The Phosphoinositide-Specific Phospholipase C Inhibitor U73122 (1-(6-((17β-3-Methoxyestra-1,3,5(10)-trien-17-yl)amino)hexyl)-1H-pyrrole-2,5-dione) Spontaneously Forms Conjugates with Common Components of Cell Culture Medium
Wilsher, Nicola E, Court, Will J, Ruddle, Ruth, Newbatt, Yvette M, Aherne, Wynne, Sheldrake, Peter W, Jones, Neil P, Katan, Matilda, Eccles, Suzanne A, Raynaud, Florence I
Published in Drug metabolism and disposition (01.07.2007)
Published in Drug metabolism and disposition (01.07.2007)
Get full text
Journal Article
Optimization of Imidazo[4,5‑b]pyridine-Based Kinase Inhibitors: Identification of a Dual FLT3/Aurora Kinase Inhibitor as an Orally Bioavailable Preclinical Development Candidate for the Treatment of Acute Myeloid Leukemia
Bavetsias, Vassilios, Crumpler, Simon, Sun, Chongbo, Avery, Sian, Atrash, Butrus, Faisal, Amir, Moore, Andrew S, Kosmopoulou, Magda, Brown, Nathan, Sheldrake, Peter W, Bush, Katherine, Henley, Alan, Box, Gary, Valenti, Melanie, de Haven Brandon, Alexis, Raynaud, Florence I, Workman, Paul, Eccles, Suzanne A, Bayliss, Richard, Linardopoulos, Spiros, Blagg, Julian
Published in Journal of medicinal chemistry (25.10.2012)
Published in Journal of medicinal chemistry (25.10.2012)
Get full text
Journal Article
Conformation Analyses, Dynamic Behavior and Amide Bond Distortions of Medium-sized Heterocycles. 1. Partially and Fully Reduced 1-Benzazepines
Qadir, Maryiam, Cobb, Jonathan, Sheldrake, Peter W, Whittall, Neil, White, Andrew J. P, Hii, King Kuok (Mimi), Horton, Peter N, Hursthouse, Michael B
Published in Journal of organic chemistry (04.03.2005)
Published in Journal of organic chemistry (04.03.2005)
Get full text
Journal Article
Conformation Analyses, Dynamic Behavior, and Amide Bond Distortions of Medium-sized Heterocycles. 2. Partially and Fully Reduced 1-Benzazocines, Benzazonines, and Benzazecines
Qadir, Maryiam, Cobb, Jonathan, Sheldrake, Peter W, Whittall, Neil, White, Andrew J. P, Hii, King Kuok (Mimi), Horton, Peter N, Hursthouse, Michael B
Published in Journal of organic chemistry (04.03.2005)
Published in Journal of organic chemistry (04.03.2005)
Get full text
Journal Article
Total synthesis of erythromycins. 4. Total synthesis of erythronolide B
Corey, E. J, Kim, Sunggak, Yoo, Sung-Eun, Nicolaou, K. C, Melvin, Lawrence S, Brunelle, Daniel J, Falck, J. R, Trybulski, Eugene J, Lett, Robert, Sheldrake, Peter W
Published in Journal of the American Chemical Society (01.07.1978)
Published in Journal of the American Chemical Society (01.07.1978)
Get full text
Journal Article
Total synthesis of erythromycins. 3. Stereoselective routes to intermediates corresponding to C(1) to C(9) and C(10) to C(13) fragments of erythronolide B
Corey, E. J, Trybulski, Eugene J, Melvin, Lawrence S, Nicolaou, K. C, Secrist, John A, Lett, Robert, Sheldrake, Peter W, Falck, J. R, Brunelle, Daniel J
Published in Journal of the American Chemical Society (01.07.1978)
Published in Journal of the American Chemical Society (01.07.1978)
Get full text
Journal Article
Preparation of 5-Hydroxy-2-iodopyridine: A Refutation of Earlier Reports
Sheldrake, Peter W, Powling, Laurence C, Slaich, Pritpal K
Published in Journal of organic chemistry (02.05.1997)
Published in Journal of organic chemistry (02.05.1997)
Get full text
Journal Article
Chapter 6. Heterocyclic compounds
Sheldrake, Peter W.
Published in Annual reports on the progress of chemistry. Section B. Organic chemistry (1996)
Published in Annual reports on the progress of chemistry. Section B. Organic chemistry (1996)
Get full text
Journal Article
Chapter 6. Heterocyclic compounds
Sheldrake, Peter W.
Published in Annual reports on the progress of chemistry. Section B. Organic chemistry (1995)
Published in Annual reports on the progress of chemistry. Section B. Organic chemistry (1995)
Get full text
Journal Article
Biosynthesis. Part 30.1 Colchicine: studies on the ring expansion step focusing on the fate of the hydrogens at C-4 of autumnaline
Sheldrake, Peter W., Suckling, Keith E., Woodhouse, Robert N., Murtagh, Amanda J., Herbert, Richard B., Barker, Alan C., Staunton, James, Battersby, Alan R.
Published in Journal of the Chemical Society, Perkin Transactions 1 (1998)
Published in Journal of the Chemical Society, Perkin Transactions 1 (1998)
Get full text
Journal Article
Synthesis of 2-substituted 1-benzyl-2,3,4,5-tetrahydro-1-benzazepines by palladium catalysis. Observation of a competitive β-hydride elimination pathway
Qadir, Maryiam, Priestley, Rachael E., Rising, Thomas W.D.F., Gelbrich, Thomas, Coles, Simon J., Hursthouse, Michael B., Sheldrake, Peter W., Whittall, Neil, Hii, K.K.(Mimi)
Published in Tetrahedron letters (28.04.2003)
Published in Tetrahedron letters (28.04.2003)
Get full text
Journal Article
The phosphoinositide-specific phospholipase C inhibitor U73122 1 -6 - (17β-3-methoxyestra-1,3,5 (10 ) -trien-17-yl)aminohexyl-1H-pyrrole-2,5-dione spontaneously forms conjugates with common components of cell culture medium
WILSHER, Nicola E, COURT, Will J, RUDDLE, Ruth, NEWBATT, Yvette M, AHERNE, Wynne, SHELDRAKE, Peter W, JONES, Neil P, KATAN, Matilda, ECCLES, Suzanne A, RAYNAUD, Florence I
Published in Drug metabolism and disposition (2007)
Get full text
Published in Drug metabolism and disposition (2007)
Journal Article
UNEXPECTED SYNTHESIS OF A 1H-PYRROLO[2,3-E]-1,2,4-TRIAZINE
WELLS, AS, SHELDRAKE, PW, LANTOS, EGGLESTON, DS
Published in Journal of the Chemical Society, Perkin Transactions 1 (1991)
Published in Journal of the Chemical Society, Perkin Transactions 1 (1991)
Get full text
Journal Article
An efficient method for the synthesis of substituted TosMIC precursors
Sisko, Joseph, Mellinger, Mark, Sheldrake, Peter W., Baine, Neil H.
Published in Tetrahedron letters (04.11.1996)
Published in Tetrahedron letters (04.11.1996)
Get full text
Journal Article
Studies of enzyme-mediated reactions. Part VII. Stereospecific syntheses of tritium-labelled (2R)- and (2S)-dopamines: stereochemical course of hydroxylation of dopamine by dopamine beta-hydroxylase (E.C. 1.14.17.1)
Battersby, A R, Sheldrake, P W, Staunton, J, Williams, D C
Published in J. Chem. Soc., Perkin Trans. 1 (1976)
Published in J. Chem. Soc., Perkin Trans. 1 (1976)
Get full text
Journal Article