X-ray structure of a bacterial oligosaccharyltransferase
Lizak, Christian, Gerber, Sabina, Numao, Shin, Aebi, Markus, Locher, Kaspar P.
Published in Nature (London) (01.06.2011)
Published in Nature (London) (01.06.2011)
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Journal Article
Feasibility and physiological relevance of designing highly potent aminopeptidase-sparing leukotriene A4 hydrolase inhibitors
Numao, Shin, Hasler, Franziska, Laguerre, Claire, Srinivas, Honnappa, Wack, Nathalie, Jäger, Petra, Schmid, Andres, Osmont, Arnaud, Röthlisberger, Patrik, Houguenade, Jeremy, Bergsdorf, Christian, Dawson, Janet, Carte, Nathalie, Hofmann, Andreas, Markert, Christian, Hardaker, Liz, Billich, Andreas, Wolf, Romain M., Penno, Carlos A., Bollbuck, Birgit, Miltz, Wolfgang, Röhn, Till A.
Published in Scientific reports (19.10.2017)
Published in Scientific reports (19.10.2017)
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Journal Article
Definition of the bacterial N-glycosylation site consensus sequence
Kowarik, Michael, Young, N Martin, Numao, Shin, Schulz, Benjamin L, Hug, Isabelle, Callewaert, Nico, Mills, Dominic C, Watson, David C, Hernandez, Marcela, Kelly, John F, Wacker, Michael, Aebi, Markus
Published in The EMBO journal (03.05.2006)
Published in The EMBO journal (03.05.2006)
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Journal Article
N-Linked Glycosylation of Folded Proteins by the Bacterial Oligosaccharyltransferase
Kowarik, Michael, Numao, Shin, Feldman, Mario F., Schulz, Benjamin L., Callewaert, Nico, Kiermaier, Eva, Catrein, Ina, Aebi, Markus
Published in Science (American Association for the Advancement of Science) (17.11.2006)
Published in Science (American Association for the Advancement of Science) (17.11.2006)
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Journal Article
A combined method for producing homogeneous glycoproteins with eukaryotic N-glycosylation
Aebi, Markus, Wang, Lai-Xi, Schwarz, Flavio, Huang, Wei, Li, Cishan, Schulz, Benjamin L, Lizak, Christian, Palumbo, Alessandro, Numao, Shin, Neri, Dario
Published in Nature chemical biology (01.04.2010)
Published in Nature chemical biology (01.04.2010)
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Journal Article
Drug discovery strategies for novel leukotriene A4 hydrolase inhibitors
Röhn, Till A, Numao, Shin, Otto, Heike, Loesche, Christian, Thoma, Gebhard
Published in Expert opinion on drug discovery (02.12.2021)
Published in Expert opinion on drug discovery (02.12.2021)
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Journal Article
Discovery of LYS006, a Potent and Highly Selective Inhibitor of Leukotriene A(4) Hydrolase
Markert, Christian, Thoma, Gebhard, Srinivas, Honnappa, Bollbuck, Birgit, Lueoend, Rainer M., Miltz, Wolfgang, Waelchli, Rudolf, Wolf, Romain, Hinrichs, Juergen, Bergsdorf, Christian, Azzaoui, Kamal, Penno, Carlos A., Klein, Kai, Wack, Nathalie, Jaeger, Petra, Hasler, Franziska, Beerli, Christian, Loetscher, Pius, Dawson, Janet, Wieczorek, Grazyna, Numao, Shin, Littlewood-Evans, Amanda, Roehn, Till A.
Published in Journal of medicinal chemistry (25.02.2021)
Published in Journal of medicinal chemistry (25.02.2021)
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Journal Article
Advancements in Assay Technologies and Strategies to Enable Drug Discovery
Busby, Scott A., Carbonneau, Seth, Concannon, John, Dumelin, Christoph E., Lee, YounKyoung, Numao, Shin, Renaud, Nicole, Smith, Thomas M., Auld, Douglas S.
Published in ACS chemical biology (16.10.2020)
Published in ACS chemical biology (16.10.2020)
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Journal Article
Evaluation of 5 H ‐Thiazolo[3,2‐α]pyrimidin‐5‐ones as Potential GluN2A PET Tracers
He, Yingfang, Whitehead, David M., Briard, Emmanuelle, Numao, Shin, Mu, Linjing, Schibli, Roger, Ametamey, Simon M., Auberson, Yves P.
