Synthesis and Biological Evaluation of 1-Aryl-4,5-dihydro-1H-pyrazolo[3,4-d]pyrimidin-4-one Inhibitors of Cyclin-Dependent Kinases
Markwalder, Jay A, Arnone, Marc R, Benfield, Pamela A, Boisclair, Michael, Burton, Catherine R, Chang, Chong-Hwan, Cox, Sarah S, Czerniak, Philip M, Dean, Charity L, Doleniak, Deborah, Grafstrom, Robert, Harrison, Barbara A, Kaltenbach, Robert F, Nugiel, David A, Rossi, Karen A, Sherk, Susan R, Sisk, Lisa M, Stouten, Pieter, Trainor, George L, Worland, Peter, Seitz, Steven P
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Published in Journal of medicinal chemistry (18.11.2004)
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Structure-activity relationships (SAR) of some tetracyclic heterocycles related to the immunosuppressive agent brequinar sodium
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Published in Bioorganic & medicinal chemistry letters (03.02.1998)
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BENZOFURAN COMPOUNDS COMPOSITIONS AND METHODS FOR TREATMENT AND PROPHYLAXIS OF HEPATITIS C VIRAL INFECTIONS AND ASSOCIATED DISEASES
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Year of Publication 29.06.2005
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Year of Publication 29.06.2005
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Synthesis and Biological Evaluation of 1-Aryl-4,5-dihydro-1 H -pyrazolo[3,4- d ]pyrimidin-4-one Inhibitors of Cyclin-Dependent Kinases
Markwalder, Jay A., Arnone, Marc R., Benfield, Pamela A., Boisclair, Michael, Burton, Catherine R., Chang, Chong-Hwan, Cox, Sarah S., Czerniak, Philip M., Dean, Charity L., Doleniak, Deborah, Grafstrom, Robert, Harrison, Barbara A., Kaltenbach, Robert F., Nugiel, David A., Rossi, Karen A., Sherk, Susan R., Sisk, Lisa M., Stouten, Pieter, Trainor, George L., Worland, Peter, Seitz, Steven P.
Published in Journal of medicinal chemistry (01.11.2004)
Published in Journal of medicinal chemistry (01.11.2004)
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Heteroatom- and carbon-linked biphenyl analogs of Brequinar as immunosuppressive agents
Batt, Douglas G., Petraitis, Joseph J., Sherk, Susan R., Copeland, Robert A., Dowling, Randine L., Taylor, Tracy L., Jones, Elizabeth A., Magolda, Ronald L., Jaffee, Bruce D.
Published in Bioorganic & medicinal chemistry letters (07.07.1998)
Published in Bioorganic & medicinal chemistry letters (07.07.1998)
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Terphenyl cyclooxygenase-2 (COX-2) inhibitors: Optimization of the central ring and o-biphenyl analogs
Pinto, Donald J.P., Batt, Douglas G., Pitts, William J., Petraitis, Joseph J., Orwat, Michael J., Wang, Shuaige, Jetter, James W., Sherk, Susan R., Houghton, Gregory C., Copeland, Robert A., Covington, Maryanne B., Trzaskos, James M., Magolda, Ronald L.
Published in Bioorganic & medicinal chemistry letters (05.04.1999)
Published in Bioorganic & medicinal chemistry letters (05.04.1999)
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2,5-Diarylisothiazolone: novel inhibitors of cytokine-induced cartilage destruction
Wright, Stephen W., Petraitis, Joseph J., Freimark, Bruce, Giannaras, John V., Pratta, Michael A., Sherk, Susan R., Williams, Jean M., Magolda, Ronald L., Arner, Elizabeth C.
Published in Bioorganic & medicinal chemistry (01.06.1996)
Published in Bioorganic & medicinal chemistry (01.06.1996)
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Heteroaryl-Fused 2-Phenylisothiazolone Inhibitors of Cartilage Breakdown
Wright, Stephen W, Petraitis, Joseph J, Abelman, Matthew M, Batt, Douglas G, Bostrom, Lori L, Corbett, Ronald L, Decicco, Carl P, Di Meo, Susan V, Freimark, Bruce
Published in Journal of medicinal chemistry (01.09.1994)
Published in Journal of medicinal chemistry (01.09.1994)
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Metabolism resistant isothiazolone inhibitors of cartilage breakdown
Wright, Stephen W., Petraitis, Joseph J., Batt, Douglas G., Corbett, Ronald L., Di Meo, Susan V., Freimark, Bruce, Giannaras, John V., Orwat, Michael J., Pinto, Donald J., Pratta, Michael A., Sherk, Susan R., Stampfli, Herman F., Williams, Jean M., Magolda, Ronald L., Arner, Elizabeth C.
Published in Bioorganic & medicinal chemistry (01.03.1995)
Published in Bioorganic & medicinal chemistry (01.03.1995)
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Synthesis, chemical, and biological properties of vinylogous hydroxamic acids: dual inhibitors of 5-lipoxygenase and IL-1 biosynthesis
Wright, Stephen W, Harris, Richard R, Kerr, Janet S, Green, Alicia M, Pinto, Donald J, Bruin, Elaine M, Collins, Robert J, Dorow, Roberta L, Mantegna, Lisa R
Published in Journal of medicinal chemistry (01.10.1992)
Published in Journal of medicinal chemistry (01.10.1992)
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Vinylogous hydroxamic acids: 5-lipoxygenase inhibitors
Wright, Stephen W., Pinto, Donald J., Sherk, Susan R., Green, Alicia M., Magolda, Ronald L.
Published in Bioorganic & medicinal chemistry letters (01.09.1992)
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Inhibition of cartilage breakdown by isothiazolones
Wright, Stephen W., Petraitis, Joseph J., Abelman, Matthew M., Bostrom, Lori L., Corbett, Ronald L., Green, Alicia M., Kindt, Rachel M., Sherk, Susan R., Magolda, Ronald L.
Published in Bioorganic & medicinal chemistry letters (01.12.1993)
Published in Bioorganic & medicinal chemistry letters (01.12.1993)
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