Alteration of Lymphocyte Trafficking by Sphingosine-1-Phosphate Receptor Agonists
Mandala, Suzanne, Hajdu, Richard, Bergstrom, James, Quackenbush, Elizabeth, Xie, Jenny, Milligan, James, Thornton, Rosemary, Shei, Gan-Ju, Card, Deborah, Keohane, CarolAnn, Rosenbach, Mark, Hale, Jeffrey, Lynch, Christopher L., Rupprecht, Kathleen, Parsons, William, Rosen, Hugh
Published in Science (American Association for the Advancement of Science) (12.04.2002)
Published in Science (American Association for the Advancement of Science) (12.04.2002)
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Characterization of a Novel Sphingosine 1-Phosphate Receptor, Edg-8
Im, Dong-Soon, Heise, Christopher E., Ancellin, Nicolas, O'Dowd, Brian F., Shei, Gan-ju, Heavens, Robert P., Rigby, Michael R., Hla, Timothy, Mandala, Suzanne, McAllister, George, George, Susan R., Lynch, Kevin R.
Published in The Journal of biological chemistry (12.05.2000)
Published in The Journal of biological chemistry (12.05.2000)
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Potent S1P receptor agonists replicate the pharmacologic actions of the novel immune modulator FTY720
Hale, Jeffrey J., Neway, William, Mills, Sander G., Hajdu, Richard, Ann Keohane, Carol, Rosenbach, Mark, Milligan, James, Shei, Gan-Ju, Chrebet, Gary, Bergstrom, James, Card, Deborah, Koo, Gloria C., Koprak, Sam L., Jackson, Jesse J., Rosen, Hugh, Mandala, Suzanne
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
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Synthesis, stereochemical determination and biochemical characterization of the enantiomeric phosphate esters of the novel immunosuppressive agent FTY720
Hale, Jeffrey J., Yan, Lin, Neway, William E., Hajdu, Richard, Bergstrom, James D., Milligan, James A., Shei, Gan-Ju, Chrebet, Gary L., Thornton, Rosemary A., Card, Deborah, Rosenbach, Mark, HughRosen, Mandala, Suzanne
Published in Bioorganic & medicinal chemistry (15.09.2004)
Published in Bioorganic & medicinal chemistry (15.09.2004)
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Phytosphingosine 1-phosphate: a high affinity ligand for the S1P4/Edg-6 receptor
Rios Candelore, Mari, Wright, Michael J, Tota, Laurie M, Milligan, James, Shei, Gan-ju, Bergstrom, James D, Mandala, Suzanne M
Published in Biochemical and biophysical research communications (01.09.2002)
Published in Biochemical and biophysical research communications (01.09.2002)
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Discovery of Potent 3,5-Diphenyl-1,2,4-oxadiazole Sphingosine-1-phosphate-1 (S1P1) Receptor Agonists with Exceptional Selectivity against S1P2 and S1P3
Li, Zhen, Chen, Weirong, Hale, Jeffrey J, Lynch, Christopher L, Mills, Sander G, Hajdu, Richard, Keohane, Carol Ann, Rosenbach, Mark J, Milligan, James A, Shei, Gan-Ju, Chrebet, Gary, Parent, Stephen A, Bergstrom, James, Card, Deborah, Forrest, Michael, Quackenbush, Elizabeth J, Wickham, L. Alexandra, Vargas, Hugo, Evans, Rose M, Rosen, Hugh, Mandala, Suzanne
Published in Journal of medicinal chemistry (06.10.2005)
Published in Journal of medicinal chemistry (06.10.2005)
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A Rational Utilization of High-Throughput Screening Affords Selective, Orally Bioavailable 1-Benzyl-3-carboxyazetidine Sphingosine-1-phosphate-1 Receptor Agonists
Hale, Jeffrey J, Lynch, Christopher L, Neway, William, Mills, Sander G, Hajdu, Richard, Keohane, Carol Ann, Rosenbach, Mark J, Milligan, James A, Shei, Gan-Ju, Parent, Stephen A, Chrebet, Gary, Bergstrom, James, Card, Deborah, Ferrer, Marc, Hodder, Peter, Strulovici, Berta, Rosen, Hugh, Mandala, Suzanne
Published in Journal of medicinal chemistry (30.12.2004)
Published in Journal of medicinal chemistry (30.12.2004)
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Selecting against S1P3 enhances the acute cardiovascular tolerability of 3-(N-benzyl)aminopropylphosphonic acid S1P receptor agonists
Hale, Jeffrey J., Doherty, George, Toth, Leslie, Mills, Sander G., Hajdu, Richard, Ann Keohane, Carol, Rosenbach, Mark, Milligan, James, Shei, Gan-Ju, Chrebet, Gary, Bergstrom, James, Card, Deborah, Forrest, Michael, Sun, Shu-Yu, West, Sarah, Xie, Huijuan, Nomura, Naomi, Rosen, Hugh, Mandala, Suzanne
Published in Bioorganic & medicinal chemistry letters (05.07.2004)
Published in Bioorganic & medicinal chemistry letters (05.07.2004)
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SAR studies of 3-arylpropionic acids as potent and selective agonists of sphingosine-1-phosphate receptor-1 (S1P 1) with enhanced pharmacokinetic properties
Yan, Lin, Huo, Pei, Hale, Jeffrey J., Mills, Sander G., Hajdu, Richard, Keohane, Carol A., Rosenbach, Mark J., Milligan, James A., Shei, Gan-Ju, Chrebet, Gary, Bergstrom, James, Card, Deborah, Mandala, Suzanne M.
