G-quadruplex forming regions in GCK and TM6SF2 are targets for differential DNA methylation in metabolic disease and hepatocellular carcinoma patients
Lahnsteiner, Angelika, Ellmer, Victoria, Oberlercher, Anna, Liutkeviciute, Zita, Schönauer, Esther, Paulweber, Bernhard, Aigner, Elmar, Risch, Angela
Published in Scientific reports (30.08.2024)
Published in Scientific reports (30.08.2024)
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N‑Aryl-3-mercaptosuccinimides as Antivirulence Agents Targeting Pseudomonas aeruginosa Elastase and Clostridium Collagenases
Konstantinović, Jelena, Yahiaoui, Samir, Alhayek, Alaa, Haupenthal, Jörg, Schönauer, Esther, Andreas, Anastasia, Kany, Andreas M, Müller, Rolf, Koehnke, Jesko, Berger, Fabian K, Bischoff, Markus, Hartmann, Rolf W, Brandstetter, Hans, Hirsch, Anna K. H
Published in Journal of medicinal chemistry (13.08.2020)
Published in Journal of medicinal chemistry (13.08.2020)
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Cloning, Purification and Characterization of the Collagenase ColA Expressed by Bacillus cereus ATCC 14579
Abfalter, Carmen M, Schönauer, Esther, Ponnuraj, Karthe, Huemer, Markus, Gadermaier, Gabriele, Regl, Christof, Briza, Peter, Ferreira, Fatima, Huber, Christian G, Brandstetter, Hans, Posselt, Gernot, Wessler, Silja
Published in PloS one (02.09.2016)
Published in PloS one (02.09.2016)
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Discovery and Characterization of Synthesized and FDA-Approved Inhibitors of Clostridial and Bacillary Collagenases
Alhayek, Alaa, Abdelsamie, Ahmed S., Schönauer, Esther, Camberlein, Virgyl, Hutterer, Evelyn, Posselt, Gernot, Serwanja, Jamil, Blöchl, Constantin, Huber, Christian G., Haupenthal, Jörg, Brandstetter, Hans, Wessler, Silja, Hirsch, Anna K. H.
Published in Journal of medicinal chemistry (13.10.2022)
Published in Journal of medicinal chemistry (13.10.2022)
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Discovery of a Potent Inhibitor Class with High Selectivity toward Clostridial Collagenases
Schönauer, Esther, Kany, Andreas M, Haupenthal, Jörg, Hüsecken, Kristina, Hoppe, Isabel J, Voos, Katrin, Yahiaoui, Samir, Elsässer, Brigitta, Ducho, Christian, Brandstetter, Hans, Hartmann, Rolf W
Published in Journal of the American Chemical Society (13.09.2017)
Published in Journal of the American Chemical Society (13.09.2017)
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Inhibitors of the Elastase LasB for the Treatment of Pseudomonas aeruginosa Lung Infections
Konstantinović, Jelena, Kany, Andreas M., Alhayek, Alaa, Abdelsamie, Ahmed S., Sikandar, Asfandyar, Voos, Katrin, Yao, Yiwen, Andreas, Anastasia, Shafiei, Roya, Loretz, Brigitta, Schönauer, Esther, Bals, Robert, Brandstetter, Hans, Hartmann, Rolf W., Ducho, Christian, Lehr, Claus-Michael, Beisswenger, Christoph, Müller, Rolf, Rox, Katharina, Haupenthal, Jörg, Hirsch, Anna K.H.
Published in ACS central science (27.12.2023)
Published in ACS central science (27.12.2023)
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Structure-Based Design of α‑Substituted Mercaptoacetamides as Inhibitors of the Virulence Factor LasB from Pseudomonas aeruginosa
Kaya, Cansu, Walter, Isabell, Alhayek, Alaa, Shafiei, Roya, Jézéquel, Gwenaëlle, Andreas, Anastasia, Konstantinović, Jelena, Schönauer, Esther, Sikandar, Asfandyar, Haupenthal, Jörg, Müller, Rolf, Brandstetter, Hans, Hartmann, Rolf W., Hirsch, Anna K.H.
Published in ACS infectious diseases (13.05.2022)
Published in ACS infectious diseases (13.05.2022)
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A conserved strategy to attack collagen: The activator domain in bacterial collagenases unwinds triple-helical collagen
Serwanja, Jamil, Wieland, Alexander C, Haubenhofer, Astrid, Brandstetter, Hans, Schönauer, Esther
Published in Proceedings of the National Academy of Sciences - PNAS (16.04.2024)
Published in Proceedings of the National Academy of Sciences - PNAS (16.04.2024)
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Phosphonate as a Stable Zinc‐Binding Group for “Pathoblocker” Inhibitors of Clostridial Collagenase H (ColH)
Voos, Katrin, Schönauer, Esther, Alhayek, Alaa, Haupenthal, Jörg, Andreas, Anastasia, Müller, Rolf, Hartmann, Rolf W., Brandstetter, Hans, Hirsch, Anna K. H., Ducho, Christian
Published in ChemMedChem (20.04.2021)
Published in ChemMedChem (20.04.2021)
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Front Cover: Phosphonate as a Stable Zinc‐Binding Group for “Pathoblocker” Inhibitors of Clostridial Collagenase H (ColH) (ChemMedChem 8/2021)
Voos, Katrin, Schönauer, Esther, Alhayek, Alaa, Haupenthal, Jörg, Andreas, Anastasia, Müller, Rolf, Hartmann, Rolf W., Brandstetter, Hans, Hirsch, Anna K. H., Ducho, Christian
Published in ChemMedChem (20.04.2021)
Published in ChemMedChem (20.04.2021)
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Inhibition of Collagenase Q1 of Bacillus cereus as a Novel Antivirulence Strategy for the Treatment of Skin‐Wound Infections
Alhayek, Alaa, Khan, Essak S., Schönauer, Esther, Däinghaus, Tobias, Shafiei, Roya, Voos, Katrin, Han, Mitchell K. L., Ducho, Christian, Posselt, Gernot, Wessler, Silja, Brandstetter, Hans, Haupenthal, Jörg, del Campo, Aránzazu, Hirsch, Anna K. H.
Published in Advanced therapeutics (01.03.2022)
Published in Advanced therapeutics (01.03.2022)
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universal strategy for high-yield production of soluble and functional clostridial collagenases in E. coli
Ducka, Paulina, Eckhard, Ulrich, Schönauer, Esther, Kofler, Stefan, Gottschalk, Gerhard, Brandstetter, Hans, Nüss, Dorota
Published in Applied microbiology and biotechnology (01.07.2009)
Published in Applied microbiology and biotechnology (01.07.2009)
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Crystallization and preliminary X-ray characterization of the catalytic domain of collagenase G from Clostridium histolyticum
Eckhard, Ulrich, Nüss, Dorota, Ducka, Paulina, Schönauer, Esther, Brandstetter, Hans
Published in Acta crystallographica. Section F, Structural biology and crystallization communications (01.05.2008)
Published in Acta crystallographica. Section F, Structural biology and crystallization communications (01.05.2008)
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