Discovery of 6-N,N-Bis(2,2,2-trifluoroethyl)amino- 4-trifluoromethylquinolin-2(1H)-one as a Novel Selective Androgen Receptor Modulator
van Oeveren, Arjan, Motamedi, Mehrnouch, Mani, Neelakandha S, Marschke, Keith B, López, Francisco J, Schrader, William T, Negro-Vilar, Andrés, Zhi, Lin
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Published in Journal of medicinal chemistry (19.10.2006)
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William R. Brinkley: A giant in biomedical research and public policy
Gerbi, Susan A., Palazzo, Robert E., Earnshaw, William C., Schrader, William T.
Published in The Journal of cell biology (04.10.2021)
Published in The Journal of cell biology (04.10.2021)
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Regulation of progesterone receptor-mediated transcription by phosphorylation
Denner, L.A. (Baylor College of Medicine, Houston, TX), Weigel, N.L, Maxwell, B.L, Schrader, W.T, O'Malley, B.W
Published in Science (American Association for the Advancement of Science) (21.12.1990)
Published in Science (American Association for the Advancement of Science) (21.12.1990)
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Synthesis and biological activity of 5-methylidene 1,2-dihydrochromeno[3,4- f]quinoline derivatives as progesterone receptor modulators
Zhi, Lin, Tegley, Christopher M, Pio, Barbara, Edwards, James P, Jones, Todd K, Marschke, Keith B, Mais, Dale E, Risek, Boris, Schrader, William T
Published in Bioorganic & medicinal chemistry letters (16.06.2003)
Published in Bioorganic & medicinal chemistry letters (16.06.2003)
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Preparation, Resolution, and Biological Evaluation of 5-Aryl-1,2-dihydro-5H-chromeno[3,4-f]quinolines: Potent, Orally Active, Nonsteroidal Progesterone Receptor Agonists
Edwards, James P, Zhi, Lin, Pooley, Charlotte L. F, Tegley, Christopher M, West, Sarah J, Wang, Ming-Wei, Gottardis, Marco M, Pathirana, Charles, Schrader, William T, Jones, Todd K
Published in Journal of medicinal chemistry (16.07.1998)
Published in Journal of medicinal chemistry (16.07.1998)
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Differential Hormone-Dependent Phosphorylation of Progesterone Receptor A and B Forms Revealed by a Phosphoserine Site-Specific Monoclonal Antibody
Clemm, David L, Sherman, Lori, Boonyaratanakornkit, Viroj, Schrader, William T, Weigel, Nancy L, Edwards, Dean P
Published in Molecular endocrinology (Baltimore, Md.) (01.01.2000)
Published in Molecular endocrinology (Baltimore, Md.) (01.01.2000)
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Novel Series of Potent, Nonsteroidal, Selective Androgen Receptor Modulators Based on 7H-[1,4]Oxazino[3,2-g]quinolin-7-ones
Higuchi, Robert I, Arienti, Kristen L, López, Francisco J, Mani, Neelakhanda S, Mais, Dale E, Caferro, Thomas R, Long, Yun Oliver, Jones, Todd K, Edwards, James P, Zhi, Lin, Schrader, William T, Negro-Vilar, Andrés, Marschke, Keith B
Published in Journal of medicinal chemistry (17.05.2007)
Published in Journal of medicinal chemistry (17.05.2007)
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Photocytotoxicity of the Fluorescent Nonsteroidal Androgen Receptor Ligand TDPQ
Bilski, Piotr J., Risek, Boris, Chignell, Colin F., Schrader, William T.
Published in Photochemistry and photobiology (01.09.2009)
Published in Photochemistry and photobiology (01.09.2009)
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5-Benzylidene-1,2-dihydrochromeno[3,4-f]quinolines as Selective Progesterone Receptor Modulators
Zhi, Lin, Tegley, Christopher M, Pio, Barbara, Edwards, James P, Motamedi, Mehrnouch, Jones, Todd K, Marschke, Keith B, Mais, Dale E, Risek, Boris, Schrader, William T
Published in Journal of medicinal chemistry (11.09.2003)
Published in Journal of medicinal chemistry (11.09.2003)
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Potent, nonsteroidal selective androgen receptor modulators (SARMs) based on 8H-[1,4 ]oxazino [2,3 -f] quinolin-8-ones
HIGUCHI, Robert I, THOMPSON, Anthony W, ADAM KALLEL, E, KARANEWSKY, Donald S, SCHRADER, William T, MARSCHKE, Keith B, LIN ZHI, CHEN, Jyun-Hung, CAFERRO, Thomas R, CUMMINGS, Marquis L, DECKHUT, Charlotte P, ADAMS, Mark E, TEGLEY, Christopher M, EDWARDS, James P, LOPEZ, Francisco J
Published in Bioorganic & medicinal chemistry letters (01.10.2007)
Published in Bioorganic & medicinal chemistry letters (01.10.2007)
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The mechanism of RU486 antagonism is dependent on the conformation of the carboxy-terminal tail of the human progesterone receptor
Vegeto, Elisabetta, Allan, George F., Schrader, William T., Tsai, Ming-Jer, McDonnell, Donald P., O'Malley, Bert W.
Published in Cell (15.05.1992)
Published in Cell (15.05.1992)
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Development of progesterone receptor antagonists from 1,2-dihydrochromeno[3,4- f]quinoline agonist pharmacophore
Zhi, Lin, Ringgenberg, Josef D, Edwards, James P, Tegley, Christopher M, West, Sarah J, Pio, Barbara, Motamedi, Mehrnouch, Jones, Todd K, Marschke, Keith B, Mais, Dale E, Schrader, William T
Published in Bioorganic & medicinal chemistry letters (16.06.2003)
Published in Bioorganic & medicinal chemistry letters (16.06.2003)
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Progesterone-binding components of chick oviduct: partial purification and characterization of a calcium-activated protease which hydrolyzes the progesterone receptor
Vedeckis, Wayne V, Freeman, Marinan R, Schrader, William T, O'Malley, Bert W
Published in Biochemistry (Easton) (22.01.1980)
Published in Biochemistry (Easton) (22.01.1980)
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The A and B forms of the chicken progesterone receptor arise by alternate initiation of translation of a unique mRNA
Conneely, Orla M., Maxwell, Beth Lynn, Toft, David O., Schrader, William T., O'Malley, Bert W.
Published in Biochemical and biophysical research communications (16.12.1987)
Published in Biochemical and biophysical research communications (16.12.1987)
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Molecular cloning of the chicken progesterone receptor
Conneely, O.M, Sullivan, W.P, Toft, D.O, Birnbaumer, M, Cook, R.G, Maxwell, B.L, Zarucki-Schulz, T, Greene, G.L, Schrader, W.T, O'Malley, B.W
Published in Science (American Association for the Advancement of Science) (15.08.1986)
Published in Science (American Association for the Advancement of Science) (15.08.1986)
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Chicken progesterone receptor expressed in Saccharomyces cerevisiae is correctly phosphorylated at all four Ser-Pro phosphorylation sites
Poletti, Angelo, Conneely, Orla M, McDonnell, Donald P, Schrader, William T, O'Malley, Bert W, Weigel, Nancy L
Published in Biochemistry (Easton) (21.09.1993)
Published in Biochemistry (Easton) (21.09.1993)
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