Synthesis and Biological Evaluation of Novel Dispiro -Indolinones with Anticancer Activity
Ivanenkov, Yan A, Kukushkin, Maxim E, Beloglazkina, Anastasia A, Shafikov, Radik R, Barashkin, Alexander A, Ayginin, Andrey A, Serebryakova, Marina S, Majouga, Alexander G, Skvortsov, Dmitry A, Tafeenko, Viktor A, Beloglazkina, Elena K
Published in Molecules (Basel, Switzerland) (30.01.2023)
Published in Molecules (Basel, Switzerland) (30.01.2023)
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Synthesis of Prostate-Specific Membrane Antigen-Targeted Bimodal Conjugates of Cytotoxic Agents and Antiandrogens and Their Comparative Assessment with Monoconjugates
Zyk, Nikolai Y, Garanina, Anastasiia S, Plotnikova, Ekaterina A, Ber, Anton P, Nimenko, Ekaterina A, Dashkova, Natalia S, Uspenskaia, Anastasiia A, Shafikov, Radik R, Skvortsov, Dmitry A, Petrov, Stanislav A, Pankratov, Andrey A, Zyk, Nikolai V, Majouga, Alexander G, Beloglazkina, Elena K, Machulkin, Aleksei E
Published in International journal of molecular sciences (01.07.2023)
Published in International journal of molecular sciences (01.07.2023)
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New ferrocene-based 2-thio-imidazol-4-ones and their copper complexes. Synthesis and cytotoxicity
Guk, D A, Krasnovskaya, O O, Dashkova, N S, Skvortsov, D A, Rubtsova, M P, Dyadchenko, V P, Yudina, E S, Kosarev, M A, Soldatov, A V, Shapovalov, V V, Semkina, A S, Vlasova, K Y, Pergushov, V I, Shafikov, R R, Andreeva, A A, Melnikov, M Ya, Zyk, N V, Majouga, A G, Beloglazkina, E K
Published in Dalton transactions : an international journal of inorganic chemistry (11.12.2018)
Published in Dalton transactions : an international journal of inorganic chemistry (11.12.2018)
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Journal Article
Correction: New ferrocene-based 2-thio-imidazol-4-ones and their copper complexes. Synthesis and cytotoxicity
Guk, D. A, Krasnovskaya, O. O, Dashkova, N. S, Skvortsov, D. A, Rubtsova, M. P, Dyadchenko, V. P, Yudina, E. S, Kosarev, M. A, Soldatov, A. V, Shapovalov, V. V, Semkina, A. S, Vlasova, K. Y, Pergushov, V. I, Shafikov, R. R, Moiseeva, A. A, Andreeva, A. V, Melnikov, M. Ya, Zyk, N. V, Majouga, A. G, Beloglazkina, E. K
Published in Dalton transactions : an international journal of inorganic chemistry (02.01.2019)
Published in Dalton transactions : an international journal of inorganic chemistry (02.01.2019)
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Optimization of the dipeptide motifs in the PSMA ligands linker structure: synthesis and in vitro evaluation
Uspenskaya, Anastasiia A., Nimenko, Ekaterina A., Shafikov, Radik R., Zyk, Nikolay Y., Evteev, Sergei A., Dashkova, Natalia S., Ivanenkov, Yan A., Majouga, Alexander G., Skvortsov, Dmitry A., Garanina, Anastasiia S., Beloglazkina, Elena K., Machulkin, Aleksei E.
Published in Medicinal chemistry research (2023)
Published in Medicinal chemistry research (2023)
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Synthesis, Characterization, and Preclinical Evaluation of a Small-Molecule Prostate-Specific Membrane Antigen-Targeted Monomethyl Auristatin E Conjugate
Machulkin, Aleksei E, Uspenskaya, Anastasia A, Zyk, Nikolay U, Nimenko, Ekaterina A, Ber, Anton P, Petrov, Stanislav A, Polshakov, Vladimir I, Shafikov, Radik R, Skvortsov, Dmitry A, Plotnikova, Ekaterina A, Pankratov, Andrei A, Smirnova, Galina B, Borisova, Yulia A, Pokrovsky, Vadim S, Kolmogorov, Vasilii S, Vaneev, Alexander N, Khudyakov, Alexander D, Chepikova, Olga E, Kovalev, Sergey, Zamyatnin Jr, Andrey A, Erofeev, Alexander, Gorelkin, Petr, Beloglazkina, Elena K, Zyk, Nikolay V, Khazanova, Elena S, Majouga, Alexander G
Published in Journal of medicinal chemistry (09.12.2021)
Published in Journal of medicinal chemistry (09.12.2021)
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New copper(II) thiohydantoin complexes: Synthesis, characterization, and assessment of their interaction with bovine serum albumin and DNA
Tishchenko, Ksenia, Beloglazkina, Elena, Proskurnin, Mikhail, Malinnikov, Vladislav, Guk, Dmitriy, Muratova, Marina, Krasnovskaya, Olga, Udina, Anna, Skvortsov, Dmitry, Shafikov, Radik R., Ivanenkov, Yan, Aladinskiy, Vladimir, Sorokin, Ivan, Gromov, Oleg, Majouga, Alexander, Zyk, Nikolay
Published in Journal of inorganic biochemistry (01.10.2017)
Published in Journal of inorganic biochemistry (01.10.2017)
