Search Results - "Sbacchi, Massimo" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Modification of Nociception and Morphine Tolerance by the Selective Opiate Receptor-Like Orphan Receptor Antagonist (â€“)-cis-1-Methyl-7-[[4-(2,6-dichlorophenyl)piperidin-1-yl]methyl]-6,7,8,9-tetrahydro-5H-benzocyclohepten-5-ol (SB-612111)

Modification of Nociception and Morphine Tolerance by the Selective Opiate Receptor-Like Orphan Receptor Antagonist (â)-cis-1-Methyl-7-[[4-(2,6-dichlorophenyl)piperidin-1-yl]methyl]-6,7,8,9-tetrahydro-5H-benzocyclohepten-5-ol (SB-612111)

by Zaratin, Paola F, Petrone, Giuseppe, Sbacchi, Massimo, Garnier, Martine, Fossati, Claudia, Petrillo, Paola, Ronzoni, Silvio, Giardina, Giuseppe A M, Scheideler, Mark A
Published in The Journal of pharmacology and experimental therapeutics (01.02.2004)

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(1S)-1-(Aminomethyl)-2-(arylacetyl)-1,2,3,4-tetrahydroisoquinoline and heterocycle-condensed tetrahydropyridine derivatives: members of a novel class of very potent .kappa. opioid analgesics

(1S)-1-(Aminomethyl)-2-(arylacetyl)-1,2,3,4-tetrahydroisoquinoline and heterocycle-condensed tetrahydropyridine derivatives: members of a novel class of very potent .kappa. opioid analgesics

by Vecchietti, Vittorio, Clarke, Geoffrey D, Colle, Roberto, Giardina, Giuseppe, Petrone, Giuseppe, Sbacchi, Massimo
Published in Journal of medicinal chemistry (01.08.1991)

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Evidence for a selective role of the delta-opioid agonist [8R-(4bS,8aalpha,8abeta, 12bbeta)]7,10-Dimethyl-1-methoxy-11-(2-methylpropyl)oxycarbonyl 5,6,7,8,12,12b-hexahydro-(9H)-4,8-methanobenzofuro[3,2-e]pyrrolo[2,3-g]isoquinoline hydrochloride (SB-235863) in blocking hyperalgesia associated with inflammatory and neuropathic pain responses

Evidence for a selective role of the delta-opioid agonist [8R-(4bS,8aalpha,8abeta, 12bbeta)]7,10-Dimethyl-1-methoxy-11-(2-methylpropyl)oxycarbonyl 5,6,7,8,12,12b-hexahydro-(9H)-4,8-methanobenzofuro[3,2-e]pyrrolo[2,3-g]isoquinoline hydrochloride (SB-235863) in blocking hyperalgesia associated with inflammatory and neuropathic pain responses

by Petrillo, Paola, Angelici, Ornella, Bingham, Sharon, Ficalora, Giovanna, Garnier, Martine, Zaratin, Paola F, Petrone, Giuseppe, Pozzi, Ottorino, Sbacchi, Massimo, Stean, Tania O, Upton, Neil, Dondio, Guillio M, Scheideler, Mark A
Published in The Journal of pharmacology and experimental therapeutics (01.12.2003)

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Synthesis, Biological Evaluation, and Receptor Docking Simulations of 2-[(Acylamino)ethyl]-1,4-benzodiazepines as κ-Opioid Receptor Agonists Endowed with Antinociceptive and Antiamnesic Activity

Synthesis, Biological Evaluation, and Receptor Docking Simulations of 2-[(Acylamino)ethyl]-1,4-benzodiazepines as κ-Opioid Receptor Agonists Endowed with Antinociceptive and Antiamnesic Activity

by Anzini, Maurizio, Canullo, Laura, Braile, Carlo, Cappelli, Andrea, Gallelli, Andrea, Vomero, Salvatore, Menziani, M. Cristina, De Benedetti, Pier G, Rizzo, Milena, Collina, Simona, Azzolina, Ornella, Sbacchi, Massimo, Ghelardini, Carla, Galeotti, Nicoletta
Published in Journal of medicinal chemistry (28.08.2003)

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Modification of Nociception and Morphine Tolerance by the Selective Opiate Receptor-Like Orphan Receptor Antagonist (–)- cis -1-Methyl-7-[[4-(2,6-dichlorophenyl)piperidin-1-yl]methyl]-6,7,8,9-tetrahydro-5 H -benzocyclohepten-5-ol (SB-612111)

