Novel 3-Arylideneindolin-2-ones as Inhibitors of NAD+-Dependent Histone Deacetylases (Sirtuins)
Huber, Kilian, Schemies, Jörg, Uciechowska, Urszula, Wagner, Julia M, Rumpf, Tobias, Lewrick, Felicitas, Süss, Regine, Sippl, Wolfgang, Jung, Manfred, Bracher, Franz
Published in Journal of medicinal chemistry (11.02.2010)
Published in Journal of medicinal chemistry (11.02.2010)
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Structural and Synthetic Investigations of Tanikolide Dimer, a SIRT2 Selective Inhibitor, and Tanikolide seco-Acid from the Madagascar Marine Cyanobacterium Lyngbya majuscula
Gutiérrez, Marcelino, Andrianasolo, Eric H, Shin, Won Kyo, Goeger, Douglas E, Yokochi, Alexandre, Schemies, Jörg, Jung, Manfred, France, Dennis, Cornell-Kennon, Susan, Lee, Eun, Gerwick, William H
Published in Journal of organic chemistry (07.08.2009)
Published in Journal of organic chemistry (07.08.2009)
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Benzodeazaoxaflavins as Sirtuin Inhibitors with Antiproliferative Properties in Cancer Stem Cells
Rotili, Dante, Tarantino, Domenico, Carafa, Vincenzo, Paolini, Chantal, Schemies, Jörg, Jung, Manfred, Botta, Giorgia, Di Maro, Salvatore, Novellino, Ettore, Steinkühler, Christian, De Maria, Ruggero, Gallinari, Paola, Altucci, Lucia, Mai, Antonello
Published in Journal of medicinal chemistry (27.09.2012)
Published in Journal of medicinal chemistry (27.09.2012)
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Two-Step Synthesis of Novel, Bioactive Derivatives of the Ubiquitous Cofactor Nicotinamide Adenine Dinucleotide (NAD)
Pesnot, Thomas, Kempter, Julia, Schemies, Jörg, Pergolizzi, Giulia, Uciechowska, Urszula, Rumpf, Tobias, Sippl, Wolfgang, Jung, Manfred, Wagner, Gerd K
Published in Journal of medicinal chemistry (26.05.2011)
Published in Journal of medicinal chemistry (26.05.2011)
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NAD+-dependent histone deacetylases (sirtuins) as novel therapeutic targets
Schemies, Jörg, Uciechowska, Urszula, Sippl, Wolfgang, Jung, Manfred
Published in Medicinal research reviews (01.11.2010)
Published in Medicinal research reviews (01.11.2010)
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Malyngolide Dimer, a Bioactive Symmetric Cyclodepside from the Panamanian Marine Cyanobacterium Lyngbya majuscula
Gutiérrez, Marcelino, Tidgewell, Kevin, Capson, Todd L, Engene, Niclas, Almanza, Alejandro, Schemies, Jörg, Jung, Manfred, Gerwick, William H
Published in Journal of natural products (Washington, D.C.) (23.04.2010)
Published in Journal of natural products (Washington, D.C.) (23.04.2010)
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Synthesis and biological activity of splitomicin analogs targeted at human NAD +-dependent histone deacetylases (sirtuins)
Freitag, Marcus, Schemies, Jörg, Larsen, Tim, El Gaghlab, Khattab, Schulz, Felix, Rumpf, Tobias, Jung, Manfred, Link, Andreas
Published in Bioorganic & medicinal chemistry (15.06.2011)
Published in Bioorganic & medicinal chemistry (15.06.2011)
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Binding free energy calculations and biological testing of novel thiobarbiturates as inhibitors of the human NAD+ dependent histone deacetylase Sirt2
Uciechowska, Urszula, Schemies, Jörg, Scharfe, Michael, Lawson, Michael, Wichapong, Kanin, Jung, Manfred, Sippl, Wolfgang
Published in MedChemComm (01.02.2012)
Published in MedChemComm (01.02.2012)
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Thiobarbiturates as Sirtuin Inhibitors: Virtual Screening, Free‐Energy Calculations, and Biological Testing
Uciechowska, Urszula, Schemies, Jörg, Neugebauer, Robert C., Huda, Elisabeth‐Maria, Schmitt, Martin L., Meier, Rene, Verdin, Eric, Jung, Manfred, Sippl, Wolfgang
Published in ChemMedChem (15.12.2008)
Published in ChemMedChem (15.12.2008)
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Identification of Tri- and Tetracyclic Pyrimidinediones as Sirtuin Inhibitors
Rotili, Dante, Tarantino, Domenico, Carafa, Vincenzo, Lara, Ester, Meade, Sarah, Botta, Giorgia, Nebbioso, Angela, Schemies, Jörg, Jung, Manfred, Kazantsev, Aleksey G., Esteller, Manel, Fraga, Mario F., Altucci, Lucia, Mai, Antonello
Published in ChemMedChem (03.05.2010)
Published in ChemMedChem (03.05.2010)
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Synthesis and biological activity of splitomicin analogs targeted at human NAD+-dependent histone deacetylases (sirtuins) : Epigenetic drug Discovery
FREITAG, Marcus, SCHEMIES, Jörg, LARSEN, Tim, EL GAGHLAB, Khattab, SCHULZ, Felix, RUMPF, Tobias, JUNG, Manfred, LINK, Andreas
Published in Bioorganic & medicinal chemistry (2011)
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Published in Bioorganic & medicinal chemistry (2011)
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