Discovery of Thiadiazoleamide Derivatives as Potent, Selective, and Orally Available Antagonists Disrupting Androgen Receptor Homodimer
Liao, Jianing, Hu, Chenxian, Fu, Weitao, Liao, Jinbiao, Chai, Xin, Shan, Luhu, Xu, Xiaohong, Hou, Tingjun, Sheng, Rong, Li, Dan
Published in Journal of medicinal chemistry (10.10.2024)
Published in Journal of medicinal chemistry (10.10.2024)
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Journal Article
Discovery of 5-Nitro- N -(3-(trifluoromethyl)phenyl) Pyridin-2-amine as a Novel Pure Androgen Receptor Antagonist against Antiandrogen Resistance
Wang, Huating, Wang, Xuwen, Zhong, Haiyang, Cai, Lvtao, Fu, Weitao, Chai, Xin, Liao, Jianing, Sheng, Rong, Shan, Luhu, Xu, Xiaohong, Xu, Lei, Pan, Peichen, Hou, Tingjun, Li, Dan
Published in Journal of medicinal chemistry (07.11.2024)
Published in Journal of medicinal chemistry (07.11.2024)
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Journal Article
Discovery of a Novel Androgen Receptor Antagonist Manifesting Evidence to Disrupt the Dimerization of the Ligand-Binding Domain via Attenuating the Hydrogen-Bonding Network Between the Two Monomers
Fu, Weitao, Zhang, Minkui, Liao, Jianing, Tang, Qing, Lei, Yixuan, Gong, Zhou, Shan, Luhu, Duan, Mojie, Chai, Xin, Pang, Jinping, Tang, Chun, Wang, Xuwen, Xu, Xiaohong, Li, Dan, Sheng, Rong, Hou, Tingjun
Published in Journal of medicinal chemistry (09.12.2021)
Published in Journal of medicinal chemistry (09.12.2021)
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Journal Article
Discovery of N‑(4-(Benzyloxy)-phenyl)-sulfonamide Derivatives as Novel Antagonists of the Human Androgen Receptor Targeting the Activation Function 2
Chai, Xin, Sun, Huiyong, Zhou, Wenfang, Chen, Changwei, Shan, Luhu, Yang, Yuhui, He, Junzhao, Pang, Jinping, Yang, Liu, Wang, Xinyue, Cui, Sunliang, Fu, Yaqin, Xu, Xiaohong, Xu, Lei, Yao, Xiaojun, Li, Dan, Hou, Tingjun
Published in Journal of medicinal chemistry (10.02.2022)
Published in Journal of medicinal chemistry (10.02.2022)
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