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Substituted 2H-isoquinolin-1-ones as potent Rho-kinase inhibitors: Part 3, aryl substituted pyrrolidines
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Published in Bioorganic & medicinal chemistry letters (15.06.2010)
Published in Bioorganic & medicinal chemistry letters (15.06.2010)
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Journal Article
Agonist activation of the G protein-coupled receptor GPR35 involves transmembrane domain III and is transduced via G[alpha]13 and [beta]-arrestin-2
Jenkins, Laura, Alvarez-Curto, Elisa, Campbell, Kate, de Munnik, Sabrina, Canals, Meritxell, Schlyer, Sabine, Milligan, Graeme
Published in British journal of pharmacology (01.02.2011)
Published in British journal of pharmacology (01.02.2011)
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Journal Article
Agonist activation of the G protein‐coupled receptor GPR35 involves transmembrane domain III and is transduced via Gα13 and β‐arrestin‐2
Jenkins, Laura, Alvarez‐Curto, Elisa, Campbell, Kate, de Munnik, Sabrina, Canals, Meritxell, Schlyer, Sabine, Milligan, Graeme
Published in British journal of pharmacology (01.02.2011)
Published in British journal of pharmacology (01.02.2011)
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SAR studies of non-zinc-chelating MMP-13 inhibitors: Improving selectivity and metabolic stability
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Published in Bioorganic & medicinal chemistry letters (01.09.2010)
Published in Bioorganic & medicinal chemistry letters (01.09.2010)
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Substituted 2 H-isoquinolin-1-ones as potent Rho-kinase inhibitors: Part 2, optimization for blood pressure reduction in spontaneously hypertensive rats
Ginn, John D., Bosanac, Todd, Chen, Rhonda, Cywin, Charles, Hickey, Eugene, Kashem, Mohammed, Kerr, Steven, Kugler, Stanley, Li, Xiang, Prokopowicz, Anthony, Schlyer, Sabine, Smith, James D., Turner, Michael R., Wu, Frank, Young, Erick R.R.
Published in Bioorganic & medicinal chemistry letters (2010)
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Published in Bioorganic & medicinal chemistry letters (15.07.2008)
Published in Bioorganic & medicinal chemistry letters (15.07.2008)
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Synthesis of N-alkyl glycine amides as potent inhibitors of leukotriene A sub(4) hydrolase
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Published in Bioorganic & medicinal chemistry (01.07.2008)
Published in Bioorganic & medicinal chemistry (01.07.2008)
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Synthesis of N-alkyl glycine amides as potent inhibitors of leukotriene A 4 hydrolase
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Published in Bioorganic & medicinal chemistry letters (2008)
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Year of Publication 21.04.2020
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Year of Publication 10.04.2019
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Year of Publication 06.12.2018
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Year of Publication 12.07.2017
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