Synthesis Development of the Selective Estrogen Receptor Degrader (SERD) LSZ102 from a Suzuki Coupling to a C–H Activation Strategy
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Published in Organic process research & development (21.08.2020)
Published in Organic process research & development (21.08.2020)
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Development of a cyclosporin A derivative with excellent anti-hepatitis C virus potency
Fu, Jiping, Becker, Christopher, Cao, Li, Capparelli, Michael, Denay, Regis, Fujimoto, Roger, Gai, Yu, Gao, Zhaobo, Guenat, Christian, Karur, Subramanian, Kim, Hongyong, Li, Weikuan, Li, Xiaolin, Li, Wei, Lochmann, Thomas, Lu, Amy, Lu, Peichao, Luneau, Alexandre, Meier, Nicole, Mergo, Wosenu, Ng, Simon, Parker, David, Peng, Yunshan, Riss, Bernard, Rivkin, Alexey, Roggo, Silvio, Schroeder, Harald, Schuerch, Friedrich, Simmons, Robert L., Sun, Feng, Sweeney, Zachary K., Tjandra, Meiliana, Wang, Michael, Wang, Ruidong, Weiss, Andrew H., Wenger, Nicolas, Wu, Quanbing, Xiong, Xin, Xu, Su, Xu, Wenjian, Yifru, Aregahegn, Zhao, Jibin, Zhou, Jianguang, Zürcher, Christian, Gallou, Fabrice
Published in Bioorganic & medicinal chemistry (15.02.2018)
Published in Bioorganic & medicinal chemistry (15.02.2018)
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The identification of 7-[(R)-2-((1S,2S)-2-benzyloxycyclopentylamino)-1-hydroxyethyl]-4-hydroxybenzothiazolone as an inhaled long-acting β2-adrenoceptor agonist
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Published in Bioorganic & medicinal chemistry letters (01.09.2014)
Published in Bioorganic & medicinal chemistry letters (01.09.2014)
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Journal Article
The identification of 7-[(R)-2-((1S,2S)-2-benzyloxycyclopentylamino)-1-hydroxyethyl]-4-hydroxybenzothiazolone as an inhaled long-acting beta(2)-adrenoceptor agonist
Arnold, Nicola, Beattie, David, Bradley, Michelle, Brearley, Andrew, Brown, Lyndon, Charlton, Steven J., Fairhurst, Robin A., Farr, David, Fozard, John, Fullerton, Joe, Gosling, Martin, Hatto, Julia, Janus, Diana, Jones, Darryl, Jordan, Lynne, Lewis, Christine, Maas, Janet, McCarthy, Clive, Mercer, Mark, Oakman, Helen, Press, Neil, Profit, Rachel, Schuerch, Friedrich, Sykes, David, Taylor, Roger J., Trifilieff, Alexandre, Tuffnell, Andrew
Published in Bioorganic & medicinal chemistry letters (01.09.2014)
Published in Bioorganic & medicinal chemistry letters (01.09.2014)
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Large-Scale Synthesis of the Anti-Cancer Marine Natural Product (+)-Discodermolide. Part 3: Synthesis of Fragment C15 - 21
Mickel, Stuart J, Sedelmeier, Gottfried H, Niederer, Daniel, Schuerch, Friedrich, Koch, Guido, Kuesters, E, Daeffler, Robert, Osmani, Adnan, Seeger-Weibel, Manuela, Schmid, E, Hirni, Alfred, Schaer, Karl, Gamboni, Remo, Bach, Andrew, Chen, Stephen, Chen, Weichun, Geng, Peng, Jagoe, Christopher T, Kinder, Frederick R, Lee, George T, McKenna, Joseph, Ramsey, Timothy M, Repič, Oljan, Rogers, Larry, Shieh, Wen-Chung, Wang, Run-Ming, Waykole, Liladhar
Published in Organic process research & development (01.01.2004)
Published in Organic process research & development (01.01.2004)
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Large-Scale Synthesis of the Anti-Cancer Marine Natural Product (+)-Discodermolide. Part 4: Preparation of Fragment C7 - 24
Mickel, Stuart J, Sedelmeier, Gottfried H, Niederer, Daniel, Schuerch, Friedrich, Seger, Manuela, Schreiner, Klaus, Daeffler, Robert, Osmani, Adnan, Bixel, Dominique, Loiseleur, Olivier, Cercus, Jacques, Stettler, Hans, Schaer, Karl, Gamboni, Remo, Bach, Andrew, Chen, Guang-Pei, Chen, Weichun, Geng, Peng, Lee, George T, Loeser, Eric, McKenna, Joseph, Kinder, Frederick R, Konigsberger, Kurt, Prasad, Kapa, Ramsey, Timothy M, Reel, Noela, Repič, Oljan, Rogers, Larry, Shieh, Wen-Chung, Wang, Run-Ming, Waykole, Liladhar, Xue, Song, Florence, Gordon, Paterson, Ian
Published in Organic process research & development (01.01.2004)
Published in Organic process research & development (01.01.2004)
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Large-Scale Synthesis of the Anti-Cancer Marine Natural Product (+)-Discodermolide. Part 2: Synthesis of Fragments C1 - 6 and C9-14
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Published in Organic process research & development (16.01.2004)
Published in Organic process research & development (16.01.2004)
