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Shi, Qing, Ornstein, Paul L., Briner, Karin, Richardson, Timothy I., Arnold, Macklin B., Backer, Ryan T., Buckmaster, Jennifer L., Canada, Emily J., Doecke, Christopher W., Hertel, Larry W., Honigschmidt, Nick, Hsiung, Hansen M., Husain, Saba, Kuklish, Steve L., Martinelli, Michael J., Mullaney, Jeffrey T., O’Brien, Thomas P., Reinhard, Matt R., Rothhaar, Roger, Shah, Jikesh, Wu, Zhipei, Xie, Chaoyu, Zgombick, John M., Fisher, Matthew J.
Published in Bioorganic & medicinal chemistry letters (01.05.2006)
Published in Bioorganic & medicinal chemistry letters (01.05.2006)
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Benzopyrans as selective estrogen receptor β agonists (SERBAs). Part 3: Synthesis of cyclopentanone and cyclohexanone intermediates for C-ring modification
Richardson, Timothy I., Dodge, Jeffrey A., Durst, Gregory L., Pfeifer, Lance A., Shah, Jikesh, Wang, Yong, Durbin, Jim D., Krishnan, Venkatesh, Norman, Bryan H.
Published in Bioorganic & medicinal chemistry letters (01.09.2007)
Published in Bioorganic & medicinal chemistry letters (01.09.2007)
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Synthesis and Structure−Activity Relationships of Novel Arylpiperazines as Potent and Selective Agonists of the Melanocortin Subtype-4 Receptor
Richardson, Timothy I, Ornstein, Paul L, Briner, Karin, Fisher, Matthew J, Backer, Ryan T, Biggers, C. Kelly, Clay, Michael P, Emmerson, Paul J, Hertel, Larry W, Hsiung, Hansen M, Husain, Saba, Kahl, Steven D, Lee, Jonathan A, Lindstrom, Terry D, Martinelli, Michael J, Mayer, John P, Mullaney, Jeffery T, O'Brien, Thomas P, Pawlak, Joseph M, Revell, Kevin D, Shah, Jikesh, Zgombick, John M, Herr, R. Jason, Melekhov, Alex, Sampson, Peter B, King, Chi-Hsin R
Published in Journal of medicinal chemistry (29.01.2004)
Published in Journal of medicinal chemistry (29.01.2004)
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Discovery of a Potent, Dual Serotonin and Norepinephrine Reuptake Inhibitor
Dreyfus, Nicolas, Myers, Jason K, Badescu, Valentina O, de Frutos, Oscar, de la Puente, Maria Luz, Ding, Chunjin, Filla, Sandra A, Fynboe, Karsten, Gernert, Douglas L, Heinz, Beverly A, Hemrick-Luecke, Susan K, Johnson, Kirk W, Johnson, Michael P, López, Pilar, Love, Patrick L, Martin, Laura J, Masquelin, Thierry, McCoy, Michael J, Mendiola, Javier, Morrow, Denise, Muhlhauser, Mark, Pascual, Gustavo, Perun, Thomas J, Pfeifer, Lance A, Phebus, Lee A, Richards, Simon J, Rincón, Juan Antonio, Seest, Eric P, Shah, Jikesh, Shaojuan, Jia, Simmons, Rosa Maria A, Stephenson, Gregory A, Tromiczak, Eric G, Thompson, Linda K, Walter, Magnus W, Weber, Wayne W, Zarrinmayeh, Hamideh, Thomas, Craig E, Joshi, Elizabeth, Iyengar, Smriti, Johansson, Anette M
Published in ACS medicinal chemistry letters (13.06.2013)
Published in ACS medicinal chemistry letters (13.06.2013)
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Privileged structure based ligands for melanocortin receptors—Substituted benzylic piperazine derivatives
Fisher, Matthew J., Backer, Ryan T., Collado, Iván, de Frutos, Óscar, Husain, Saba, Hsiung, Hansen M., Kuklish, Steve L., Mateo, Ana I., Mullaney, Jeffrey T., Ornstein, Paul L., Paredes, Cristina García, O’Brian, Thomas P., Richardson, Timothy I., Shah, Jikesh, Zgombick, John M., Briner, Karin
Published in Bioorganic & medicinal chemistry letters (15.11.2005)
Published in Bioorganic & medicinal chemistry letters (15.11.2005)
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Inhibidor de recaptación de serotonina y norepinefrina
FILLA, SANDRA, TROMICZAK, ERIC, MASQUELIN, THIERRY, SHAH, JIKESH, JOHANSSON, ANETTE, WALTER, MAGNUS, DREYFUS, NICOLAS
Year of Publication 10.03.2014
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Year of Publication 10.03.2014
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