Homo-PROTAC mediated suicide of MDM2 to treat non-small cell lung cancer
He, Shipeng, Ma, Junhui, Fang, Yuxin, Liu, Ying, Wu, Shanchao, Dong, Guoqiang, Wang, Wei, Sheng, Chunquan
Published in Acta pharmaceutica Sinica. B (01.06.2021)
Published in Acta pharmaceutica Sinica. B (01.06.2021)
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Journal Article
One-Pot Synthesis of Deuterated Aldehydes from Arylmethyl Halides
Li, Xiangmin, Wu, Shanchao, Chen, Shuqiang, Lai, Zengwei, Luo, Hai-Bin, Sheng, Chunquan
Published in Organic letters (06.04.2018)
Published in Organic letters (06.04.2018)
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Journal Article
A novel route for the synthesis of androgen receptor antagonist enzalutamide
Meng, Xiangguo, Bi, Siju, Jin, Shixin, Wu, Kai, Wu, Shanchao, Shao, Lei, Bonnet, Pierre-Antoine, Sheng, Chunquan
Published in Chinese chemical letters (01.06.2023)
Published in Chinese chemical letters (01.06.2023)
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Journal Article
Tackling Fungal Resistance by Biofilm Inhibitors
Wu, Shanchao, Wang, Yan, Liu, Na, Dong, Guoqiang, Sheng, Chunquan
Published in Journal of medicinal chemistry (23.03.2017)
Published in Journal of medicinal chemistry (23.03.2017)
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Journal Article
Potent Dual BET/HDAC Inhibitors for Efficient Treatment of Pancreatic Cancer
He, Shipeng, Dong, Guoqiang, Li, Yu, Wu, Shanchao, Wang, Wei, Sheng, Chunquan
Published in Angewandte Chemie International Edition (17.02.2020)
Published in Angewandte Chemie International Edition (17.02.2020)
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Journal Article
Small Molecules Simultaneously Inhibiting p53-Murine Double Minute 2 (MDM2) Interaction and Histone Deacetylases (HDACs): Discovery of Novel Multitargeting Antitumor Agents
He, Shipeng, Dong, Guoqiang, Wu, Shanchao, Fang, Kun, Miao, Zhenyuan, Wang, Wei, Sheng, Chunquan
Published in Journal of medicinal chemistry (23.08.2018)
Published in Journal of medicinal chemistry (23.08.2018)
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Journal Article
Small Molecules Simultaneously Inhibiting p53-Murine Double Minute 2 (MDM2) Interaction and Histone Deacetylases (HDACs): Discovery of Novel Multitargeting Antitumor Agents
He, Shipeng, Dong, Guoqiang, Wu, Shanchao, Fang, Kun, Miao, Zhenyuan, Wang, Wei, Sheng, Chunquan
Published in Journal of medicinal chemistry (23.08.2018)
Published in Journal of medicinal chemistry (23.08.2018)
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Journal Article
Evodiamine-Inspired Topoisomerase-Histone Deacetylase Dual Inhibitors: Novel Orally Active Antitumor Agents for Leukemia Therapy
Wu, Shanchao, Huang, Yahui, Wang, Ting, Li, Keliang, Lu, Junjie, Huang, Min, Dong, Guoqiang, Sheng, Chunquan
Published in Journal of medicinal chemistry (24.03.2022)
Published in Journal of medicinal chemistry (24.03.2022)
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Journal Article
Open innovation strategy in the process of technological capability development: Conceptual framework aspect
Shanchao Wu, Jun Jin, Jin Chen, Vanhaverbeke, W.
Published in 2009 16th International Conference on Industrial Engineering and Engineering Management (01.10.2009)
Published in 2009 16th International Conference on Industrial Engineering and Engineering Management (01.10.2009)
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Conference Proceeding
Ispinesib as an Effective Warhead for the Design of Autophagosome-Tethering Chimeras: Discovery of Potent Degraders of Nicotinamide Phosphoribosyltransferase (NAMPT)
Dong, Guoqiang, Wu, Ying, Cheng, Junfei, Chen, Long, Liu, Rui, Ding, Yu, Wu, Shanchao, Ma, Junhui, Sheng, Chunquan
Published in Journal of medicinal chemistry (09.06.2022)
Published in Journal of medicinal chemistry (09.06.2022)
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Journal Article
Scaffold Hopping of Natural Product Evodiamine: Discovery of a Novel Antitumor Scaffold with Excellent Potency against Colon Cancer
Wang, Lei, Fang, Kun, Cheng, Junfei, Li, Yu, Huang, Yahui, Chen, Shuqiang, Dong, Guoqiang, Wu, Shanchao, Sheng, Chunquan
Published in Journal of medicinal chemistry (23.01.2020)
Published in Journal of medicinal chemistry (23.01.2020)
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Journal Article
Meeting Organocatalysis with Drug Discovery: Asymmetric Synthesis of 3,3′-Spirooxindoles Fused with Tetrahydrothiopyrans as Novel p53-MDM2 Inhibitors
Wang, Shengzheng, Jiang, Yan, Wu, Shanchao, Dong, Guoqiang, Miao, Zhenyuan, Zhang, Wannian, Sheng, Chunquan
Published in Organic letters (04.03.2016)
Published in Organic letters (04.03.2016)
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Journal Article
Discovery of Indolo3,2-cisoquinoline Derivatives as Novel Top1/2 Dual Inhibitors with Orally Efficacious Antitumor Activity and Low Toxicity
Wang, Bichuan, Wu, Shanchao, Jia, Shuolei, Ruan, Xiuqin, Sheng, Chunquan, Zhou, Qingfa
Published in Journal of medicinal chemistry (22.08.2024)
Published in Journal of medicinal chemistry (22.08.2024)
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Journal Article
Discovery of Indolo[3,2‑c]isoquinoline Derivatives as Novel Top1/2 Dual Inhibitors with Orally Efficacious Antitumor Activity and Low Toxicity
Wang, Bichuan, Wu, Shanchao, Jia, Shuolei, Ruan, Xiuqin, Sheng, Chunquan, Zhou, Qingfa
Published in Journal of medicinal chemistry (22.08.2024)
Published in Journal of medicinal chemistry (22.08.2024)
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Journal Article
Water-soluble derivatives of evodiamine: Discovery of evodiamine-10-phosphate as an orally active antitumor lead compound
Chen, Shuqiang, Bi, Kaijian, Wu, Shanchao, Li, Yu, Huang, Yahui, Sheng, Chunquan, Dong, Guoqiang
Published in European journal of medicinal chemistry (05.08.2021)
Published in European journal of medicinal chemistry (05.08.2021)
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Journal Article