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Gong, Yong, Barbay, J. Kent, Dyatkin, Alexey B, Miskowski, Tamara A, Kimball, Edward S, Prouty, Stephen M, Fisher, M. Carolyn, Santulli, Rosemary J, Schneider, Craig R, Wallace, Nathaniel H, Ballentine, Scott A, Hageman, William E, Masucci, John A, Maryanoff, Bruce E, Damiano, Bruce P, Andrade-Gordon, Patricia, Hlasta, Dennis J, Hornby, Pamela J, He, Wei
Published in Journal of medicinal chemistry (01.06.2006)
Published in Journal of medicinal chemistry (01.06.2006)
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Selection of a 2-azabicyclo[2.2.2]octane-based α4β1 integrin antagonist as an inhaled anti-asthmatic agent
LAWSON, Edward C, SANTULLI, Rosemary J, MARYANOFF, Bruce E, DYATKIN, Alexey B, BALLENTINE, Scott A, ABRAHAM, William M, RUDMAN, Sandra, PAGE, Clive P, DE GARAVILLA, Lawrence, DAMIANO, Bruce P, KINNEY, William A
Published in Bioorganic & medicinal chemistry (01.06.2006)
Published in Bioorganic & medicinal chemistry (01.06.2006)
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Process Development for Scale-Up of a Novel 3,5-Substituted Thiazolidine-2,4-dione Compound as a Potent Inhibitor for Estrogen-Related Receptor 1
Li, Xun, Russell, Ronald K, Spink, Jan, Ballentine, Scott, Teleha, Christopher, Branum, Shawn, Wells, Kenneth, Beauchamp, Derek, Patch, Raymond, Huang, Hui, Player, Mark, Murray, William
Published in Organic process research & development (21.02.2014)
Published in Organic process research & development (21.02.2014)
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Synthesis of Mavatrep: A Potent Antagonist of Transient Receptor Potential Vanilloid‑1
Wells, Kenneth M, Mehrman, Steven J, Abdel-Magid, Ahmed F, Ferraro, Caterina, Scott, Lorraine, Zhong, Hua Marlon, Teleha, Christopher A, Ballentine, Scott, Li, Xun, Russell, Ronald K, Spink, Jan M, Diamond, Craig, Youells, Scott, Zhang, Yongzheng, Tsay, Fuh-Rong, Cesco-Cancia, Sergio, Manzo, Stephen M, Beauchamp, Derek A
Published in Organic process research & development (20.11.2015)
Published in Organic process research & development (20.11.2015)
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Synthesis and biological evaluation of novel pyridazinone-based alpha(4) integrin receptor antagonists
Gong, Yong, Barbay, J. Kent, Dyatkin, Alexey B., Miskowski, Tamara A., Kimball, Edward S., Prouty, Stephen M., Fisher, M. Carolyn, Santulli, Rosemary J., Schneider, Craig R., Wallace, Nathaniel H., Ballentine, Scott A., Hageman, William E., Masucci, John A., Maryanoff, Bruce E., Damiano, Bruce P., Andrade-Gordon, Patricia, Hlasta, Dennis J., Hornby, Pamela J., He, Wei
Published in Journal of medicinal chemistry (01.06.2006)
Published in Journal of medicinal chemistry (01.06.2006)
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Suzuki-Miyaura approach to JNJ-26076713, an orally active tetrahydroquinoline-containing alpha(V)beta(3)/alpha(V)beta(5) integrin antagonist. Enantioselective synthesis and stereochemical studies
Kinney, William A., Teleha, Christopher A., Thompson, Andrew S., Newport, Maria, Hansen, Ryan, Ballentine, Scott, Ghosh, Shyamali, Mahan, Andrew, Grasa, Gabriela, Zanotti-Gerosa, Antonio, Dingenen, Jules, Schubert, Carsten, Zhou, Yong, Leo, Gregory C., McComsey, David F., Santulli, Rosemary J., Maryanoff, Bruce E.
Published in Journal of organic chemistry (21.03.2008)
Published in Journal of organic chemistry (21.03.2008)
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Suzuki−Miyaura Approach to JNJ-26076713, an Orally Active Tetrahydroquinoline-Containing αVβ3/αVβ5 Integrin Antagonist. Enantioselective Synthesis and Stereochemical Studies
Kinney, William A, Teleha, Christopher A, Thompson, Andrew S, Newport, Maria, Hansen, Ryan, Ballentine, Scott, Ghosh, Shyamali, Mahan, Andrew, Grasa, Gabriela, Zanotti-Gerosa, Antonio, Dingenen, Jules, Schubert, Carsten, Zhou, Yong, Leo, Gregory C, McComsey, David F, Santulli, Rosemary J, Maryanoff, Bruce E
Published in Journal of organic chemistry (21.03.2008)
Published in Journal of organic chemistry (21.03.2008)
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Regio- and diastereoselective ring-opening of (S)-(−)-2-(trifluoromethyl)oxirane with chiral 2,5-disubstituted tetrahydroquinolines in hexafluoro-2-propanol
Li, Xun, Russell, Ronald K, Chen, Hongfeng, Zhang, Yongzheng, Ballentine, Scott, Spink, Jan, Branum, Shawn, Liu, Fuqiang, Chen, Yanping, Rammeloo, Thomas, Aelterman, Wim, Sorgi, Kirk L, Murray, William V
Published in Green chemistry : an international journal and green chemistry resource : GC (01.01.2010)
Published in Green chemistry : an international journal and green chemistry resource : GC (01.01.2010)
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Suzuki-Miyaura approach to JNJ-26076713, an orally active tetrahydroquinoline-containing alphaVbeta3/alphaVbeta5 integrin antagonist. enantioselective synthesis and stereochemical studies
Kinney, William A, Teleha, Christopher A, Thompson, Andrew S, Newport, Maria, Hansen, Ryan, Ballentine, Scott, Ghosh, Shyamali, Mahan, Andrew, Grasa, Gabriela, Zanotti-Gerosa, Antonio, Dingenen, Jules, Schubert, Carsten, Zhou, Yong, Leo, Gregory C, McComsey, David F, Santulli, Rosemary J, Maryanoff, Bruce E
Published in Journal of organic chemistry (21.03.2008)
Published in Journal of organic chemistry (21.03.2008)
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Suzuki−Miyaura Approach to JNJ-26076713, an Orally Active Tetrahydroquinoline-Containing α V β 3 /α V β 5 Integrin Antagonist. Enantioselective Synthesis and Stereochemical Studies
Kinney, William A., Teleha, Christopher A., Thompson, Andrew S., Newport, Maria, Hansen, Ryan, Ballentine, Scott, Ghosh, Shyamali, Mahan, Andrew, Grasa, Gabriela, Zanotti-Gerosa, Antonio, Dingenen, Jules, Schubert, Carsten, Zhou, Yong, Leo, Gregory C., McComsey, David F., Santulli, Rosemary J., Maryanoff, Bruce E.
Published in Journal of organic chemistry (01.03.2008)
Published in Journal of organic chemistry (01.03.2008)
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Journal Article
Suzuki-Miyaura Approach to JNJ-26076713, an Orally Active Tetrahydroquinoline-Containing αVβ3αVβ5 Integrin Antagonist. Enantioselective Synthesis and Stereochemical Studies
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Published in Journal of organic chemistry (2008)
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Published in Journal of organic chemistry (2008)
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