Inhibitors of HIV Nucleocapsid Protein Zinc Fingers as Candidates for the Treatment of AIDS
Rice, William G., Supko, Jeffrey G., Malspeis, Louis, Buckheit, Robert W., Clanton, David, Bu, Ming, Graham, Lisa, Schaeffer, Catherine A., Turpin, Jim A., Domagala, John, Gogliotti, Rocco, Bader, John P., Halliday, Susan M., Coren, Lori, Sowder, Raymond C., Arthur, Larry O., Henderson, Louis E.
Published in Science (American Association for the Advancement of Science) (17.11.1995)
Published in Science (American Association for the Advancement of Science) (17.11.1995)
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Journal Article
Inhibition of HIV-1 infectivity by zinc-ejecting aromatic C -nitroso compounds
Rice, William G, Schaeffer, Catherine A, Harten, Brad, Villinger, Francois, South, Terri L, Summers, Michael F, Henderson, Louis E, Bess, Julian W, Arthur, Larry O, McDougal, J. Steven, Orloff, Sherry L, Mendeleyev, Jerome, Kun, Ernest
Published in Nature (London) (04.02.1993)
Published in Nature (London) (04.02.1993)
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Journal Article
Inhibition of Acute-, Latent-, and Chronic-Phase Human Immunodeficiency Virus Type 1 (HIV-1) Replication by a Bistriazoloacridone Analog That Selectively Inhibits HIV-1 Transcription
TURPIN, J. A, BUCKHEIT, R. W, MING BU, MINGJUN HUANG, CHOLODY, W. M, MICHEJDA, C. J, RICE, W. G, DERSE, D, HOLLINGSHEAD, M, WILLIAMSON, K, PALAMONE, C, OSTERLING, M. C, HILL, S. A, GRAHAM, L, SCHAEFFER, C. A
Published in Antimicrobial Agents and Chemotherapy (01.03.1998)
Published in Antimicrobial Agents and Chemotherapy (01.03.1998)
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Journal Article
Evaluation of Selected Chemotypes in Coupled Cellular and Molecular Target-Based Screens Identifies Novel HIV-1 Zinc Finger Inhibitors
Rice, William G, Turpin, Jim A, Schaeffer, Catherine A, Graham, Lisa, Clanton, David, Buckheit, Robert W, Zaharevitz, Daniel, Summers, Michael F, Wallqvist, Anders, Covell, David G
Published in Journal of medicinal chemistry (13.09.1996)
Published in Journal of medicinal chemistry (13.09.1996)
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Journal Article
New Alkenyldiarylmethanes with Enhanced Potencies as Anti-HIV Agents Which Act as Non-Nucleoside Reverse Transcriptase Inhibitors
Cushman, Mark, Casimiro-Garcia, Agustin, Hejchman, Elzbieta, Ruell, Jeffrey A, Huang, Mingjun, Schaeffer, Catherine A, Williamson, Karen, Rice, William G, Buckheit, Robert W
Published in Journal of medicinal chemistry (04.06.1998)
Published in Journal of medicinal chemistry (04.06.1998)
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Journal Article
All-Atom Models for the Non-Nucleoside Binding Site of HIV-1 Reverse Transcriptase Complexed with Inhibitors: A 3D QSAR Approach
Gussio, Rick, Pattabiraman, Nagarajan, Zaharevitz, Daniel W, Kellogg, Glen E, Topol, Igor A, Rice, William G, Schaeffer, Catherine A, Erickson, John W, Burt, Stanley K
Published in Journal of medicinal chemistry (12.04.1996)
Published in Journal of medicinal chemistry (12.04.1996)
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Journal Article
The Site of Antiviral Action of 3-Nitrosobenzamide on the Infectivity Process of Human Immunodeficiency Virus in Human Lymphocytes
Rice, William G., Schaeffer, Catherine A., Graham, Lisa, Bu, Ming, McDougal, J. Steven, Orloff, Sherry L., Villinger, Francois, Young, Matthew, Oroszlan, Stephan, Fesen, Mark R., Pommier, Yves, Mendeleyev, Jerome, Kun, Ernest
Published in Proceedings of the National Academy of Sciences - PNAS (15.10.1993)
Published in Proceedings of the National Academy of Sciences - PNAS (15.10.1993)
