Synthesis, biological evaluation, and molecular docking studies of novel N-substituted piperazine-tethered thiophene-3-carboxamide selenides as potent antiproliferative agents with EGFR kinase inhibitory activity
Makhal, Priyanka N., Dayare, Lahu N., Chilvery, Shrilekha, Devi, Priyanka, Sujat Shaikh, Arbaz, Sharma, Anamika, Negi, Aakansha, Godugu, Chandraiah, Rao Kaki, Venkata
Published in Bioorganic chemistry (01.10.2024)
Published in Bioorganic chemistry (01.10.2024)
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Journal Article
Synthesis of indolo/pyrroloazepinone-oxindoles as potential cytotoxic, DNA-intercalating and Topo I inhibitors
Kadagathur, Manasa, Sujat Shaikh, Arbaz, Panda, Biswajit, George, Joel, Phanindranath, Regur, Kumar Sigalapalli, Dilep, Bhale, Nagesh A., Godugu, Chandraiah, Nagesh, Narayana, Shankaraiah, Nagula, Tangellamudi, Neelima D.
Published in Bioorganic chemistry (01.05.2022)
Published in Bioorganic chemistry (01.05.2022)
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Journal Article
Quest for selective MMP9 inhibitors: a computational approach
Shaikh, Arbaz Sujat, Sethi, Aaftaab, Makhal, Priyanka N., Rathi, Brijesh, Kaki, Venkata Rao
Published in Journal of biomolecular structure & dynamics (29.12.2023)
Published in Journal of biomolecular structure & dynamics (29.12.2023)
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Journal Article
Design, synthesis of DNA-interactive 4-thiazolidinone-based indolo-/pyrroloazepinone conjugates as potential cytotoxic and topoisomerase I inhibitors
Kadagathur, Manasa, Patra, Sandip, Devabattula, Geetanjali, George, Joel, Phanindranath, Regur, Shaikh, Arbaz Sujat, Sigalapalli, Dilep Kumar, Godugu, Chandraiah, Nagesh, Narayana, Tangellamudi, Neelima D., Shankaraiah, Nagula
Published in European journal of medicinal chemistry (05.08.2022)
Published in European journal of medicinal chemistry (05.08.2022)
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Journal Article
selenocyclization of secondary allylic carboxamides using Woollins' reagent: to 2,5-disubstituted selenazolines
Makhal, Priyanka N, Dannarm, Srinivas Reddy, Shaikh, Arbaz Sujat, Ahmed, Rezwan, Chilvery, Shrilekha, Dayare, Lahu N, Sonti, Rajesh, Godugu, Chandraiah, Kaki, Venkata Rao
Published in Chemical communications (Cambridge, England) (23.03.2023)
Published in Chemical communications (Cambridge, England) (23.03.2023)
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Journal Article
Exo-trig selenocyclization of secondary allylic carboxamides using Woollins' reagent: en route to 2,5-disubstituted selenazolines
Makhal, Priyanka N., Dannarm, Srinivas Reddy, Shaikh, Arbaz Sujat, Ahmed, Rezwan, Chilvery, Shrilekha, Dayare, Lahu N., Sonti, Rajesh, Godugu, Chandraiah, Kaki, Venkata Rao
Published in Chemical communications (Cambridge, England) (23.03.2023)
Published in Chemical communications (Cambridge, England) (23.03.2023)
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Journal Article
Design, synthesis, anti-cancer activity and in-silico studies of some novel 4,5-dihydroisoxazole-5-carboxamide derivatives
Endoori, Srinivas, Gulipalli, Kali Charan, Bodige, Srinu, Shaikh, Arbaz Sujat, Vemula, Divya, Surapureddi, Sri Ramakrishna, Seelam, Nareshvarma
Published in Synthetic communications (17.11.2021)
Published in Synthetic communications (17.11.2021)
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Journal Article
Naringenin-Zinc Oxide Nanocomposites Amalgamated Polymeric Gel Augmented Drug Delivery and Attenuated Experimental Cutaneous Candidiasis in Balb/c Mice: In Vitro and In Vivo Studies
Katta, Chanti babu, Bahuguna, Deepankar, Veerabomma, Harithasree, Gollapalli, Spandana, Shaikh, Arbaz Sujat, Bhale, Nagesh A., Dikundwar, Amol G., Kaki, Venkat Rao, Singh, Pankaj Kumar, Madan, Jitender
Published in AAPS PharmSciTech (06.06.2024)
Published in AAPS PharmSciTech (06.06.2024)
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Journal Article
Exploration of mercaptoacetamide-linked pyrimidine-1,3,4-oxadiazole derivatives as DNA intercalative topo II inhibitors: Cytotoxicity and apoptosis induction
Shaikh, Arbaz Sujat, Kiranmai, Gaddam, Parimala Devi, G., Makhal, Priyanka N., Sigalapalli, Dilep Kumar, Tokala, Ramya, Kaki, Venkata Rao, Shankaraiah, Nagula, Nagesh, Narayana, Babu, Bathini Nagendra, Tangellamudi, Neelima D.
