Biased allosteric modulation at the CaS receptor engendered by structurally diverse calcimimetics
Cook, A E, Mistry, S N, Gregory, K J, Furness, S G B, Sexton, P M, Scammells, P J, Conigrave, A D, Christopoulos, A, Leach, K
Published in British journal of pharmacology (01.01.2015)
Published in British journal of pharmacology (01.01.2015)
Get full text
Journal Article
Discovery of antiandrogen activity of nonsteroidal scaffolds of marketed drugs
Bisson, W.H, Cheltsov, A.V, Bruey-Sedano, N, Lin, B, Chen, J, Goldberger, N, May, L.T, Christopoulos, A, Dalton, J.T, Sexton, P.M, Zhang, X.-K, Abagyan, R
Published in Proceedings of the National Academy of Sciences - PNAS (17.07.2007)
Published in Proceedings of the National Academy of Sciences - PNAS (17.07.2007)
Get full text
Journal Article
Impact of species variability and ‘probe‐dependence’ on the detection and in vivo validation of allosteric modulation at the M4 muscarinic acetylcholine receptor
Suratman, S, Leach, K, Sexton, PM, Felder, CC, Loiacono, RE, Christopoulos, A
Published in British journal of pharmacology (01.04.2011)
Published in British journal of pharmacology (01.04.2011)
Get full text
Journal Article
Hematological defects in the oc/oc mouse, a model of infantile malignant osteopetrosis
BLIN-WAKKACH, C, WAKKACH, A, SEXTON, P. M, ROCHET, N, CARLE, G. F
Published in Leukemia (01.09.2004)
Published in Leukemia (01.09.2004)
Get full text
Journal Article
Involvement of the sigma1 (σ1) receptor in the anti‐amnesic, but not antidepressant‐like, effects of the aminotetrahydrofuran derivative ANAVEX1‐41
Espallergues, J, Lapalud, P, Christopoulos, A, Avlani, V A, Sexton, P M, Vamvakides, A, Maurice, T
Published in British journal of pharmacology (01.09.2007)
Published in British journal of pharmacology (01.09.2007)
Get full text
Journal Article
Amylin receptors: molecular composition and pharmacology
Hay, D L, Christopoulos, G, Christopoulos, A, Sexton, P M
Published in Biochemical Society transactions (01.11.2004)
Published in Biochemical Society transactions (01.11.2004)
Get more information
Journal Article
In vitro autoradiographic localization of amylin binding sites in rat brain
Sexton, P.M., Paxinos, G., Kenney, M.A., Wookey, P.J., Beaumont, K.
Published in Neuroscience (01.09.1994)
Published in Neuroscience (01.09.1994)
Get full text
Journal Article
Allosteric Modulation of G Protein-Coupled Receptors
May, L T, Avlani, V A, Sexton, P M, Christopoulos, A
Published in Current pharmaceutical design (01.01.2004)
Published in Current pharmaceutical design (01.01.2004)
Get full text
Journal Article
G-protein-coupled receptor allosterism: the promise and the problem(s)
Christopoulos, A, May, L T, Avlani, V A, Sexton, P M
Published in Biochemical Society transactions (01.11.2004)
Published in Biochemical Society transactions (01.11.2004)
Get more information
Journal Article
Calcitonin receptor antibodies in the identification of osteoclasts
Quinn, J.M.W, Morfis, M, Lam, M.H.C, Elliott, J, Kartsogiannis, V, Williams, E.D, Gillespie, M.T, Martin, T.J, Sexton, P.M
Published in Bone (New York, N.Y.) (01.07.1999)
Published in Bone (New York, N.Y.) (01.07.1999)
Get full text
Journal Article
Conference Proceeding
Identification of brain isoforms of the rat calcitonin receptor
SEXTON, P. M, SOUHEIR HOUSSAMI, HILTON, J. M, O'KEEFFE, L. M, CENTER, R. J, GILLESPIE, M. T, DARCY, P, FINDLAY, D. M
Published in Molecular endocrinology (Baltimore, Md.) (01.06.1993)
Published in Molecular endocrinology (Baltimore, Md.) (01.06.1993)
Get full text
Journal Article
Mouse receptor-activity-modifying proteins 1, -2 and -3: amino acid sequence, expression and function
Husmann, Knut, Sexton, P.M, Fischer, J.A, Born, W
Published in Molecular and cellular endocrinology (25.04.2000)
Published in Molecular and cellular endocrinology (25.04.2000)
Get full text
Journal Article
In vitro autoradiographic localization of calcitonin and amylin binding sites in monkey brain
Paxinos, G, Chai, S.Y, Christopoulos, G, Huang, X.-F, Toga, A.W, Wang, H.Q, Sexton, P.M
Published in Journal of chemical neuroanatomy (01.07.2004)
Published in Journal of chemical neuroanatomy (01.07.2004)
Get full text
Journal Article
Abundant calcitonin receptors in isolated rat osteoclasts: biochemical and autoradiographic characterization
NICHOLSON, G. C, MOSELEY, J. M, SEXTON, P. M, MENDELSOHN, F. A. O, MARTIN, T. J
Published in The Journal of clinical investigation (01.08.1986)
Published in The Journal of clinical investigation (01.08.1986)
Get full text
Conference Proceeding
Journal Article