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Journal Article
Extension of the Polyanionic Cosalane Pharmacophore as a Strategy for Increasing Anti-HIV Potency
Cushman, Mark, Insaf, Shabana, Paul, Gitendra, Ruell, Jeffrey A, De Clercq, Erik, Schols, Dominique, Pannecouque, Christophe, Witvrouw, Myriam, Schaeffer, Catherine A, Turpin, Jim A, Williamson, Karen, Rice, William G
Published in Journal of medicinal chemistry (20.05.1999)
Published in Journal of medicinal chemistry (20.05.1999)
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Journal Article
Inhibition of multiple phases of human immunodeficiency virus type 1 replication by a dithiane compound that attacks the conserved zinc fingers of retroviral nucleocapsid proteins
RICE, W. G, BAKER, D. C, FIELD, L, SINGH, P. K, TURPIN, A. J. A, SCHAEFFER, C. A, GRAHAM, L, BU, M, TERPENING, S, CLANTON, D, SCHULTZ, R, BADER, J. P, BUCKHEIT, R. W
Published in Antimicrobial Agents and Chemotherapy (01.02.1997)
Published in Antimicrobial Agents and Chemotherapy (01.02.1997)
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Journal Article
Inhibitors of human immunodeficiency virus type 1 zinc fingers prevent normal processing of gag precursors and result in the release of noninfectious virus particles
Turpin, J A, Terpening, S J, Schaeffer, C A, Yu, G, Glover, C J, Felsted, R L, Sausville, E A, Rice, W G
Published in Journal of Virology (01.09.1996)
Published in Journal of Virology (01.09.1996)
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Journal Article
Induction of Endonuclease-Mediated Apoptosis in Tumor Cells by C-Nitroso- Substituted Ligands of Poly(ADP-Ribose) Polymerase
Rice, William G., Hillyer, Christopher D., Harten, Brad, Schaeffer, Catherine A., Dorminy, Mark, Lackey, Dixon A., Kirsten, Eva, Mendeleyev, Jerome, Buki, Kalman G., Hakam, Alaeddin, Kun, Ernest
Published in Proceedings of the National Academy of Sciences - PNAS (15.08.1992)
Published in Proceedings of the National Academy of Sciences - PNAS (15.08.1992)
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Journal Article
Synthesis of a cosalane analog with an extended polyanionic pharmacophore conferring enhanced potency as an anti-HIV agent
Cushman, Mark, Insaf, Shabana, Ruell, Jeffrey A., Schaeffer, Catherine A., Rice, William G.
Published in Bioorganic & medicinal chemistry letters (07.04.1998)
Published in Bioorganic & medicinal chemistry letters (07.04.1998)
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Journal Article
Human immunodeficiency virus type-1 (HIV-1) replication is unaffected by human secretory leukocyte protease inhibitor
Turpin, Jim A., Schaeffer, Catherine A., Bu, Ming, Graham, Lisa, Buckheit, Robert W., Clanton, David, Rice, William G.
Published in Antiviral research (01.03.1996)
Published in Antiviral research (01.03.1996)
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Journal Article
Inhibition of the replication of native and 3′-azido-2′,3′-dideoxy-thymidine (AZT)-resistant simian immunodeficiency virus (SIV) by 3-nitrosobenzamide
Chuang, Ann J., Killam, Keith F., Chuang, Ronald Y., Rice, William G., Schaeffer, Catherine A., Mendeleyev, Jerome, Kun, Ernest
Published in FEBS letters (01.07.1993)
Published in FEBS letters (01.07.1993)
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Journal Article
IN THE KNOW: SPORTS FINAL Edition
Julian Kesner, Brittany Schaeffer, Isabel Forgang, Catherine Clifford, Jo Piazza
Published in Daily news (New York, N.Y. : 1920) (10.03.2005)
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Published in Daily news (New York, N.Y. : 1920) (10.03.2005)
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