Design, synthesis, kinetic mechanism and molecular docking studies of novel 1-pentanoyl-3-arylthioureas as inhibitors of mushroom tyrosinase and free radical scavengers
Larik, Fayaz Ali, Saeed, Aamer, Channar, Pervaiz Ali, Muqadar, Urooj, Abbas, Qamar, Hassan, Mubashir, Seo, Sung-Yum, Bolte, Michael
Published in European journal of medicinal chemistry (01.12.2017)
Published in European journal of medicinal chemistry (01.12.2017)
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Journal Article
The exploration of novel Alzheimer’s therapeutic agents from the pool of FDA approved medicines using drug repositioning, enzyme inhibition and kinetic mechanism approaches
Hassan, Mubashir, Raza, Hussain, Abbasi, Muhammad Athar, Moustafa, Ahmed A., Seo, Sung-Yum
Published in Biomedicine & pharmacotherapy (01.01.2019)
Published in Biomedicine & pharmacotherapy (01.01.2019)
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Journal Article
Hybrid Pharmacophoric Approach in the Design and Synthesis of Coumarin Linked Pyrazolinyl as Urease Inhibitors, Kinetic Mechanism and Molecular Docking
Saeed, Aamer, Mahesar, Parvez Ali, Channar, Pervaiz Ali, Larik, Fayaz Ali, Abbas, Qamar, Hassan, Mubashir, Raza, Hussain, Seo, Sung‐Yum
Published in Chemistry & biodiversity (01.08.2017)
Published in Chemistry & biodiversity (01.08.2017)
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Journal Article
Novel C-2 Symmetric Molecules as α-Glucosidase and α-Amylase Inhibitors: Design, Synthesis, Kinetic Evaluation, Molecular Docking and Pharmacokinetics
Shahzad, Danish, Saeed, Aamer, Larik, Fayaz Ali, Channar, Pervaiz Ali, Abbas, Qamar, Alajmi, Mohamed F, Arshad, M Ifzan, Erben, Mauricio F, Hassan, Mubashir, Raza, Hussain, Seo, Sung-Yum, El-Seedi, Hesham R
Published in Molecules (Basel, Switzerland) (17.04.2019)
Published in Molecules (Basel, Switzerland) (17.04.2019)
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Journal Article
Novel 1,3‐oxazine‐tetrazole hybrids as mushroom tyrosinase inhibitors and free radical scavengers: Synthesis, kinetic mechanism, and molecular docking studies
Qamar, Rabia, Saeed, Aamer, Larik, Fayaz Ali, Abbas, Qamar, Hassan, Mubashir, Raza, Hussain, Seo, Sung‐Yum
Published in Chemical biology & drug design (01.02.2019)
Published in Chemical biology & drug design (01.02.2019)
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Journal Article
Design and Synthesis of New Porphyrin Analogues as Potent Photosensitizers for Photodynamic Therapy: Spectroscopic Approach
Mahajan, Prasad G., Dige, Nilam C., Vanjare, Balasaheb D., Kim, Chong-Hyeak, Seo, Sung-Yum, Lee, Ki Hwan
Published in Journal of fluorescence (01.03.2020)
Published in Journal of fluorescence (01.03.2020)
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Journal Article
Sulfonamide-Linked Ciprofloxacin, Sulfadiazine and Amantadine Derivatives as a Novel Class of Inhibitors of Jack Bean Urease; Synthesis, Kinetic Mechanism and Molecular Docking
Channar, Pervaiz Ali, Saeed, Aamer, Albericio, Fernando, Larik, Fayaz Ali, Abbas, Qamar, Hassan, Mubashir, Raza, Hussain, Seo, Sung-Yum
Published in Molecules (Basel, Switzerland) (16.08.2017)
Published in Molecules (Basel, Switzerland) (16.08.2017)
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Journal Article
Novel 1,2,4-triazole analogues as mushroom tyrosinase inhibitors: synthesis, kinetic mechanism, cytotoxicity and computational studies
Vanjare, Balasaheb D., Mahajan, Prasad G., Dige, Nilam C., Raza, Hussain, Hassan, Mubashir, Han, Yohan, Kim, Song Ja, Seo, Sung-Yum, Lee, Ki Hwan
Published in Molecular diversity (01.11.2021)
Published in Molecular diversity (01.11.2021)
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Journal Article
