Structure-activity relationship (SAR) study and design strategies of nitrogen-containing heterocyclic moieties for their anticancer activities
Akhtar, Jawaid, Khan, Ahsan Ahmed, Ali, Zulphikar, Haider, Rafi, Shahar Yar, M.
Published in European journal of medicinal chemistry (05.01.2017)
Published in European journal of medicinal chemistry (05.01.2017)
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Design, synthesis, docking and QSAR study of substituted benzimidazole linked oxadiazole as cytotoxic agents, EGFR and erbB2 receptor inhibitors
Akhtar, Md Jawaid, Siddiqui, Anees Ahmad, Khan, Ahsan Ahmed, Ali, Zulphikar, Dewangan, Rikeshwer Prasad, Pasha, Santosh, Yar, M. Shahar
Published in European journal of medicinal chemistry (27.01.2017)
Published in European journal of medicinal chemistry (27.01.2017)
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Journal Article
Design, synthesis, biological evaluation, and in silico studies of 2‐aminobenzothiazole derivatives as potent PI3Kα inhibitors
Haider, Kashif, Ahmad, Kamal, Najmi, Abul Kalam, Das, Subham, Joseph, Alex, Shahar Yar, M.
Published in Archiv der Pharmazie (Weinheim) (01.10.2022)
Published in Archiv der Pharmazie (Weinheim) (01.10.2022)
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Journal Article
1,2,3-triazole tethered Indole-3-glyoxamide derivatives as multiple inhibitors of 5-LOX, COX-2 & tubulin: Their anti-proliferative & anti-inflammatory activity
Naaz, Fatima, Preeti Pallavi, M.C., Shafi, Syed, Mulakayala, Naveen, Shahar Yar, M., Sampath Kumar, H.M.
Published in Bioorganic chemistry (01.12.2018)
Published in Bioorganic chemistry (01.12.2018)
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Journal Article
Synthesis and Cytotoxic Activity of 1,2,4-Triazolo-Linked Bis-Indolyl Conjugates as Dual Inhibitors of Tankyrase and PI3K
Yakkala, Prasanna A., Panda, Samir R., Shafi, Syed, Naidu, V. G. M., Yar, M. Shahar, Ubanako, Philemon N., Adeyemi, Samson A., Kumar, Pradeep, Choonara, Yahya E., Radchenko, Eugene V., Palyulin, Vladimir A., Kamal, Ahmed
Published in Molecules (Basel, Switzerland) (07.11.2022)
Published in Molecules (Basel, Switzerland) (07.11.2022)
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Journal Article
Molecular properties prediction, synthesis and antimicrobial activity of some newer oxadiazole derivatives
Bakht, Mohammed Afroz, Yar, M. Shahar, Abdel-Hamid, Sami Gaber, Al Qasoumi, Saleh I., Samad, Abdul
Published in European journal of medicinal chemistry (01.12.2010)
Published in European journal of medicinal chemistry (01.12.2010)
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Journal Article
Updates on synthesis and biological activities of 1,3,4-oxadiazole: A review
Salahuddin, Mazumder, A., Yar, M. Shahar, Mazumder, R., Chakraborthy, G. S., Ahsan, Mohamed Jawed, Rahman, Mujeeb Ur
Published in Synthetic communications (18.10.2017)
Published in Synthetic communications (18.10.2017)
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Journal Article
Design and synthesis of newer 1,3,4-oxadiazole and 1,2,4-triazole based Topsentin analogues as anti-proliferative agent targeting tubulin
Naaz, Fatima, Ahmad, Faiz, Lone, Bilal Ahmad, Pokharel, Yuba Raj, Fuloria, Neeraj Kumar, Fuloria, Shivkanya, Ravichandran, Manickam, Pattabhiraman, Lalitha, Shafi, Syed, Shahar Yar, M.
Published in Bioorganic chemistry (01.01.2020)
Published in Bioorganic chemistry (01.01.2020)
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Journal Article
Recent Advances in the Synthesis and Anticancer Activity of Some Molecules Other Than Nitrogen Containing Heterocyclic Moeities
Akhtar, Md Jawaid, Yar, M Shahar, Khan, Ahsan Ahmed, Ali, Zulphikar, Haider, Md Rafi
Published in Mini reviews in medicinal chemistry (01.01.2017)
Published in Mini reviews in medicinal chemistry (01.01.2017)
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Current trends and future directions for the synthesis and pharmacological applications of 2-(2-cyanopyrrolidin-1-yl)-N-3-hydroxyadamantan-1-yl) acetamide (Gliptins
Yahya, Shaikh, Shaikh, Mohammad Usman, Deshpande, Prathmesh Pramod, Jaiprakash Navnath, Sangshetti, Choudhary, Akram, Sharma, Nisha, Shafeeque, Mohd, Shahar Yar, M.
Published in Medicinal chemistry research (01.07.2024)
Published in Medicinal chemistry research (01.07.2024)
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Journal Article
Pharmacophore based drug design and synthesis of oxindole bearing hybrid as anticancer agents
Pathak, Ankita, Pandey, Vivek, Raj Pokharel, Yuba, Devaraji, Vinod, Ali, Abuzer, Haider, Kashif, Saad, Suma, Dewangan, Rikeshwer Prasad, Siddiqui, Nadeem, Shahar Yar, M.
Published in Bioorganic chemistry (01.11.2021)
Published in Bioorganic chemistry (01.11.2021)
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Journal Article
Medicinal prospects of antioxidants: A review
Neha, Kumari, Haider, Md Rafi, Pathak, Ankita, Yar, M. Shahar
Published in European journal of medicinal chemistry (15.09.2019)
Published in European journal of medicinal chemistry (15.09.2019)
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Journal Article
Anti-tubulin agents of natural origin: Targeting taxol, vinca, and colchicine binding domains
Naaz, Fatima, Haider, Md Rafi, Shafi, Syed, Yar, M. Shahar
Published in European journal of medicinal chemistry (01.06.2019)
Published in European journal of medicinal chemistry (01.06.2019)
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Journal Article
Design, in-silico study and biological evaluation of newly synthesized 3-chlorobenzofuran congeners as antitubercular agents
Mustaqeem Abdullah, Mohammad, Siddiqui, Nasir A., Mothana, Ramzi A., Nasr, Fahd A., Al-Rehaily, Adnan J., Almarfadi, Omer M., Karim, Shahid, Haider, Kashif, Rafi Haider, Md, Shahar Yar, M.
Published in Arabian journal of chemistry (01.04.2021)
Published in Arabian journal of chemistry (01.04.2021)
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Journal Article
Free radical scavengers: An overview on heterocyclic advances and medicinal prospects
Haider, Kashif, Haider, Md Rafi, Neha, Kumari, Yar, M. Shahar
Published in European journal of medicinal chemistry (15.10.2020)
Published in European journal of medicinal chemistry (15.10.2020)
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Journal Article
Tubulin inhibitors as novel anticancer agents: an overview on patents (2013-2018)
Haider, Kashif, Rahaman, Shaik, Yar, M Shahar, Kamal, Ahmed
Published in Expert opinion on therapeutic patents (03.08.2019)
Published in Expert opinion on therapeutic patents (03.08.2019)
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