Spiperone: Tritium labelling at high specific activity
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Published in Applied radiation and isotopes (01.05.2019)
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Discovery and structure–activity relationship of 2-phenyl-oxazole-4-carboxamide derivatives as potent apoptosis inducers
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Published in Bioorganic & medicinal chemistry letters (01.09.2006)
Published in Bioorganic & medicinal chemistry letters (01.09.2006)
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Highly potent non-peptidic inhibitors of the HCV NS3/NS4A serine protease
Sperandio, David, Gangloff, Anthony R., Litvak, Joane, Goldsmith, Richard, Hataye, Jason M., Wang, Vivian R., Shelton, Emma J., Elrod, Kyle, Janc, James W., Clark, James M., Rice, Ken, Weinheimer, Steve, Yeung, Kap-Sun, Meanwell, Nicholas A., Hernandez, Dennis, Staab, Andrew J., Venables, Brian L., Spencer, Jeffrey R.
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
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Identification of metabolites of the tryptase inhibitor CRA-9249: Observation of a metabolite derived from an unexpected hydroxylation pathway
Yu, Walter, Dener, Jeffrey M., Dickman, Daniel A., Grothaus, Paul, Ling, Yun, Liu, Liang, Havel, Chris, Malesky, Kimberly, Mahajan, Tania, O’Brian, Colin, Shelton, Emma J., Sperandio, David, Tong, Zhiwei, Yee, Robert, Mordenti, Joyce J.
Published in Bioorganic & medicinal chemistry letters (01.08.2006)
Published in Bioorganic & medicinal chemistry letters (01.08.2006)
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Electrophilic addition of benzeneselenenyl chloride to hydroxyalkynes
Filer, Crist N, Ahern, David, Fazio, Robert, Shelton, Emma J
Published in Journal of organic chemistry (01.03.1980)
Published in Journal of organic chemistry (01.03.1980)
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Selective Inhibition of Mammalian Lanosterol 14.alpha.-Demethylase by RS-21607 in vitro and in vivo
Swinney, David C, So, On-Yee, Watson, David M, Berry, Pamela W, Webb, Austin S, Kertesz, Denis J, Shelton, Emma J, Walker, Keith A. M, Burton, Pamela M
Published in Biochemistry (Easton) (01.04.1994)
Published in Biochemistry (Easton) (01.04.1994)
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Development of a scalable synthesis of a nonbasic inhibitor of the serine protease tryptase
Dener, Jeffrey M., O’Bryan, Colin, Yee, Robert, Shelton, Emma J., Sperandio, David, Mahajan, Tania, Palmer, James T., Spencer, Jeffrey R., Tong, Zhiwei
Published in Tetrahedron letters (03.07.2006)
Published in Tetrahedron letters (03.07.2006)
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Selective inhibition of mammalian lanosterol 14α-demethylase by RS-21607 in vitro and in vivo
SWINNEY, D. C, ON-YEE SO, WATSON, D. M, BERRY, P. W, WEBB, A. S, KERTESZ, D. J, SHELTON, E. J, BURTON, P. M, WALKER, K. A. M
Published in Biochemistry (Easton) (19.04.1994)
Published in Biochemistry (Easton) (19.04.1994)
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INHIBITORS OF TRYPTASE
LIU, WEILI, YEE, ROBERT, WINSLOW-LOHMAN, JULIA, HIRSCHBEIN, BERNARD, SPENCER, JEFFREY, R, LITVAK, JOANE, SENDZIK, MARTIN, TAI, VINCENT, W-F, LEE, CHANG SUN, SHELTON, EMMA, J, SPERANDIO, DAVID
Year of Publication 01.02.2007
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Year of Publication 01.02.2007
Patent
INHIBITORS OF TRYPTASE
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Year of Publication 17.08.2006
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Year of Publication 17.08.2006
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SYNTHESIS OF SPECIFICALLY LABELED PEPTIDES
PARNES, H, SHELTON, EJ
Published in International journal of peptide and protein research (01.03.1986)
Published in International journal of peptide and protein research (01.03.1986)
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Novel phenyl derivatives as inducers of apoptosis
CAI SUI XIONG, CEBON BEN, LITVAK JOANE, YEE ROBERT M, SPRENGELER PAUL A, SHELTON EMMA J, SPENCER JEFFREY R, PARARAJASINGHAM KEITH, SPERANDIO DAVID, TAI VINCENT W.-F
Year of Publication 03.02.2005
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Year of Publication 03.02.2005
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Novel compounds and compositions for treating hepatitis c infections
JASON M. HATAYE, VIVIAN R. WANG, JEFFREY R. SPENCER, KENNETH RICE, EMMA J. SHELTON
Year of Publication 26.04.2000
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Year of Publication 26.04.2000
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NOVEL COMPOUNDS AND COMPOSITIONS FOR TREATING HEPATITIS C INFECTIONS
WANG, VIVIAN, R, SPENCER, JEFFREY, R, RICE, KENNETH, HATAYE, JASON, M, SHELTON, EMMA, J
Year of Publication 13.04.2000
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Year of Publication 13.04.2000
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NOVEL PHENYL DERIVATIVES AS INDUCERS OF APOPTOSIS
TAI, VINCENT, W.-F, CAI, SUI, XIONG, SPRENGELER, PAUL, A, YEE, ROBERT, M, SPENCER, JEFFREY, R, LITVAK, JOANE, CEBON, BEN, SHELTON, EMMA, J, PARARAJASINGHAM, KEITH, SPERANDIO, DAVID
Year of Publication 25.03.2004
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Year of Publication 25.03.2004
Patent
Synthesis of 14C-labelled peptides by asymmetric reduction of dehydroamino acids
Parnes, H, Shelton, E J, Huang, G T
Published in International journal of peptide and protein research (01.10.1986)
Published in International journal of peptide and protein research (01.10.1986)
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