Stereodivergent synthesis of 5-aminopipecotic acids and application in the preparation of a cyclic RGD peptidomimetic as a nanomolar alpha(v)beta(3) integrin ligand
Sernissi, Lorenzo, Ricci, Luciano, Scarpi, Dina, Bianchini, Francesca, Arosio, Daniela, Contini, Alessandro, Occhiato, Ernesto G.
Published in Organic & biomolecular chemistry (14.05.2018)
Published in Organic & biomolecular chemistry (14.05.2018)
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Journal Article
Cyclic RGD peptidomimetics containing 4- and 5-amino-cyclopropane pipecolic acid (CPA) templates as dual αVβ3 and α5β1 integrin ligands
Sernissi, Lorenzo, Trabocchi, Andrea, Scarpi, Dina, Bianchini, Francesca, Occhiato, Ernesto G.
Published in Bioorganic & medicinal chemistry (15.02.2016)
Published in Bioorganic & medicinal chemistry (15.02.2016)
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Journal Article
Cyclic RGD peptidomimetics containing 4-and 5-aminocyclopropane pipecolic acid (CPA) templates as dual alpha(V)beta(3) and alpha(5)beta(1) integrin ligands
Sernissi, Lorenzo, Trabocchi, Andrea, Scarpi, Dina, Bianchini, Francesca, Occhiato, Ernesto G.
Published in Bioorganic & medicinal chemistry (15.02.2016)
Published in Bioorganic & medicinal chemistry (15.02.2016)
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Journal Article
Cyclopropane Pipecolic Acids as Templates for Linear and Cyclic Peptidomimetics: Application in the Synthesis of an Arg-Gly-Asp (RGD)-Containing Peptide as an alpha(v)beta(3) Integrin Ligand
Sernissi, Lorenzo, Petrovic, Martina, Scarpi, Dina, Guarna, Antonio, Trabocchi, Andrea, Bianchini, Francesca, Occhiato, Ernesto G.
Published in Chemistry : a European journal (25.08.2014)
Published in Chemistry : a European journal (25.08.2014)
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Journal Article
In search of constrained FTY720 and phytosphingosine analogs as dual acting anticancer agents targeting metabolic and epigenetic pathways
Garsi, Jean-Baptiste, Sernissi, Lorenzo, Vece, Vito, Hanessian, Stephen, McCracken, Alison N., Simitian, Grigor, Edinger, Aimee L.
Published in European journal of medicinal chemistry (05.11.2018)
Published in European journal of medicinal chemistry (05.11.2018)
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Journal Article
Stereodivergent synthesis of 5-aminopipecolic acids and application in the preparation of a cyclic RGD peptidomimetic as a nanomolar αVβ3 integrin ligandElectronic supplementary information (ESI) available: Further computational calculations and NMR spectra of all new compounds. See DOI: 10.1039/c8ob00534f
Sernissi, Lorenzo, Ricci, Luciano, Scarpi, Dina, Bianchini, Francesca, Arosio, Daniela, Contini, Alessandro, Occhiato, Ernesto G
Year of Publication 09.05.2018
Year of Publication 09.05.2018
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Journal Article
Stereodivergent synthesis of 5-aminopipecolic acids and application in the preparation of a cyclic RGD peptidomimetic as a nanomolar αVβ3 integrin ligand
Sernissi, Lorenzo, Ricci, Luciano, Scarpi, Dina, Bianchini, Francesca, Arosio, Daniela, Contini, Alessandro, Occhiato, Ernesto G
Published in Organic & biomolecular chemistry (2018)
Published in Organic & biomolecular chemistry (2018)
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Journal Article
Synthesis and conformational analysis of peptides embodying 2,3-methanopipecolic acidsElectronic supplementary information (ESI) available: Experimental procedures, characterization data and NMR spectra of all new compounds, computational calculations and biological assays. See DOI: 10.1039/c7ob01617d
Ricci, Luciano, Sernissi, Lorenzo, Scarpi, Dina, Bianchini, Francesca, Contini, Alessandro, Occhiato, Ernesto G
Year of Publication 16.08.2017
Year of Publication 16.08.2017
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Journal Article
Cyclopropane Pipecolic Acids as Templates for Linear and Cyclic Peptidomimetics: Application in the Synthesis of an Arg-Gly-Asp (RGD)-Containing Peptide as an αvβ3 Integrin Ligand
Sernissi, Lorenzo, Petrović, Martina, Scarpi, Dina, Guarna, Antonio, Trabocchi, Andrea, Bianchini, Francesca, Occhiato, Ernesto G.
