Molecular dynamics simulation and in vitro evaluation of herb–drug interactions involving dietary polyphenols and CDK inhibitors in breast cancer chemotherapy
Patil, Prajakta H., Birangal, Sumit, Shenoy, G. Gautham, Rao, Mahadev, Kadari, Sandeep, Wankhede, Amit, Rastogi, Himanshu, Sharma, Tarun, Pinjari, Jakir, Puralae Channabasavaiah, Jagadish
Published in Phytotherapy research (01.10.2022)
Published in Phytotherapy research (01.10.2022)
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Journal Article
Preparation and characterization of co-amorphous Ritonavir–Indomethacin systems by solvent evaporation technique: Improved dissolution behavior and physical stability without evidence of intermolecular interactions
Dengale, Swapnil J., Ranjan, Om Prakash, Hussen, Syed Sajjad, Krishna, B.S.M., Musmade, Prashant B., Gautham Shenoy, G., Bhat, Krishnamurthy
Published in European journal of pharmaceutical sciences (01.10.2014)
Published in European journal of pharmaceutical sciences (01.10.2014)
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Journal Article
Fabrication, solid state characterization and bioavailability assessment of stable binary amorphous phases of Ritonavir with Quercetin
Dengale, Swapnil J., Hussen, Syed Sajjad, Krishna, B.S.M., Musmade, Prashant B., Gautham Shenoy, G., Bhat, Krishnamurthy
Published in European journal of pharmaceutics and biopharmaceutics (01.01.2015)
Published in European journal of pharmaceutics and biopharmaceutics (01.01.2015)
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Journal Article
Computational drug repurposing of Akt-1 allosteric inhibitors for non-small cell lung cancer
Baby, Krishnaprasad, Maity, Swastika, Mehta, Chetan Hasmukh, Nayak, Usha Y, Shenoy, Gautham G, Pai, Karkala Sreedhara Ranganath, Harikumar, Kuzhuvelil B, Nayak, Yogendra
Published in Scientific reports (16.05.2023)
Published in Scientific reports (16.05.2023)
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Journal Article
Design, synthesis, in silico and in vitro evaluation of novel diphenyl ether derivatives as potential antitubercular agents
Tiwari, Ashutosh Prasad, Sridhar, B., Boshoff, Helena I., Arora, Kriti, Gautham Shenoy, G., Vandana, K. E., Varadaraj Bhat, G.
Published in Molecular diversity (01.11.2020)
Published in Molecular diversity (01.11.2020)
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Journal Article
Molecular Insights into the Mechanism of Modulatory Effects of Proton Pump Inhibitors on P-glycoprotein Mediated Drug Transport of Palbociclib and Ribociclib
Desai, Mrunal Pradeep, Harish Patil, Prajakta, Vullendula, Sai Krishna Anand, Birangal, Sumit, Shenoy, G Gautham, Rao, Mahadev, Jayant Dengale, Swapnil, Bhat, Krishnamurthy, Puralae Channabasavaiah, Jagadish
Published in Current drug metabolism (01.01.2023)
Published in Current drug metabolism (01.01.2023)
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Synthesis, evaluation, molecular docking, and molecular dynamics studies of novel N‐(4‐[pyridin‐2‐yloxy]benzyl)arylamine derivatives as potential antitubercular agents
Verma, Ruchi, Boshoff, Helena I. M., Arora, Kriti, Bairy, Indira, Tiwari, Mradul, Varadaraj, Bhat G., Shenoy, G. Gautham
Published in Drug development research (01.05.2020)
Published in Drug development research (01.05.2020)
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Journal Article
Solvent Free Twin Screw Processed Silybin Nanophytophospholipid: In Silico, In Vitro and In Vivo Insights
Fernandes, Gasper, Pusuluri, Sai Lalitha Alekhya, Nikam, Ajinkya Nitin, Birangal, Sumit, Shenoy, Gautham G, Mutalik, Srinivas
Published in Pharmaceutics (06.12.2022)
Published in Pharmaceutics (06.12.2022)
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Journal Article
Histone Demethylase KDM5B as a Therapeutic Target for Cancer Therapy
Jose, Anmi, Shenoy, Gautham G., Sunil Rodrigues, Gabriel, Kumar, Naveena A. N., Munisamy, Murali, Thomas, Levin, Kolesar, Jill, Rai, Ganesha, Rao, Praveen P. N., Rao, Mahadev
Published in Cancers (01.08.2020)
Published in Cancers (01.08.2020)
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Journal Article
