chemistry (08.03.2012)
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Semi-synthetic and synthetic 1,2,4-trioxaquines and 1,2,4-trioxolaquines : synthesis, preliminary SAR and comparison with acridine endoperoxide conjugates
ARAUJO, Nuna C. P, BARTON, Victoria, JONES, Michael, STOCKS, Paul A, WARD, Stephen A, DAVIES, Jill, BRAY, Patrick G, SHONE, Alison E, CRISTIANO, Maria L. S, O'NEILL, Paul M
Published in Bioorganic & medicinal chemistry letters (01.04.2009)
Published in Bioorganic & medicinal chemistry letters (01.04.2009)
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Endoperoxide Carbonyl Falcipain 2/3 Inhibitor Hybrids: Toward Combination Chemotherapy of Malaria through a Single Chemical Entity
Gibbons, Peter, Verissimo, Edite, Araujo, Nuna C, Barton, Victoria, Nixon, Gemma L, Amewu, Richard K, Chadwick, James, Stocks, Paul A, Biagini, Giancarlo A, Srivastava, Abhishek, Rosenthal, Philip J, Gut, Jiri, Guedes, Rita C, Moreira, Rui, Sharma, Raman, Berry, Neil, Cristiano, M. Lurdes S, Shone, Alison E, Ward, Stephen A, O’Neill, Paul M
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Published in Journal of medicinal chemistry (25.11.2010)
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Synthesis, Antimalarial Activity, and Preclinical Pharmacology of a Novel Series of 4′-Fluoro and 4′-Chloro Analogues of Amodiaquine. Identification of a Suitable “Back-Up” Compound for N-tert-Butyl Isoquine
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Published in Journal of medicinal chemistry (09.04.2009)
Published in Journal of medicinal chemistry (09.04.2009)
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Identification of Novel Antimalarial Chemotypes via Chemoinformatic Compound Selection Methods for a High-Throughput Screening Program against the Novel Malarial Target, PfNDH2: Increasing Hit Rate via Virtual Screening Methods
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Published in Journal of medicinal chemistry (12.04.2012)
Published in Journal of medicinal chemistry (12.04.2012)
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The development of quinolone esters as novel antimalarial agents targeting the Plasmodium falciparum bc1 protein complex
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Published in MedChemComm (01.01.2012)
Published in MedChemComm (01.01.2012)
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Comparative preclinical drug metabolism and pharmacokinetic evaluation of novel 4-aminoquinoline anti-malarials
Davis, Charles B., Bambal, Ramesh, Moorthy, Ganesh S., Hugger, Erin, Xiang, Hong, Park, Brian Kevin, Shone, Allison E., O’Neill, Paul M., Ward, Stephen A.
Published in Journal of pharmaceutical sciences (01.01.2009)
Published in Journal of pharmaceutical sciences (01.01.2009)
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P5.034 British Co-Operative Clinical Group (BCCG) Project - How Often Are Men Who Have Sex with Men (MSM) Advised to Attend For Repeat Sexual Health Screening in the UK?
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Published in Sexually transmitted infections (01.07.2013)
Published in Sexually transmitted infections (01.07.2013)
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The development of quinoloneesters as novel antimalarial agents targeting the Plasmodium falciparum bc 1 protein complex
Cowley, Robin, Leung, Suet, Fisher, Nicholas, Al-Helal, Mohammed, Berry, Neil G., Lawrenson, Alexandre S., Sharma, Raman, Shone, Alison E., Ward, Stephen A., Biagini, Giancarlo A., O′Neill, Paul M.
Published in MedChemComm (2012)
Published in MedChemComm (2012)
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