Published in Chemistry : a European journal (25.08.2014)
Published in Chemistry : a European journal (25.08.2014)
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Journal Article
Stereodivergent synthesis of 5-aminopipecolic acids and application in the preparation of a cyclic RGD peptidomimetic as a nanomolar α V β 3 integrin ligand
Sernissi, Lorenzo, Ricci, Luciano, Scarpi, Dina, Bianchini, Francesca, Arosio, Daniela, Contini, Alessandro, Occhiato, Ernesto G
Published in Organic & biomolecular chemistry (09.05.2018)
Published in Organic & biomolecular chemistry (09.05.2018)
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Journal Article
Design, synthesis and anticancer activity of constrained sphingolipid-phenoxazine/phenothiazine hybrid constructs targeting protein phosphatase 2A
Garsi, Jean-Baptiste, Vece, Vito, Sernissi, Lorenzo, Auger-Morin, Catherine, Hanessian, Stephen, McCracken, Alison N., Selwan, Elizabeth, Ramirez, Cuauhtemoc, Dahal, Amogha, Romdhane, Nadine Ben, Finicle, Brendan T., Edinger, Aimee L.
Published in Bioorganic & medicinal chemistry letters (15.09.2019)
Published in Bioorganic & medicinal chemistry letters (15.09.2019)
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Journal Article
Cyclic RGD peptidomimetics containing 4- and 5-amino-cyclopropane pipecolic acid (CPA) templates as dual alpha sub(V) beta sub(3) and alpha sub(5) beta sub(1) integrin ligands
Sernissi, Lorenzo, Trabocchi, Andrea, Scarpi, Dina, Bianchini, Francesca, Occhiato, Ernesto G
Published in Bioorganic & medicinal chemistry (15.02.2016)
Published in Bioorganic & medicinal chemistry (15.02.2016)
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Journal Article
Cyclopropane Pipecolic Acids as Templates for Linear and Cyclic Peptidomimetics: Application in the Synthesis of an Arg-Gly-Asp (RGD)-Containing Peptide as an [alpha]v[beta]3 Integrin Ligand
Sernissi, Lorenzo, Petrovic, Martina, Scarpi, Dina, Guarna, Antonio, Trabocchi, Andrea, Bianchini, Francesca, Occhiato, Ernesto G
Published in Chemistry : a European journal (25.08.2014)
Published in Chemistry : a European journal (25.08.2014)
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Journal Article
Cyclopropane Pipecolic Acids as Templates for Linear and Cyclic Peptidomimetics: Application in the Synthesis of an Arg‐Gly‐Asp (RGD)‐Containing Peptide as an α v β 3 Integrin Ligand
Sernissi, Lorenzo, Petrović, Martina, Scarpi, Dina, Guarna, Antonio, Trabocchi, Andrea, Bianchini, Francesca, Occhiato, Ernesto G.
Published in Chemistry : a European journal (25.08.2014)
Published in Chemistry : a European journal (25.08.2014)
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Journal Article
Cyclopropane Pipecolic Acids as Templates for Linear and Cyclic Peptidomimetics: Application in the Synthesis of an Arg-Gly-Asp (RGD)-Containing Peptide as an alpha sub(v) beta sub(3) Integrin Ligand
Sernissi, Lorenzo, Petrovic, Martina, Scarpi, Dina, Guarna, Antonio, Trabocchi, Andrea, Bianchini, Francesca, Occhiato, Ernesto G
Published in Chemistry : a European journal (01.08.2014)
Published in Chemistry : a European journal (01.08.2014)
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Journal Article
Phosphorylation of a constrained azacyclic FTY720 analog enhances anti-leukemic activity without inducing S1P receptor activation
McCracken, A N, McMonigle, R J, Tessier, J, Fransson, R, Perryman, M S, Chen, B, Keebaugh, A, Selwan, E, Barr, S A, Kim, S M, Roy, S G, Liu, G, Fallegger, D, Sernissi, L, Brandt, C, Moitessier, N, Snider, A J, Clare, S, Müschen, M, Huwiler, A, Kleinman, M T, Hanessian, S, Edinger, A L
Published in Leukemia (01.03.2017)
Published in Leukemia (01.03.2017)
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SUBSTITUTED THIOPHENE FUSED DERIVATIVES, COMPOSITIONS COMPRISING THE SAME AND THEIR USE AS PHARMACEUTICALS
VAISBURG, Arkadii, GUAY, Daniel, CARON, Antoine, SEGUELA, Philippe, ASE, Ariel Ruben, SERNISSI, Lorenzo, GUERIN, Vincent, STURINO, Claudio, EPIFANOV, Maxim, SABBATANI, Juliette, ST-GEORGES, Catherine, BERGER, Kathleen Jessie, FATEMI, Solmaz
Year of Publication 26.09.2024
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Year of Publication 26.09.2024
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