Published in Bioorganic & medicinal chemistry letters (01.02.2007)
Published in Bioorganic & medicinal chemistry letters (01.02.2007)
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Discovery of 3-arylpropionic acids as potent agonists of sphingosine-1-phosphate receptor-1 (S1P 1) with high selectivity against all other known S1P receptor subtypes
Yan, Lin, Huo, Pei, Doherty, George, Toth, Lesile, Hale, Jeffrey J., Mills, Sander G., Hajdu, Richard, Keohane, Carol A., Rosenbach, Mark J., Milligan, James A., Shei, Gan-Ju, Chrebet, Gary, Bergstrom, James, Card, Deborah, Quackenbush, Elizabeth, Wickham, Alexandra, Mandala, Suzanne M.
Published in Bioorganic & medicinal chemistry letters (15.07.2006)
Published in Bioorganic & medicinal chemistry letters (15.07.2006)
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2-Aryl(pyrrolidin-4-yl)acetic acids are potent agonists of sphingosine-1-phosphate (S1P) receptors
Yan, Lin, Budhu, Richard, Huo, Pei, Lynch, Christopher L., Hale, Jeffrey J., Mills, Sander G., Hajdu, Richard, Keohane, Carol A., Rosenbach, Mark J., Milligan, James A., Shei, Gan-Ju, Chrebet, Gary, Bergstrom, James, Card, Deborah, Mandala, Suzanne M.
Published in Bioorganic & medicinal chemistry letters (01.07.2006)
Published in Bioorganic & medicinal chemistry letters (01.07.2006)
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2,5-Disubstituted pyrrolidine carboxylates as potent, orally active sphingosine-1-phosphate (S1P) receptor agonists
Colandrea, Vincent J., Legiec, Irene E., Huo, Pei, Yan, Lin, Hale, Jeffrey J., Mills, Sander G., Bergstrom, James, Card, Deborah, Chebret, Gary, Hajdu, Richard, Keohane, Carol Ann, Milligan, James A., Rosenbach, Mark J., Shei, Gan-Ju, Mandala, Suzanne M.
Published in Bioorganic & medicinal chemistry letters (01.06.2006)
Published in Bioorganic & medicinal chemistry letters (01.06.2006)
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Design and synthesis of conformationally constrained 3-( N-alkylamino)propylphosphonic acids as potent agonists of sphingosine-1-phosphate (S1P) receptors
Yan, Lin, Hale, Jeffrey J., Lynch, Christopher L., Budhu, Richard, Gentry, Amy, Mills, Sander G., Hajdu, Richard, Keohane, Carol Ann, Rosenbach, Mark J., Milligan, James A., Shei, Gan-Ju, Chrebet, Gary, Bergstrom, James, Card, Deborah, Rosen, Hugh, Mandala, Suzanne M.
Published in Bioorganic & medicinal chemistry letters (04.10.2004)
Published in Bioorganic & medicinal chemistry letters (04.10.2004)
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The discovery of 3-(N-alkyl)aminopropylphosphonic acids as potent S1P receptor agonists
Hale, Jeffrey J., Doherty, George, Toth, Leslie, Li, Zhen, Mills, Sander G., Hajdu, Richard, Ann Keohane, Carol, Rosenbach, Mark, Milligan, James, Shei, Gan-Ju, Chrebet, Gary, Bergstrom, James, Card, Deborah, Rosen, Hugh, Mandala, Suzanne
Published in Bioorganic & medicinal chemistry letters (05.07.2004)
Published in Bioorganic & medicinal chemistry letters (05.07.2004)
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Mutations in the HML E silencer of Saccharomyces cerevisiae yield metastable inheritance of transcriptional repression
MAHONEY, D. J, MARQUARDT, R, SHEI, G.-J, ROSE, A. B, BROACH, J. R
Published in Genes & development (01.04.1991)
Published in Genes & development (01.04.1991)
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Phytosphingosine 1-phosphate: a high affinity ligand for the S1P(4)/Edg-6 receptor
Candelore, Mari Rios, Wright, Michael J, Tota, Laurie M, Milligan, James, Shei, Gan-ju, Bergstrom, James D, Mandala, Suzanne M
Published in Biochemical and biophysical research communications (27.09.2002)
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Published in Biochemical and biophysical research communications (27.09.2002)
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Development of a cyclic adenosine monophosphate assay for Gi-coupled G protein-coupled receptors by utilizing the endogenous calcitonin activity in Chinese hamster ovary cells
Wang, Yuren, Kong, Yan, Shei, Gan Ju, Kang, Liya, Cvijic, Mary Ellen
Published in Assay and drug development technologies (01.10.2011)
Published in Assay and drug development technologies (01.10.2011)
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Discovery of 3-arylpropionic acids as potent agonists of sphingosine-1-phosphate receptor-1 (S1P1) with high selectivity against all other known S1Preceptor subtypes
LIN YAN, PEI HUO, SHEI, Gan-Ju, CHREBET, Gary, BERGSTROM, James, CARD, Deborah, QUACKENBUSH, Elizabeth, WICKHAM, Alexandra, MANDALA, Suzanne M, DOHERTY, George, TOTH, Lesile, HALE, Jeffrey J, MILLS, Sander G, HAJDU, Richard, KEOHANE, Carol A, ROSENBACH, Mark J, MILLIGAN, James A
Published in Bioorganic & medicinal chemistry letters (2006)
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Published in Bioorganic & medicinal chemistry letters (2006)
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