Synthesis and structure–activity relationships of new carbonyl guanidine derivatives as novel dual 5-HT2B and 5-HT7 receptor antagonists
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Published in Bioorganic & medicinal chemistry (15.12.2013)
Published in Bioorganic & medicinal chemistry (15.12.2013)
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Synthesis and structure–activity relationships of new carbonyl guanidine derivatives as novel dual 5-HT2B and 5-HT7 receptor antagonists. Part 2
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Published in Bioorganic & medicinal chemistry (01.08.2014)
Published in Bioorganic & medicinal chemistry (01.08.2014)
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Synthesis and pharmacological evaluation of optically pure, novel carbonyl guanidine derivatives as dual 5-HT2B and 5-HT7 receptor antagonists
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Published in Bioorganic & medicinal chemistry (01.11.2014)
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Published in European journal of pharmacology (14.11.2007)
Published in European journal of pharmacology (14.11.2007)
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Inhibitory Effects of Ramosetron, a Potent and Selective 5-HT3–Receptor Antagonist, on Conditioned Fear Stress–Induced Abnormal Defecation and Normal Defecation in Rats: Comparative Studies With Antidiarrheal and Spasmolytic Agents
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Effects of serotonin 5-HT3 receptor antagonists on CRF-induced abnormal colonic water transport and defecation in rats
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Published in European journal of pharmacology (10.06.2008)
Published in European journal of pharmacology (10.06.2008)
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A novel GABAB receptor positive allosteric modulator, ASP8062, exerts analgesic effects in a rat model of fibromyalgia
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Published in European journal of pharmacology (15.12.2019)
Published in European journal of pharmacology (15.12.2019)
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Effect of antiemetics on zolbetuximab-induced gastric injury and emesis in ferrets
Kinugasa, Fumitaka, Kajikawa, Satoru, Weng, Jane, Ugawa, Tohru, Fushiki, Hiroshi, Yamanaka, Yosuke, Nagata, Masanori, Haggerty, Gillian, Akuzawa, Shinobu, Nakazawa, Taisuke, Suzuki, Hiroshi, Sawamoto, Taiji
Published in Journal of pharmacological sciences (01.11.2024)
Published in Journal of pharmacological sciences (01.11.2024)
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Inhibitory Effects of Ramosetron, a Potent and Selective 5-HT3-Receptor Antagonist, on Conditioned Fear Stress-Induced Abnormal Defecation and Normal Defecation in Rats：Comparative Studies With Antidiarrheal and Spasmolytic Agents
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Published in Journal of Pharmacological Sciences (01.02.2008)
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Published in Journal of Pharmacological Sciences (01.02.2008)
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New thiazole derivatives as potent and selective 5-hydroxytriptamine 3 (5-HT3) receptor agonists for the treatment of constipation
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Published in Bioorganic & medicinal chemistry (03.04.2003)
Published in Bioorganic & medicinal chemistry (03.04.2003)
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116.1 GABA-B Agonist Baclofen Normalizes Auditory-Evoked Neural Oscillations and Some Cognitive Deficits in a Fragile X Syndrome Mouse Model
Siegel, Steven, Sinclair, Dunan, Matsumoto, Mitsuyuki, Featherstone, Robert, Melnechenko, Olya, Nascheck, Melissa, Weger, Rachel, Akuzawa, Shinobu, Pance, Katarina, Wright, Saidha, Nam, Jehee, Du, Austin
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Comparison of [3H]YM060 binding to native and cloned rat 5-HT3 receptors
AKUZAWA, S, MIYAKE, A, MIYATA, K, FUKUTOMI, H
Published in European journal of pharmacology (25.01.1996)
Published in European journal of pharmacology (25.01.1996)
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A novel GABA B receptor positive allosteric modulator, ASP8062, exerts analgesic effects in a rat model of fibromyalgia
Murai, Nobuhito, Kondo, Yuji, Akuzawa, Shinobu, Mihara, Takuma, Shiraishi, Nobuyuki, Kakimoto, Shuichiro, Matsumoto, Mitsuyuki
Published in European journal of pharmacology (15.12.2019)
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Published in European journal of pharmacology (15.12.2019)
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Synthesis and pharmacological evaluation of optically pure, novel carbonyl guanidine derivatives as dual 5-HT sub(2B) and 5-HT sub(7) receptor antagonists
Moritomo, Ayako, Yamada, Hiroyoshi, Matsuzawa-Nomura, Takaho, Watanabe, Toshihiro, Itahana, Hirotsune, Oku, Makoto, Akuzawa, Shinobu, Okada, Minoru
Published in Bioorganic & medicinal chemistry (01.11.2014)
Published in Bioorganic & medicinal chemistry (01.11.2014)
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Biological Activity of Analogues of YM022. Novel (3-Amino Substituted Phenyl)urea Derivatives of 1, 4-Benzodiazepin-2-one as Gastrin : Cholecystokinin-B Receptor Antagonists
SATOH, Masato, OKAMOTO, Yoshinori, KOSHIO, Hiroyuki, OHTA, Mitsuaki, NISHIDA, Akito, AKUZAWA, Shinobu, MIYATA, Keiji, MASE, Toshiyasu, SEMPLE, Graeme
Published in Chemical & pharmaceutical bulletin (01.07.1996)
Published in Chemical & pharmaceutical bulletin (01.07.1996)
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Hepatic accumulation and hepatotoxicity of luteoskyrin in mice
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Published in Toxicology letters (01.06.1992)
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Effects of serotonin 5-HT(3) receptor antagonists on CRF-induced abnormal colonic water transport and defecation in rats
Hirata, Takuya, Keto, Yoshihiro, Nakata, Mari, Takeuchi, Asako, Funatsu, Toshiyuki, Akuzawa, Shinobu, Sasamata, Masao, Miyata, Keiji
Published in European journal of pharmacology (10.06.2008)
Published in European journal of pharmacology (10.06.2008)
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