The atypical ‘hippocampal’ glutamate receptor coupled to phospholipase D that controls stretch‐sensitivity in primary mechanosensory nerve endings is homomeric purely metabotropic GluK2
Thompson, Karen J., Watson, Sonia, Zanato, Chiara, Dall'Angelo, Sergio, De Nooij, Joriene C., Pace‐Bonello, Bethany, Shenton, Fiona C., Sanger, Helen E., Heinz, Beverly A., Broad, Lisa M., Grosjean, Noelle, McQuillian, Jessica R., Dubini, Marina, Pyner, Susan, Greig, Iain, Zanda, Matteo, Bleakman, David, Banks, Robert W., Bewick, Guy S.
Published in Experimental physiology (01.01.2024)
Published in Experimental physiology (01.01.2024)
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Journal Article
[F-18]-5-Fluoro-5-deoxyribose, an efficient peptide bioconjugation ligand for positron emission tomography (PET) imaging
Li, Xiang-Guo, Dall'Angelo, Sergio, Schweiger, Lutz F., Zanda, Matteo, O'Hagan, David
Published in Chemical communications (Cambridge, England) (28.05.2012)
Published in Chemical communications (Cambridge, England) (28.05.2012)
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Journal Article
A Weakened Immune Response to Synthetic Exo-Peptides Predicts a Potential Biosecurity Risk in the Retrieval of Exo-Microorganisms
Schaefer, Katja, Dambuza, Ivy M, Dall'Angelo, Sergio, Yuecel, Raif, Jaspars, Marcel, Trembleau, Laurent, Zanda, Matteo, Brown, Gordon D, Netea, Mihai G, Gow, Neil A R
Published in Microorganisms (Basel) (17.07.2020)
Published in Microorganisms (Basel) (17.07.2020)
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Journal Article
Protein tyrosine phosphatase 1B in metabolic diseases and drug development
Delibegović, Mirela, Dall'Angelo, Sergio, Dekeryte, Ruta
Published in Nature reviews. Endocrinology (01.06.2024)
Published in Nature reviews. Endocrinology (01.06.2024)
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Journal Article
Protection of Sinorhizobium against host cysteine-rich antimicrobial peptides is critical for symbiosis
Haag, Andreas F, Baloban, Mikhail, Sani, Monica, Kerscher, Bernhard, Pierre, Olivier, Farkas, Attila, Longhi, Renato, Boncompagni, Eric, Hérouart, Didier, Dall'angelo, Sergio, Kondorosi, Eva, Zanda, Matteo, Mergaert, Peter, Ferguson, Gail P
Published in PLoS biology (01.10.2011)
Published in PLoS biology (01.10.2011)
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Journal Article
The Trifluoromethyl Group as a Bioisosteric Replacement of the Aliphatic Nitro Group in CB1 Receptor Positive Allosteric Modulators
Tseng, Chih-Chung, Baillie, Gemma, Donvito, Giulia, Mustafa, Mohammed A, Juola, Sophie E, Zanato, Chiara, Massarenti, Chiara, Dall’Angelo, Sergio, Harrison, William T. A, Lichtman, Aron H, Ross, Ruth A, Zanda, Matteo, Greig, Iain R
Published in Journal of medicinal chemistry (23.05.2019)
Published in Journal of medicinal chemistry (23.05.2019)
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Journal Article
NGR Tumor-Homing Peptides: Structural Requirements for Effective APN (CD13) Targeting
Graziadio, Alessandra, Zanda, Matteo, Frau, Simona, Fleming, Ian N, Musolino, Manuele, Dall’Angelo, Sergio, Baldassarre, Massimiliano, Piras, Monica
Published in Bioconjugate chemistry (18.05.2016)
Published in Bioconjugate chemistry (18.05.2016)
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Journal Article
Binding of αvβ3 Integrin-Specific Radiotracers Is Modulated by Both Integrin Expression Level and Activation Status
Andriu, Alexandra, Crockett, Julie, Dall’Angelo, Sergio, Piras, Monica, Zanda, Matteo, Fleming, Ian N.
Published in Molecular imaging and biology (01.02.2018)
Published in Molecular imaging and biology (01.02.2018)
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Journal Article
Design, Synthesis, Conjugation, and Reactivity of Novel trans,trans-1,5-Cyclooctadiene-Derived Bioorthogonal Linkers
Longo, Beatrice, Zanato, Chiara, Piras, Monica, Dall’Angelo, Sergio, Windhorst, Albert D, Vugts, Danielle J, Baldassarre, Massimiliano, Zanda, Matteo
Published in Bioconjugate chemistry (16.09.2020)
Published in Bioconjugate chemistry (16.09.2020)
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Journal Article
Design, synthesis, in vitro characterization and preliminary imaging studies on fluorinated bile acid derivatives as PET tracers to study hepatic transporters
Testa, Andrea, Dall’Angelo, Sergio, Mingarelli, Marco, Augello, Andrea, Schweiger, Lutz, Welch, Andy, Elmore, Charles S., Sharma, Pradeep, Zanda, Matteo
Published in Bioorganic & medicinal chemistry (01.02.2017)
Published in Bioorganic & medicinal chemistry (01.02.2017)
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Journal Article
Preclinical Evaluation of [18F]LCATD as a PET Tracer to Study Drug-Drug Interactions Caused by Inhibition of Hepatic Transporters
Zanda, Matteo, Sharma, Pradeep, Elmore, Charles S., Welch, Andrew, Schweiger, Lutz, Augello, Andrea, Mingarelli, Marco, Dall’Angelo, Sergio, Testa, Andrea, Dawson, Dana
Published in Contrast media and molecular imaging (01.01.2018)
Published in Contrast media and molecular imaging (01.01.2018)
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Journal Article
The Trifluoromethyl Group as a Bioisosteric Replacement of the Aliphatic Nitro Group in CB 1 Receptor Positive Allosteric Modulators
Tseng, Chih-Chung, Baillie, Gemma, Donvito, Giulia, Mustafa, Mohammed A, Juola, Sophie E, Zanato, Chiara, Massarenti, Chiara, Dall'Angelo, Sergio, Harrison, William T A, Lichtman, Aron H, Ross, Ruth A, Zanda, Matteo, Greig, Iain R
Published in Journal of medicinal chemistry (23.05.2019)
Published in Journal of medicinal chemistry (23.05.2019)
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Journal Article
Chemoenzymatic Late‐Stage Modifications Enable Downstream Click‐Mediated Fluorescent Tagging of Peptides
Colombano, Alessandro, Dalponte, Luca, Dall'Angelo, Sergio, Clemente, Claudia, Idress, Mohannad, Ghazal, Ahmad, Houssen, Wael E.
Published in Angewandte Chemie International Edition (11.04.2023)
Published in Angewandte Chemie International Edition (11.04.2023)
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Journal Article
An Efficient Route to N-Monosubstituted Guanidino-Lactams
Tommasi, Sara, Zanato, Chiara, Carabeo, Rey, Mangoni, Arduino A., Dall'Angelo, Sergio, Zanda, Matteo
Published in Synthesis (Stuttgart) (01.10.2015)
Published in Synthesis (Stuttgart) (01.10.2015)
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