Synthesis and biological evaluation of 1,2,4-triazolidine-3-thiones as potent acetylcholinesterase inhibitors: in vitro and in silico analysis through kinetics, chemoinformatics and computational approaches
Mahajan, Prasad G., Dige, Nilam C., Vanjare, Balasaheb D., Raza, Hussain, Hassan, Mubashir, Seo, Sung-Yum, Kim, Chong- Hyeak, Lee, Ki Hwan
Published in Molecular diversity (01.11.2020)
Published in Molecular diversity (01.11.2020)
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An expedient synthesis of N‐(1‐(5‐mercapto‐4‐((substituted benzylidene)amino)‐4H‐1,2,4‐triazol‐3‐yl)‐2‐phenylethyl)benzamides as jack bean urease inhibitors and free radical scavengers: Kinetic mechanism and molecular docking studies
Saeed, Aamer, Larik, Fayaz Ali, Channar, Pervaiz Ali, Mehfooz, Haroon, Ashraf, Mohammad Haseeb, Abbas, Qamar, Hassan, Mubashir, Seo, Sung‐Yum
Published in Chemical biology & drug design (01.11.2017)
Published in Chemical biology & drug design (01.11.2017)
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Journal Article
Drug-1,3,4-Thiadiazole Conjugates as Novel Mixed-Type Inhibitors of Acetylcholinesterase: Synthesis, Molecular Docking, Pharmacokinetics, and ADMET Evaluation
Ujan, Rabail, Saeed, Aamer, Channar, Pervaiz Ali, Larik, Fayaz Ali, Abbas, Qamar, Alajmi, Mohamed F, El-Seedi, Hesham R, Rind, Mahboob Ali, Hassan, Mubashir, Raza, Hussain, Seo, Sung-Yum
Published in Molecules (Basel, Switzerland) (28.02.2019)
Published in Molecules (Basel, Switzerland) (28.02.2019)
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Journal Article
Development of highly potent melanogenesis inhibitor by in vitro, in vivo and computational studies
Abbas, Qamar, Ashraf, Zaman, Hassan, Mubashir, Nadeem, Humaira, Latif, Muhammad, Afzal, Samina, Seo, Sung-Yum
Published in Drug design, development and therapy (01.01.2017)
Published in Drug design, development and therapy (01.01.2017)
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Journal Article
Extending the scope of amantadine drug by incorporation of phenolic azo Schiff bases as potent selective inhibitors of carbonic anhydrase II, drug‐likeness and binding analysis
Channar, Pervaiz A., Saeed, Aamer, Shahzad, Danish, Larik, Fayaz Ali, Hassan, Mubashir, Raza, Hussain, Abbas, Qamar, Seo, Sung‐Yum
Published in Chemical biology & drug design (01.09.2018)
Published in Chemical biology & drug design (01.09.2018)
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Journal Article
Iminothiazoline-Sulfonamide Hybrids as Jack Bean Urease Inhibitors; Synthesis, Kinetic Mechanism and Computational Molecular Modeling
Saeed, Aamer, Mahmood, Shams-ul, Rafiq, Muhammad, Ashraf, Zaman, Jabeen, Farukh, Seo, Sung-Yum
Published in Chemical biology & drug design (01.03.2016)
Published in Chemical biology & drug design (01.03.2016)
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Journal Article
Symmetrical Heterocyclic Cage Skeleton: Synthesis, Urease Inhibition Activity, Kinetic Mechanistic Insight, and Molecular Docking Analyses
Hanif, Muhammad, Kanwal, Fariha, Rafiq, Muhammad, Hassan, Mubashir, Mustaqeem, Muhammad, Seo, Sung-Yum, Zhang, Yunlong, Lu, Changrui, Chen, Ting, Saleem, Muhammad
Published in Molecules (Basel, Switzerland) (16.01.2019)
Published in Molecules (Basel, Switzerland) (16.01.2019)
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Journal Article
Convergent synthesis of carbonic anhydrase inhibiting bi‐heterocyclic benzamides: Structure–activity relationship and mechanistic explorations through enzyme inhibition, kinetics, and computational studies
Khan, Farhan M., Abbasi, Muhammad A., Aziz‐ur‐Rehman, Siddiqui, Sabahat Z., Sadiq Butt, Abdul R., Raza, Hussain, Zafar, Ayesha, Ali Shah, Syed A., Shahid, Muhammad, Seo, Sung‐Yum
Published in Journal of heterocyclic chemistry (01.05.2021)
Published in Journal of heterocyclic chemistry (01.05.2021)
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