Carbonic Anhydrase IX Inhibitors as Candidates for Combination Therapy of Solid Tumors
Kalinin, Stanislav, Malkova, Anna, Sharonova, Tatiana, Sharoyko, Vladimir, Bunev, Alexander, Supuran, Claudiu T, Krasavin, Mikhail
Published in International journal of molecular sciences (14.12.2021)
Published in International journal of molecular sciences (14.12.2021)
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Inhibitory activity against carbonic anhydrase IX and XII as a candidate selection criterion in the development of new anticancer agents
Krasavin, Mikhail, Kalinin, Stanislav, Sharonova, Tatiana, Supuran, Claudiu T
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
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Combining carbonic anhydrase and thioredoxin reductase inhibitory motifs within a single molecule dramatically increases its cytotoxicity
Krasavin, Mikhail, Sharonova, Tatiana, Sharoyko, Vladimir, Zhukovsky, Daniil, Kalinin, Stanislav, Žalubovskis, Raivis, Tennikova, Tatiana, Supuran, Claudiu T.
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
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Journal Article
Diversely substituted sulfamides for fragment-based drug discovery of carbonic anhydrase inhibitors: synthesis and inhibitory profile
Sharonova, Tatiana, Zhmurov, Petr, Kalinin, Stanislav, Nocentini, Alessio, Angeli, Andrea, Ferraroni, Marta, Korsakov, Mikhail, Supuran, Claudiu T, Krasavin, Mikhail
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2022)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2022)
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Synthesis, Structure, and Antiproliferative Action of 2-Pyridyl Urea-Based Cu(II) Complexes
Geyl, Kirill K, Baykov, Sergey V, Kalinin, Stanislav A, Bunev, Alexandr S, Troshina, Marina A, Sharonova, Tatiana V, Skripkin, Mikhail Yu, Kasatkina, Svetlana O, Presnukhina, Sofia I, Shetnev, Anton A, Krasavin, Mikhail Yu, Boyarskiy, Vadim P
Published in Biomedicines (16.02.2022)
Published in Biomedicines (16.02.2022)
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Investigation of 3-sulfamoyl coumarins against cancer-related IX and XII isoforms of human carbonic anhydrase as well as cancer cells leads to the discovery of 2-oxo-2H-benzo[h]chromene-3-sulfonamide – A new caspase-activating proapoptotic agent
Dar'in, Dmitry, Kantin, Grigory, Kalinin, Stanislav, Sharonova, Tatiana, Bunev, Alexander, Ostapenko, Gennady I., Nocentini, Alessio, Sharoyko, Vladimir, Supuran, Claudiu T., Krasavin, Mikhail
Published in European journal of medicinal chemistry (15.10.2021)
Published in European journal of medicinal chemistry (15.10.2021)
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Corrigendum to “Investigation of 3-sulfamoyl coumarins against cancer-related IX and XII isoforms of human carbonic anhydrase as well as cancer cells leads to the discovery of 2-oxo-2H-benzo[h]chromene-3-sulfonamide – A new caspase-activating proapoptotic agent” [J. Med. Chem. 222 (2021) 113589]
Dar'in, Dmitry, Kantin, Grigory, Kalinin, Stanislav, Sharonova, Tatiana, Bunev, Alexander, Ostapenko, Gennady I., Nocentini, Alessio, Sharoyko, Vladimir, Supuran, Claudiu T., Krasavin, Mikhail
Published in European journal of medicinal chemistry (05.12.2021)
Published in European journal of medicinal chemistry (05.12.2021)
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Journal Article
(E)-3-Arylidene-4-diazopyrrolidine-2,5-diones conveniently elaborated into cytotoxic compounds bearing primary sulfonamide and Michael acceptor moieties
Paramonova, Polina, Sharonova, Tatiana, Kalinin, Stanislav, Chupakhin, Evgeny, Bunev, Alexander, Krasavin, Mikhail
Published in Mendeleev communications (01.03.2022)
Published in Mendeleev communications (01.03.2022)
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Insertion of metal carbenes into the anilinic N–H bond of unprotected aminobenzenesulfonamides delivers low nanomolar inhibitors of human carbonic anhydrase IX and XII isoforms
Sharonova, Tatiana, Paramonova, Polina, Kalinin, Stanislav, Bunev, Alexander, Gasanov, Rovshan Е., Nocentini, Alessio, Sharoyko, Vladimir, Tennikova, Tatiana B., Dar’in, Dmitry, Supuran, Claudiu T., Krasavin, Mikhail
Published in European journal of medicinal chemistry (05.06.2021)
Published in European journal of medicinal chemistry (05.06.2021)
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Journal Article
Diversely substituted sulfamides for fragment-based drug discovery of carbonic anhydrase inhibitors: synthesis and inhibitory profile
Sharonova, Tatiana, Zhmurov, Petr, Kalinin, Stanislav, Nocentini, Alessio, Angeli, Andrea, Ferraroni, Marta, Korsakov, Mikhail, Supuran, Claudiu T., Krasavin, Mikhail
Published in Journal of Enzyme Inhibition and Medicinal Chemistry (31.12.2022)
Published in Journal of Enzyme Inhibition and Medicinal Chemistry (31.12.2022)
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Inhibitory activity against carbonic anhydrase IX and XII as a candidate selection criterion in the development of new anticancer agents
Krasavin, Mikhail, Kalinin, Stanislav, Sharonova, Tatiana, Supuran, Claudiu T.
Published in Journal of Enzyme Inhibition and Medicinal Chemistry (01.01.2020)
Published in Journal of Enzyme Inhibition and Medicinal Chemistry (01.01.2020)
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