Published in ChemMedChem (15.12.2020)
Published in ChemMedChem (15.12.2020)
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Journal Article
Front Cover: Evaluation of 5H‐Thiazolo[3,2‐α]pyrimidin‐5‐ones as Potential GluN2A PET Tracers (ChemMedChem 24/2020)
He, Yingfang, Whitehead, David M., Briard, Emmanuelle, Numao, Shin, Mu, Linjing, Schibli, Roger, Ametamey, Simon M., Auberson, Yves P.
Published in ChemMedChem (15.12.2020)
Published in ChemMedChem (15.12.2020)
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Journal Article
Front Cover: Evaluation of 5 H ‐Thiazolo[3,2‐α]pyrimidin‐5‐ones as Potential GluN2A PET Tracers (ChemMedChem 24/2020)
He, Yingfang, Whitehead, David M., Briard, Emmanuelle, Numao, Shin, Mu, Linjing, Schibli, Roger, Ametamey, Simon M., Auberson, Yves P.
Published in ChemMedChem (15.12.2020)
Published in ChemMedChem (15.12.2020)
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Journal Article
Evaluation of 5H‐Thiazolopyrimidin‐5‐ones as Potential GluN2A PET Tracers
He, Yingfang, Whitehead, David M, Briard, Emmanuelle, Shin Numao, Mu, Linjing, Schibli, Roger, Ametamey, Simon M, Auberson, Yves P
Published in ChemMedChem (01.12.2020)
Published in ChemMedChem (01.12.2020)
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Journal Article
Evaluation of 5H‐Thiazolo[3,2‐α]pyrimidin‐5‐ones as Potential GluN2A PET Tracers
He, Yingfang, Whitehead, David M., Briard, Emmanuelle, Numao, Shin, Mu, Linjing, Schibli, Roger, Ametamey, Simon M., Auberson, Yves P.
Published in ChemMedChem (15.12.2020)
Published in ChemMedChem (15.12.2020)
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Journal Article
Discovery of LYS006, a Potent and Highly Selective Inhibitor of Leukotriene A 4 Hydrolase
Markert, Christian, Thoma, Gebhard, Srinivas, Honnappa, Bollbuck, Birgit, Lüönd, Rainer M, Miltz, Wolfgang, Wälchli, Rudolf, Wolf, Romain, Hinrichs, Jürgen, Bergsdorf, Christian, Azzaoui, Kamal, Penno, Carlos A, Klein, Kai, Wack, Nathalie, Jäger, Petra, Hasler, Franziska, Beerli, Christian, Loetscher, Pius, Dawson, Janet, Wieczorek, Grazyna, Numao, Shin, Littlewood-Evans, Amanda, Röhn, Till A
Published in Journal of medicinal chemistry (25.02.2021)
Published in Journal of medicinal chemistry (25.02.2021)
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Journal Article
Discovery of LYS006, a Potent and Highly Selective Inhibitor of Leukotriene A4 Hydrolase
Markert, Christian, Thoma, Gebhard, Srinivas, Honnappa, Bollbuck, Birgit, Lüönd, Rainer M, Miltz, Wolfgang, Wälchli, Rudolf, Wolf, Romain, Hinrichs, Jürgen, Bergsdorf, Christian, Azzaoui, Kamal, Penno, Carlos A, Klein, Kai, Wack, Nathalie, Jäger, Petra, Hasler, Franziska, Beerli, Christian, Loetscher, Pius, Dawson, Janet, Wieczorek, Grazyna, Numao, Shin, Littlewood-Evans, Amanda, Röhn, Till A
Published in Journal of medicinal chemistry (25.02.2021)
Published in Journal of medicinal chemistry (25.02.2021)
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Journal Article
Insights into the mechanism of Drosophila melanogaster Golgi alpha-mannosidase II through the structural analysis of covalent reaction intermediates
Numao, Shin, Kuntz, Douglas A, Withers, Stephen G, Rose, David R
Published in The Journal of biological chemistry (28.11.2003)
Published in The Journal of biological chemistry (28.11.2003)
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Journal Article
Evaluation of a Liquid Dispenser for Assay Development and Enzymology in 1536-Well Format
Butendeich, Heike, Pierret, Noëlle M., Numao, Shin
Published in Journal of Laboratory Automation (01.06.2013)
Published in Journal of Laboratory Automation (01.06.2013)
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Journal Article
Acarbose Rearrangement Mechanism Implied by the Kinetic and Structural Analysis of Human Pancreatic α-Amylase in Complex with Analogues and Their Elongated Counterparts
Li, Chunmin, Begum, Anjuman, Numao, Shin, Park, Kwan Hwa, Withers, Stephen G, Brayer, Gary D
Published in Biochemistry (Easton) (08.03.2005)
Published in Biochemistry (Easton) (08.03.2005)
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