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Synthesis and Biological Evaluation of PSMA Ligands with Aromatic Residues and Fluorescent Conjugates Based on Them
Machulkin, Aleksei E, Shafikov, Radik R, Uspenskaya, Anastasia A, Petrov, Stanislav A, Ber, Anton P, Skvortsov, Dmitry A, Nimenko, Ekaterina A, Zyk, Nikolay U, Smirnova, Galina B, Pokrovsky, Vadim S, Abakumov, Maxim A, Saltykova, Irina V, Akhmirov, Rauf T, Garanina, Anastasiia S, Polshakov, Vladimir I, Saveliev, Oleg Y, Ivanenkov, Yan A, Aladinskaya, Anastasiya V, Finko, Alexander V, Yamansarov, Emil U, Krasnovskaya, Olga O, Erofeev, Alexander S, Gorelkin, Petr V, Dontsova, Olga A, Beloglazkina, Elena K, Zyk, Nikolay V, Khazanova, Elena S, Majouga, Alexander G
Published in Journal of medicinal chemistry (22.04.2021)
Published in Journal of medicinal chemistry (22.04.2021)
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Journal Article
Synthesis and initial in vitro evaluation of PSMA-targeting ligands with a modified aromatic moiety at the lysine ε-nitrogen atom
Zyk, Nikolai Y., Ber, Anton P., Nimenko, Ekaterina A., Shafikov, Radik R., Evteev, Sergei A., Petrov, Stanislav A., Uspenskaya, Anastasia A., Dashkova, Natalia S., Ivanenkov, Yan A., Skvortsov, Dmitry A., Beloglazkina, Elena K., Majouga, Alexander G., Machulkin, Aleksei E.
Published in Bioorganic & medicinal chemistry letters (01.09.2022)
Published in Bioorganic & medicinal chemistry letters (01.09.2022)
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Novel Copper-Containing Cytotoxic Agents Based on 2‑Thioxoimidazolones
Krasnovskaya, Olga O, Guk, Dmitry A, Naumov, Alexey E, Nikitina, Vita N, Semkina, Alevtina S, Vlasova, Kseniya Yu, Pokrovsky, Vadim, Ryabaya, Oksana O, Karshieva, Saida S, Skvortsov, Dmitry A, Zhirkina, Irina V, Shafikov, Radik R, Gorelkin, Petr V, Vaneev, Alexander N, Erofeev, Alexander S, Mazur, Dmitrii M, Tafeenko, Viktor A, Pergushov, Vladimir I, Melnikov, Mikhail Ya, Soldatov, Mikhail A, Shapovalov, Victor V, Soldatov, Alexander V, Akasov, Roman. A, Gerasimov, Vasily M, Sakharov, Dmitry A, Moiseeva, Anna A, Zyk, Nikolay V, Beloglazkina, Elena K, Majouga, Alexander G
Published in Journal of medicinal chemistry (12.11.2020)
Published in Journal of medicinal chemistry (12.11.2020)
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PSMA-targeted small-molecule docetaxel conjugate: Synthesis and preclinical evaluation
Machulkin, Aleksei E., Uspenskaya, Anastasia A., Zyk, Nikolay Y., Nimenko, Ekaterina A., Ber, Anton P., Petrov, Stanislav A., Shafikov, Radik R., Skvortsov, Dmitry A., Smirnova, Galina B., Borisova, Yulia A., Pokrovsky, Vadim S., Kolmogorov, Vasilii S., Vaneev, Alexander N., Ivanenkov, Yan A., Khudyakov, Alexander D., Kovalev, Sergei V., Erofeev, Alexander S., Gorelkin, Petr V., Beloglazkina, Elena K., Zyk, Nikolay V., Khazanova, Elena S., Majouga, Alexander G.
Published in European journal of medicinal chemistry (05.01.2022)
Published in European journal of medicinal chemistry (05.01.2022)
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Synthesis and biological evaluation of PSMA-targeting paclitaxel conjugates
Machulkin, Alexey E., Skvortsov, Dmitry A., Ivanenkov, Yan A., Ber, Anton P., Kavalchuk, Mikhail V., Aladinskaya, Anastasia V., Uspenskaya, Anastasia A., Shafikov, Radik R., Plotnikova, Ekaterina A., Yakubovskaya, Raisa I., Nimenko, Ekaterina A., Zyk, Nikolay U., Beloglazkina, Elena K., Zyk, Nikolay V., Koteliansky, Victor E, Majouga, Alexander G.
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
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20-hydroxyecdysone oximes and their rearrangement into lactams
Shafikov, R. V, Urazaeva, Ya. R, Afon'kina, S. R, Savchenko, R. G, Khalilov, L. M, Odinokov, V. N
Published in Russian journal of organic chemistry (01.10.2009)
Published in Russian journal of organic chemistry (01.10.2009)
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Derivatives of 1,1,2,2-tetraaminoethane. Condensation of 1,2-diacetoxy-1,2-bis(ethoxycarbonylamino)ethane and 1-acetoxy-1,2,2-tris(ethoxycarbonylamino)ethane with nitrogen-containing nucleophiles
Shafikov, R. V., Afon'kina, S. R., Savchenko, R. G., Galyautdinov, I. V., Odinokov, V. N.
Published in Russian journal of organic chemistry (01.02.2007)
Published in Russian journal of organic chemistry (01.02.2007)
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