Identification and characterization of influenza variants resistant to a viral endonuclease inhibitor
Song, Min-Suk, Kumar, Gyanendra, Shadrick, William R., Zhou, Wei, Jeevan, Trushar, Li, Zhenmei, Slavish, P. Jake, Fabrizio, Thomas P., Yoon, Sun-Woo, Webb, Thomas R., Webby, Richard J., White, Stephen W.
Published in Proceedings of the National Academy of Sciences - PNAS (29.03.2016)
Published in Proceedings of the National Academy of Sciences - PNAS (29.03.2016)
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Journal Article
Pterin–sulfa conjugates as dihydropteroate synthase inhibitors and antibacterial agents
Zhao, Ying, Shadrick, William R., Wallace, Miranda J., Wu, Yinan, Griffith, Elizabeth C., Qi, Jianjun, Yun, Mi-Kyung, White, Stephen W., Lee, Richard E.
Published in Bioorganic & medicinal chemistry letters (15.08.2016)
Published in Bioorganic & medicinal chemistry letters (15.08.2016)
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Journal Article
Discovering new medicines targeting helicases: challenges and recent progress
Shadrick, William R, Ndjomou, Jean, Kolli, Rajesh, Mukherjee, Sourav, Hanson, Alicia M, Frick, David N
Published in Journal of biomolecular screening (01.08.2013)
Published in Journal of biomolecular screening (01.08.2013)
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Journal Article
Structures of trehalose-6-phosphate phosphatase from pathogenic fungi reveal the mechanisms of substrate recognition and catalysis
Miao, Yi, Tenor, Jennifer L., Toffaletti, Dena L., Washington, Erica J., Liu, Jiuyu, Shadrick, William R., Schumacher, Maria A., Lee, Richard E., Perfect, John R., Brennan, Richard G.
Published in Proceedings of the National Academy of Sciences - PNAS (28.06.2016)
Published in Proceedings of the National Academy of Sciences - PNAS (28.06.2016)
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Journal Article
Bromodomain-Selective BET Inhibitors Are Potent Antitumor Agents against MYC-Driven Pediatric Cancer
Slavish, P Jake, Chi, Liying, Yun, Mi-Kyung, Tsurkan, Lyudmila, Martinez, Nancy E, Jonchere, Barbara, Chai, Sergio C, Connelly, Michele, Waddell, M Brett, Das, Sourav, Neale, Geoffrey, Li, Zhenmei, Shadrick, William R, Olsen, Rachelle R, Freeman, Kevin W, Low, Jonathan A, Price, Jeanine E, Young, Brandon M, Bharatham, Nagakumar, Boyd, Vincent A, Yang, Jun, Lee, Richard E, Morfouace, Marie, Roussel, Martine F, Chen, Taosheng, Savic, Daniel, Guy, R Kiplin, White, Stephen W, Shelat, Anang A, Potter, Philip M
Published in Cancer research (Chicago, Ill.) (01.09.2020)
Published in Cancer research (Chicago, Ill.) (01.09.2020)
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Journal Article
Tyrosine O-sulfation proteoforms affect HIV-1 monoclonal antibody potency
Cai, Cindy X, Doria-Rose, Nicole A, Schneck, Nicole A, Ivleva, Vera B, Tippett, Brad, Shadrick, William R, O'Connell, Sarah, Cooper, Jonathan W, Schneiderman, Zachary, Zhang, Baoshan, Gowetski, Daniel B, Blackstock, Daniel, Demirji, Jacob, Lin, Bob C, Gorman, Jason, Liu, Tracy, Li, Yile, McDermott, Adrian B, Kwong, Peter D, Carlton, Kevin, Gall, Jason G, Lei, Q Paula
Published in Scientific reports (19.05.2022)
Published in Scientific reports (19.05.2022)
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Journal Article
Mosaic quadrivalent influenza vaccine single nanoparticle characterization
Yang, Rong Sylvie, Traver, Maria, Barefoot, Nathan, Stephens, Tyler, Alabanza, Casper, Manzella-Lapeira, Javier, Zou, Guozhang, Wolff, Jeremy, Li, Yile, Resto, Melissa, Shadrick, William, Yang, Yanhong, Ivleva, Vera B, Tsybovsky, Yaroslav, Carlton, Kevin, Brzostowski, Joseph, Gall, Jason G, Lei, Q Paula
Published in Scientific reports (24.02.2024)
Published in Scientific reports (24.02.2024)
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Journal Article
Exploiting a water network to achieve enthalpy-driven, bromodomain-selective BET inhibitors
Shadrick, William R., Slavish, Peter J., Chai, Sergio C., Waddell, Brett, Connelly, Michele, Low, Jonathan A., Tallant, Cynthia, Young, Brandon M., Bharatham, Nagakumar, Knapp, Stefan, Boyd, Vincent A., Morfouace, Marie, Roussel, Martine F., Chen, Taosheng, Lee, Richard E., Kiplin Guy, R., Shelat, Anang A., Potter, Philip M.