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Journal Article
Large-Scale Synthesis of the Anti-Cancer Marine Natural Product (+)-Discodermolide. Part 3: Synthesis of Fragment C 15 - 21
Mickel, Stuart J., Sedelmeier, Gottfried H., Niederer, Daniel, Schuerch, Friedrich, Koch, Guido, Kuesters, E., Daeffler, Robert, Osmani, Adnan, Seeger-Weibel, Manuela, Schmid, E., Hirni, Alfred, Schaer, Karl, Gamboni, Remo, Bach, Andrew, Chen, Stephen, Chen, Weichun, Geng, Peng, Jagoe, Christopher T., Kinder, Frederick R., Lee, George T., McKenna, Joseph, Ramsey, Timothy M., Repič, Oljan, Rogers, Larry, Shieh, Wen-Chung, Wang, Run-Ming, Waykole, Liladhar
Published in Organic process research & development (01.01.2004)
Published in Organic process research & development (01.01.2004)
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Large-Scale Synthesis of the Anti-Cancer Marine Natural Product (+)-Discodermolide. Part 2: Synthesis of Fragments C 1 - 6 and C 9-14
Mickel, Stuart J., Sedelmeier, Gottfried H., Niederer, Daniel, Schuerch, Friedrich, Grimler, Dominique, Koch, Guido, Daeffler, Robert, Osmani, Adnan, Hirni, Alfred, Schaer, Karl, Gamboni, Remo, Bach, Andrew, Chaudhary, Apurva, Chen, Stephen, Chen, Weichun, Hu, Bin, Jagoe, Christopher T., Kim, Hong-Yong, Kinder, Frederick R., Liu, Yugang, Lu, Yansong, McKenna, Joseph, Prashad, Mahavir, Ramsey, Timothy M., Repič, Oljan, Rogers, Larry, Shieh, Wen-Chung, Wang, Run-Ming, Waykole, Liladhar
Published in Organic process research & development (01.01.2004)
Published in Organic process research & development (01.01.2004)
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Large-Scale Synthesis of the Anti-Cancer Marine Natural Product (+)-Discodermolide. Part 4: Preparation of Fragment C 7 - 24
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Published in Organic process research & development (01.01.2004)
Published in Organic process research & development (01.01.2004)
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Year of Publication 26.04.2016
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Year of Publication 26.04.2016
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Year of Publication 25.03.2015
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Year of Publication 04.09.2012
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Year of Publication 04.09.2012
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KING JONATHAN, PRASHAD MAHAVIR, BOLLINGER PIETRO, SCHMID VINCENT, SCHUERCH FRIEDRICH, HIESTAND PETER C, DAWSON KING JANET, LIU YUGANG, RISS BERNHARD
Year of Publication 04.09.2012
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Year of Publication 04.09.2012
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Organic compounds which are aza-thia-benzoazulene derivatives
RISS, BERNHARD, KING, JONATHAN, LIU, YUGANG, BOLLINGER, PIETRO, PRASHAD, MAHAVIR, SCHMID, VINCENT, DAWSON KING, JANET, SCHUERCH, FRIEDRICH, HIESTAND, PETER C
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Year of Publication 30.06.2011
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BERNHARD RISS, JONATHAN KING, FRIEDRICH SCHUERCH, PETER C. HIESTAND, JANET DAWSON KING, YUGANG LIU, MAHAVIR PRASHAD, VINCENT SCHMID, PIETRO BOLLINGER
Year of Publication 10.02.2011
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Year of Publication 18.11.2010
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Year of Publication 18.11.2010
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RISS, BERNHARD, KING, JONATHAN, LIU, YUGANG, BOLLINGER, PIETRO, PRASHAD, MAHAVIR, SCHMID, VINCENT, DAWSON KING, JANET, SCHUERCH, FRIEDRICH, HIESTAND, PETER C
Year of Publication 28.10.2009
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Year of Publication 28.10.2009
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Organic Compounds
KING JONATHAN, PRASHAD MAHAVIR, BOLLINGER PIETRO, SCHMID VINCENT, SCHUERCH FRIEDRICH, HIESTAND PETER C, DAWSON KING JANET, LIU YUGANG, RISS BERNHARD
Year of Publication 21.05.2009
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Year of Publication 21.05.2009
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KING JONATHAN, PRASHAD MAHAVIR, BOLLINGER PIETRO, SCHMID VINCENT, SCHUERCH FRIEDRICH, HIESTAND PETER C, DAWSON KING JANET, LIU YUGANG, RISS BERNHARD
Year of Publication 08.12.2008
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Year of Publication 08.12.2008
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