Anti‐inflammatory activity of phosphodiesterase (PDE)‐IV inhibitors in acute and chronic models of inflammation
SEKUT, L., YARNALL, D., STIMPSON, S. A., NOEL, L. S., BATEMAN‐FITE, R., CLARK, R. L., BRACKEEN, M. F., MENIUS, J. A., CONNOLLY, K. M.
Published in Clinical and experimental immunology (01.04.1995)
Published in Clinical and experimental immunology (01.04.1995)
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Journal Article
Anti‐inflammatory activity of salmeterol: down‐regulation of cytokine production
SEKUT, L., CHAMPION, B. R., PAGE, K., JR, J. A. MENIUS, CONNOLLY, K. M.
Published in Clinical and experimental immunology (01.03.1995)
Published in Clinical and experimental immunology (01.03.1995)
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Journal Article
Inhibition of cartilage and bone destruction in adjuvant arthritis in the rat by a matrix metalloproteinase inhibitor
Conway, J G, Wakefield, J A, Brown, R H, Marron, B E, Sekut, L, Stimpson, S A, McElroy, A, Menius, J A, Jeffreys, J J, Clark, R L
Published in The Journal of experimental medicine (01.08.1995)
Published in The Journal of experimental medicine (01.08.1995)
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Journal Article
Caspase-1 processes IFN-γ-inducing factor and regulates LPS-induced IFN- γ production
Ghayur, Tariq, Banerjee, Subhashis, Hugunin, Margaret, Butler, Deborah, Herzog, Linda, Carter, Adam, Quintal, Lucia, Sekut, Les, Talanian, Robert, Paskind, Michael, Wong, Winnie, Kamen, Robert, Tracey, Daniel, Alien, Hamish
Published in Nature (London) (10.04.1997)
Published in Nature (London) (10.04.1997)
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Journal Article
Albutropin: a growth hormone–albumin fusion with improved pharmacokinetics and pharmacodynamics in rats and monkeys
Osborn, Blaire L, Sekut, Les, Corcoran, Marta, Poortman, Carol, Sturm, Bonnie, Chen, Guoxian, Mather, Donald, Lin, Hsiu Ling, Parry, Tom J
Published in European journal of pharmacology (05.12.2002)
Published in European journal of pharmacology (05.12.2002)
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Journal Article
Regulation of tumour necrosis factor-α processing by a metalloproteinase inhibitor
McGeehan, Gerard M, Becherer, J. David, Bast, Robert C, Boyer, Cinda M, Champion, Brian, Connolly, Kevin M, Conway, James G, Furdon, Paul, Karp, Stephen, Kidao, Sudha, McElroy, Andrew B, Nichols, James, Pryzwansky, Katherine M, Schoenen, Frank, Sekut, Les, Truesdale, Anne, Verghese, Margrith, Warner, Janet, Ways, Judy P
Published in Nature (London) (18.08.1994)
Published in Nature (London) (18.08.1994)
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Journal Article
A canine model for determination of the therapeutic index of cytokine inhibitors
Sekut, L. (BASF Bioresearch Corp., Worcester, MA.), Han, B, Baer, P, Verghese, M.W, Silverstein, R, Clifton, L, Dennis, S, Numerick, M.J, Connolly, K.M
Published in Laboratory animal science (Chicago) (01.12.1995)
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Published in Laboratory animal science (Chicago) (01.12.1995)
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Pharmacokinetics and Immunological Effects of Exogenously Administered Recombinant Human B Lymphocyte Stimulator (BLyS) in Mice
Parry, T J, Riccobene, T A, Strawn, S J, Williams, R, Daoud, R, Carrell, J, Sosnovtseva, S, Miceli, R C, Poortman, C M, Sekut, L, Li, Y, Fikes, J, Sung, C
Published in The Journal of pharmacology and experimental therapeutics (01.02.2001)
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Published in The Journal of pharmacology and experimental therapeutics (01.02.2001)
Journal Article
Generation and characterization of LymphoStat‐B, a human monoclonal antibody that antagonizes the bioactivities of B lymphocyte stimulator
Baker, Kevin P., Edwards, Bryan M., Main, Sarah H., Choi, Gil H., Wager, Ruth E., Halpern, Wendy G., Lappin, Patrick B., Riccobene, Todd, Abramian, Donara, Sekut, Les, Sturm, Bonnie, Poortman, Carol, Minter, Ralph R., Dobson, Claire L., Williams, Elizabeth, Carmen, Sara, Smith, Rodger, Roschke, Viktor, Hilbert, David M., Vaughan, Tristan J., Albert, Vivian R.
Published in Arthritis and rheumatism (01.11.2003)
Published in Arthritis and rheumatism (01.11.2003)
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Journal Article
Phosphodiesterase Type IV Inhibition. Structure-Activity Relationships of 1,3-Disubstituted Pyrrolidines
Feldman, Paul L, Brackeen, Marcus F, Cowan, David J, Marron, Brian E, Schoenen, Frank J, Stafford, Jeffrey A, Suh, Edward M, Domanico, Paul L, Rose, Dudley
Published in Journal of medicinal chemistry (01.04.1995)
Published in Journal of medicinal chemistry (01.04.1995)
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Journal Article
Introduction of a conformational switching element on a pyrrolidine ring. Synthesis and evaluation of methyl (R,R)-(.+-.)-3-acetyl-4-[3- (cyclopentyloxy)-4-methoxyphenyl]-3- methyl-1-pyrrolidinecarboxylate, a potent and selective inhibitor of cAMP-specific phosphodiesterase
Stafford, Jeffrey A, Veal, James M, Feldman, Paul L, Valvano, Nicole L, Baer, Philip G, Brackeen, Marcus F, Brawley, E. Sloan, Connolly, Kevin M, Domanico, Paul L
Published in Journal of medicinal chemistry (01.12.1995)
Published in Journal of medicinal chemistry (01.12.1995)
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Journal Article
Evaluation of the significance of elevated levels of systemic and localized tumor necrosis factor in different animal models of inflammation
Sekut, L, Menius, Jr, J A, Brackeen, M F, Connolly, K M
Published in The Journal of laboratory and clinical medicine (01.12.1994)
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Published in The Journal of laboratory and clinical medicine (01.12.1994)
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