Large-Scale Stereoselective Synthesis of 1,3-Oxathiolane Nucleoside, Lamivudine, via ZrCl4‑Mediated N‑Glycosylation
Aher, Umesh P, Srivastava, Dhananjai, Jadhav, Harishchandra S, Singh, Girij P, B. S, Jayashree, Shenoy, Gautham G
Published in Organic process research & development (20.03.2020)
Published in Organic process research & development (20.03.2020)
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Journal Article
Novel isatin-indole derivatives as potential inhibitors of chorismate mutase (CM): their synthesis along with unexpected formation of 2-indolylmethylamino benzoate ester under Pd-Cu catalysis
Reddy, Gangireddy Sujeevan, Hossain, Kazi Amirul, Kumar, Jetta Sandeep, Thirupataiah, B, Edwin, Rebecca Kristina, Giliyaru, Varadaraj Bhat, Chandrashekhar Hariharapura, Raghu, Shenoy, G. Gautham, Misra, Parimal, Pal, Manojit
Published in RSC advances (02.01.2020)
Published in RSC advances (02.01.2020)
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Journal Article
Synthesis of 3-indolylmethyl substituted (pyrazolo/benzo)triazinone derivatives under Pd/Cu-catalysis: Identification of potent inhibitors of chorismate mutase (CM)
Reddy, Gangireddy Sujeevan, Snehalatha, Ampalam Venkata, Edwin, Rebecca Kristina, Hossain, Kazi Amirul, Giliyaru, Varadaraj Bhat, Hariharapura, Raghu Chandrashekhar, Gautham Shenoy, G., Misra, Parimal, Pal, Manojit
Published in Bioorganic chemistry (01.10.2019)
Published in Bioorganic chemistry (01.10.2019)
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Journal Article
An improved synthesis of latanoprost involving effective control on 15(S) diastereomer
Sasane, Sachin A., Bhise, Nandu B., Singh, Girij P., Joseph, Alex, Shenoy, Gautham G.
Published in Synthetic communications (17.09.2019)
Published in Synthetic communications (17.09.2019)
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Journal Article
Hyaluronic Acid-Protein Conjugate Modified Iron-Based MOFs (MIL-101 (Fe)) for Efficient Therapy of Neuroblastoma: Molecular Simulation, Stability and Toxicity Studies
Nikam, Ajinkya N, Pandey, Abhijeet, Nannuri, Shivanand H, Fernandes, Gasper, Kulkarni, Sanjay, Padya, Bharath Singh, Birangal, Sumit, Shenoy, Gautham G, George, Sajan D, Mutalik, Srinivas
Published in Crystals (Basel) (01.10.2022)
Published in Crystals (Basel) (01.10.2022)
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Journal Article
Molecular insights into Mmpl3 lead to the development of novel indole-2-carboxamides as antitubercular agents
Ray, Rajdeep, Birangal, Sumit Raosaheb, Fathima, Fajeelath, Boshoff, Helena I, Forbes, He Eun, Hariharapura, Raghu Chandrashekhar, Shenoy, G. Gautham
Published in Molecular systems design & engineering (06.06.2022)
Published in Molecular systems design & engineering (06.06.2022)
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Journal Article
Co-rotating twin screw process for continuous manufacturing of solid crystal suspension: A promising strategy to enhance the solubility, permeation and oral bioavailability of Carvedilol [version 3; peer review: 1 approved, 2 approved with reservations]
Navti, Prerana D., Fernandes, Gasper, Soman, Soji, Nikam, Ajinkya N., Kulkarni, Sanjay, Birangal, Sumit R, Dhas, Namdev, Shenoy, Gautham G., Rao, Vinay, Koteshwara, Kunnatur Balasundara, Mutalik, Srinivas
Published in F1000 research (01.01.2023)
Published in F1000 research (01.01.2023)
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Journal Article
Design, Synthesis and Evaluation of Antitubercular Activity of Novel 1,2,4-Triazoles Against MDR Strain of Mycobacterium tuberculosis
Ganesh Kumar, T. N. V., Gautham Shenoy, G., Kar, Sidhartha Sankar, Shenoy, Vishnu, Bairy, Indira
Published in Pharmaceutical chemistry journal (2018)
Published in Pharmaceutical chemistry journal (2018)
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Journal Article
A Comparative Study of 1D Descriptors Supported CoMFA and CoMSIA QSAR Models to Gain Novel Insights into 1,2,4-Triazoles Acting As Antitubercular Agents
Ray, Rajdeep, Shenoy, Gautham, Kumar Tummalapalli, N V Ganesh
Published in Current computer-aided drug design (01.01.2021)
Published in Current computer-aided drug design (01.01.2021)
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