Superagonist, Full Agonist, Partial Agonist, and Antagonist Actions of Arylguanidines at 5‑Hydroxytryptamine‑3 (5-HT3) Subunit A Receptors
Alix, Katie, Khatri, Shailesh, Mosier, Philip D, Casterlow, Samantha, Yan, Dong, Nyce, Heather L, White, Michael M, Schulte, Marvin K, Dukat, Małgorzata
Published in ACS chemical neuroscience (16.11.2016)
Published in ACS chemical neuroscience (16.11.2016)
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Journal Article
Deconstruction of the α4β2 Nicotinic Acetylcholine Receptor Positive Allosteric Modulator Desformylflustrabromine
German, Nadezhda, Kim, Jin-Sung, Jain, Atul, Dukat, Malgorzata, Pandya, Anshul, Ma, Yilong, Weltzin, Maegan, Schulte, Marvin K, Glennon, Richard A
Published in Journal of medicinal chemistry (27.10.2011)
Published in Journal of medicinal chemistry (27.10.2011)
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Journal Article
Rabies virus modifies host behaviour through a snake-toxin like region of its glycoprotein that inhibits neurotransmitter receptors in the CNS
Hueffer, Karsten, Khatri, Shailesh, Rideout, Shane, Harris, Michael B, Papke, Roger L, Stokes, Clare, Schulte, Marvin K
Published in Scientific reports (09.10.2017)
Published in Scientific reports (09.10.2017)
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Journal Article
Desformylflustrabromine (dFBr), a positive allosteric modulator of the α4β2 nicotinic receptor modulates the hypnotic response to ethanol
DeCristofano, Laura, Decker, Steven, Schulte, Marvin K., Suryanarayanan, Asha
Published in Alcohol (Fayetteville, N.Y.) (01.06.2021)
Published in Alcohol (Fayetteville, N.Y.) (01.06.2021)
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Journal Article
Improved Surface Modification Approach for Micromechanical Biosensors
Gao, Hongyan, Buchapudi, Koutilya R, Harms-Smyth, Abraham, Schulte, Marvin K, Xu, Xiaohe, Ji, Hai-Feng
Published in Langmuir (15.01.2008)
Published in Langmuir (15.01.2008)
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Journal Article
Multi-modal antidepressant-like action of 6- and 7-chloro-2-aminodihydroquinazolines in the mouse tail suspension test
Iyer, Kavita A., Alix, Katie, Eltit, Jose M., Solis, Ernesto, Pan, Xiaolei, Argade, Malaika D., Khatri, Shailesh, De Felice, Louis J., Sweet, Douglas H., Schulte, Marvin K., Dukat, Małgorzata
Published in Psychopharmacology (01.07.2019)
Published in Psychopharmacology (01.07.2019)
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Journal Article
N1H- and N1‑Substituted Phenylguanidines as α7 Nicotinic Acetylcholine (nACh) Receptor Antagonists: Structure–Activity Relationship Studies
Alwassil, Osama I, Khatri, Shailesh, Schulte, Marvin K, Aripaka, Sanjay S, Mikkelsen, Jens D, Dukat, Małgorzata
Published in ACS chemical neuroscience (16.06.2021)
Published in ACS chemical neuroscience (16.06.2021)
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Journal Article
Allosteric modulation of alpha4beta2 nicotinic acetylcholine receptors by HEPES
Weltzin, Maegan M., Huang, Yanzhou, Schulte, Marvin K.