Published in Bioorganic & medicinal chemistry letters (01.06.2022)
Published in Bioorganic & medicinal chemistry letters (01.06.2022)
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Journal Article
Insights into the pharmacophore-based 3D-QSAR modeling, molecular dynamics simulation studies of certain dihydroxy pyrrolidine/piperidine and aza-flavanone derivatives as α-glucosidase inhibitors
Sigalapalli, Dilep Kumar, Yele, Vidyasrilekha, Jupudi, Srikanth, Shaikh, Arbaz Sujat, Kadagathur, Manasa, Tangellamudi, Neelima D., Nagendra Babu, Bathini
Published in Journal of molecular structure (05.01.2021)
Published in Journal of molecular structure (05.01.2021)
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Journal Article
Naringenin-Capped Silver Nanoparticles Amalgamated Gel for the Treatment of Cutaneous Candidiasis
Katta, Chantibabu, Shaikh, Arbaz Sujat, Bhale, Nagesh, Jyothi, Vaskuri G. S. Sainaga, Kaki, Venkata Rao, Dikundwar, Amol G., Singh, Pankaj Kumar, Shukla, Renu, Mishra, Krishnaveni, Madan, Jitender
Published in AAPS PharmSciTech (25.05.2023)
Published in AAPS PharmSciTech (25.05.2023)
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Journal Article
Cyclodesulfurization: An Enabling Protocol for Synthesis of Various Heterocycles
Kadagathur, Manasa, Shaikh, Arbaz Sujat, Jadhav, Govinda Shivaji, Sigalapalli, Dilep Kumar, Shankaraiah, Nagula, Tangellamudi, Neelima D.
Published in ChemistrySelect (Weinheim) (12.03.2021)
Published in ChemistrySelect (Weinheim) (12.03.2021)
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Journal Article
Development of trisubstituted thiophene-3-arboxamide selenide derivatives as novel EGFR kinase inhibitors with cytotoxic activity
Makhal, Priyanka N, Sood, Anika, Shaikh, Arbaz Sujat, Dayare, Lahu N, Khatri, Dharmendra Kumar, Rao Kaki, Venkata
Published in MedChemComm (13.12.2023)
Published in MedChemComm (13.12.2023)
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Journal Article
Microwave‐Assisted TBHP‐Mediated Synthesis of 2‐Amino‐1,3,4‐oxadiazoles in Water
Kumar Sigalapalli, Dilep, Kadagathur, Manasa, Sujat Shaikh, Arbaz, Jadhav, Govinda S., Bakchi, Bulti, Nagendra Babu, Bathini, Tangellamudi, Neelima D.
Published in ChemistrySelect (Weinheim) (13.11.2020)
Published in ChemistrySelect (Weinheim) (13.11.2020)
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Journal Article