Published in Bioorganic & medicinal chemistry (01.01.2018)
Published in Bioorganic & medicinal chemistry (01.01.2018)
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Journal Article
Advances in purification of SARS-CoV-2 spike ectodomain protein using high-throughput screening and non-affinity methods
Cibelli, Nicole, Arias, Gabriel, Figur, McKenzie, Khayat, Shireen S, Leach, Kristin, Loukinov, Ivan, Shadrick, William, Chuenchor, Watchalee, Tsybovsky, Yaroslav, Gulla, Krishana, Gowetski, Daniel B
Published in Scientific reports (15.03.2022)
Published in Scientific reports (15.03.2022)
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Journal Article
Identification and analysis of hepatitis C virus NS3 helicase inhibitors using nucleic acid binding assays
Mukherjee, Sourav, Hanson, Alicia M, Shadrick, William R, Ndjomou, Jean, Sweeney, Noreena L, Hernandez, John J, Bartczak, Diana, Li, Kelin, Frankowski, Kevin J, Heck, Julie A, Arnold, Leggy A, Schoenen, Frank J, Frick, David N
Published in Nucleic acids research (01.09.2012)
Published in Nucleic acids research (01.09.2012)
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Journal Article
A fluorescence-based high throughput assay for the determination of small molecule−human serum albumin protein binding
McCallum, Megan M., Pawlak, Alan J., Shadrick, William R., Simeonov, Anton, Jadhav, Ajit, Yasgar, Adam, Maloney, David J., Arnold, Leggy A.
Published in Analytical and bioanalytical chemistry (01.03.2014)
Published in Analytical and bioanalytical chemistry (01.03.2014)
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Journal Article
Synthesis and evaluation of colletoic acid core derivatives
Ling, Taotao, Gautam, Lekh Nath, Griffith, Elizabeth, Das, Sourav, Lang, Walter, Shadrick, William R., Shelat, Anang, Lee, Richard, Rivas, Fatima
Published in European journal of medicinal chemistry (03.03.2016)
Published in European journal of medicinal chemistry (03.03.2016)
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Journal Article
The role of ZA channel water-mediated interactions in the design of bromodomain-selective BET inhibitors
Bharatham, Nagakumar, Slavish, Peter J., Shadrick, William R., Young, Brandon M., Shelat, Anang A.
Published in Journal of molecular graphics & modelling (01.05.2018)
Published in Journal of molecular graphics & modelling (01.05.2018)
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Journal Article
Ureadepsipeptides as ClpP Activators
Griffith, Elizabeth C, Zhao, Ying, Singh, Aman P, Conlon, Brian P, Tangallapally, Rajendra, Shadrick, William R, Liu, Jiuyu, Wallace, Miranda J, Yang, Lei, Elmore, John M, Li, Yong, Zheng, Zhong, Miller, Darcie J, Cheramie, Martin N, Lee, Robin B, LaFleur, Michael D, Lewis, Kim, Lee, Richard E
Published in ACS infectious diseases (08.11.2019)
Published in ACS infectious diseases (08.11.2019)
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Journal Article
Kinetics of DNA Unwinding by the RecD2 Helicase from Deinococcus radiodurans
Shadrick, William R., Julin, Douglas A.
Published in The Journal of biological chemistry (04.06.2010)
Published in The Journal of biological chemistry (04.06.2010)
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Journal Article
Primuline Derivatives That Mimic RNA to Stimulate Hepatitis C Virus NS3 Helicase-catalyzed ATP Hydrolysis
Sweeney, Noreena L., Shadrick, William R., Mukherjee, Sourav, Li, Kelin, Frankowski, Kevin J., Schoenen, Frank J., Frick, David N.
Published in The Journal of biological chemistry (05.07.2013)
Published in The Journal of biological chemistry (05.07.2013)
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Journal Article
An Ire1–Phk1 Chimera Reveals a Dispensable Role of Autokinase Activity in Endoplasmic Reticulum Stress Response
Mannan, M. Amin-ul, Shadrick, William R., Biener, Gabriel, Shin, Byung-Sik, Anshu, Ashish, Raicu, Valerica, Frick, David N., Dey, Madhusudan
Published in Journal of molecular biology (26.06.2013)
Published in Journal of molecular biology (26.06.2013)
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Journal Article
Fluorescent primuline derivatives inhibit hepatitis C virus NS3-catalyzed RNA unwinding, peptide hydrolysis and viral replicase formation
Ndjomou, Jean, Kolli, Rajesh, Mukherjee, Sourav, Shadrick, William R., Hanson, Alicia M., Sweeney, Noreena L., Bartczak, Diana, Li, Kelin, Frankowski, Kevin J., Schoenen, Frank J., Frick, David N.
Published in Antiviral research (01.11.2012)
Published in Antiviral research (01.11.2012)
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Journal Article