Published in European journal of pharmacology (05.06.2014)
Published in European journal of pharmacology (05.06.2014)
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Journal Article
Desformylflustrabromine Modulates α4β2 Neuronal Nicotinic Acetylcholine Receptor High- and Low-Sensitivity Isoforms at Allosteric Clefts Containing the β2 Subunit
Weltzin, Maegan M, Schulte, Marvin K
Published in The Journal of pharmacology and experimental therapeutics (01.08.2015)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2015)
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Journal Article
Attenuation of Compulsive-Like Behavior Through Positive Allosteric Modulation of α4β2 Nicotinic Acetylcholine Receptors in Non-Induced Compulsive-Like Mice
Mitra, Swarup, Mucha, Mckenzie, Khatri, Shailesh N, Glenon, Richard, Schulte, Marvin K, Bult-Ito, Abel
Published in Frontiers in behavioral neuroscience (05.01.2017)
Published in Frontiers in behavioral neuroscience (05.01.2017)
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Journal Article
des-Formylflustrabromine (dFBr): A Structure–Activity Study on Its Ability To Potentiate the Action of Acetylcholine at α4β2 Nicotinic Acetylcholine Receptors
Dukat, Małgorzata, Jain, Atul, German, Nadezhda, Ferrara-Pontoriero, Rossana, Huang, Yanzhou, Ma, Yilong, Schulte, Marvin K, Glennon, Richard A
Published in ACS chemical neuroscience (19.12.2018)
Published in ACS chemical neuroscience (19.12.2018)
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Journal Article
Evaluation of galantamine and deconstructed analogs as α7 nAChR and AChE ligands
Argade, Malaika D., DeCristofano, Laura, Bhattarai, Nirajan, Schulte, Marvin K., Dukat, Malgorzata
Published in Results in Chemistry (01.01.2022)
Published in Results in Chemistry (01.01.2022)
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Journal Article
“Methylene Bridge” to 5‑HT3 Receptor Antagonists: Conformationally Constrained Phenylguanidines
Abdelkhalek, Ahmed S, Alley, Genevieve S, Alwassil, Osama I, Khatri, Shailesh, Mosier, Philip D, Nyce, Heather L, White, Michael M, Schulte, Marvin K, Dukat, Małgorzata
Published in ACS chemical neuroscience (20.03.2019)
Published in ACS chemical neuroscience (20.03.2019)
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Journal Article
"Methylene Bridge" to 5-HT 3 Receptor Antagonists: Conformationally Constrained Phenylguanidines
Abdelkhalek, Ahmed S, Alley, Genevieve S, Alwassil, Osama I, Khatri, Shailesh, Mosier, Philip D, Nyce, Heather L, White, Michael M, Schulte, Marvin K, Dukat, Małgorzata
Published in ACS chemical neuroscience (20.03.2019)
Published in ACS chemical neuroscience (20.03.2019)
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Journal Article
Synthesis of desformylflustrabromine and its evaluation as an alpha 4 beta 2 and alpha 7 nACh receptor modulator
Kim, Jin-Sung, Padnya, Anshul, Weltzin, Maegan, Edmonds, Brian W, Schulte, Marvin K, Glennon, Richard A
Published in Bioorganic & medicinal chemistry letters (01.09.2007)
Published in Bioorganic & medicinal chemistry letters (01.09.2007)
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Journal Article
Synthesis of desformylflustrabromine and its evaluation as an α4β2 and α7 nACh receptor modulator
Kim, Jin-Sung, Padnya, Anshul, Weltzin, Maegan, Edmonds, Brian W., Schulte, Marvin K., Glennon, Richard A.
Published in Bioorganic & medicinal chemistry letters (01.09.2007)
Published in Bioorganic & medicinal chemistry letters (01.09.2007)
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Journal Article
Microcantilever biosensors based on conformational change of proteins
JI, Hai-Feng, HONGYAN GAO, BUCHAPUDI, Koutilya R, XIN YANG, XIAOHE XU, SCHULTE, Marvin K
Published in Analyst (London) (01.04.2008)
Published in Analyst (London) (01.04.2008)
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Journal Article
A comprehensive study on the 5-hydroxytryptamine3A receptor binding of agonists serotonin and m-chlorophenylbiguanidine
HAZAI, Eszter, JOSHI, Prasad, SKOVIAK, Edward C, SURYANARAYANAN, Asha, SCHULTE, Marvin K, BIKADI, Zsolt
Published in Bioorganic & medicinal chemistry (15.08.2009)
Published in Bioorganic & medicinal chemistry (15.08.2009)
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