Modification of Nociception and Morphine Tolerance by the Selective Opiate Receptor-Like Orphan Receptor Antagonist (–)- cis -1-Methyl-7-[[4-(2,6-dichlorophenyl)piperidin-1-yl]methyl]-6,7,8,9-tetrahydro-5 H -benzocyclohepten-5-ol (SB-612111)

by Zaratin, Paola F., Petrone, Giuseppe, Sbacchi, Massimo, Garnier, Martine, Fossati, Claudia, Petrillo, Paola, Ronzoni, Silvio, Giardina, Giuseppe A. M., Scheideler, Mark A.
Published in The Journal of pharmacology and experimental therapeutics (01.02.2004)

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Side-Chain Lactam-Bridge Conformational Constraints Differentiate the Activities of Salmon and Human Calcitonins and Reveal a New Design Concept for Potent Calcitonin Analogues

Side-Chain Lactam-Bridge Conformational Constraints Differentiate the Activities of Salmon and Human Calcitonins and Reveal a New Design Concept for Potent Calcitonin Analogues

by Taylor, John W, Jin, Qian K, Sbacchi, Massimo, Wang, Lu, Belfiore, Piero, Garnier, Martine, Kazantzis, Athanasios, Kapurniotu, Aphrodite, Zaratin, Paola F, Scheideler, Mark A
Published in Journal of medicinal chemistry (28.02.2002)

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Evidence for a Selective Role of the Î´-Opioid Agonist [8R-(4bS,8aÎ±,8aÎ²,12bÎ²)]7,10-Dimethyl-1-methoxy-11-(2-methylpropyl)oxycarbonyl 5,6,7,8,12,12b-hexahydro-(9H)-4,8-methanobenzofuro[3,2-e]pyrrolo[2,3-g]isoquinoline Hydrochloride (SB-235863) in Blocking Hyperalgesia Associated with Inflammatory and Neuropathic Pain Responses

Evidence for a Selective Role of the Î´-Opioid Agonist [8R-(4bS,8aÎ±,8aÎ²,12bÎ²)]7,10-Dimethyl-1-methoxy-11-(2-methylpropyl)oxycarbonyl 5,6,7,8,12,12b-hexahydro-(9H)-4,8-methanobenzofuro[3,2-e]pyrrolo[2,3-g]isoquinoline Hydrochloride (SB-235863) in Blocking Hyperalgesia Associated with Inflammatory and Neuropathic Pain Responses

by Paola Petrillo, Ornella Angelici, Sharon Bingham, Giovanna Ficalora, Martine Garnier, Paola F. Zaratin, Giuseppe Petrone, Ottorino Pozzi, Massimo Sbacchi, Tania O. Stean, Neil Upton, Guillio M. Dondio, Mark A. Scheideler
Published in The Journal of pharmacology and experimental therapeutics (01.12.2003)

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Synthesis and antinociceptive activity of pyrrolidinylnaphthalenes

Synthesis and antinociceptive activity of pyrrolidinylnaphthalenes

by COLLINA, S, AZZOLINA, O, VERCESI, D, SBACCHI, M, SCHEIDELER, M. A, BARBIERI, A, LANZA, E, GHISLANDI, V
Published in Bioorganic & medicinal chemistry (01.08.2000)

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Synthesis, Biological Evaluation, and Quantitative Receptor Docking Simulations of 2-[(Acylamino)ethyl]-1,4-benzodiazepines as Novel Tifluadom-like Ligands with High Affinity and Selectivity for κ-Opioid Receptors

Synthesis, Biological Evaluation, and Quantitative Receptor Docking Simulations of 2-[(Acylamino)ethyl]-1,4-benzodiazepines as Novel Tifluadom-like Ligands with High Affinity and Selectivity for κ-Opioid Receptors

by Cappelli, Andrea, Anzini, Maurizio, Vomero, Salvatore, Menziani, M. Cristina, De Benedetti, Pier G, Sbacchi, Massimo, Clarke, Geoffrey D, Mennuni, Laura
Published in Journal of medicinal chemistry (16.02.1996)

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Comparison of the Water Diuretic Activity of KappaReceptor Agonists and a Vasopressin Receptor Antagonist in Dogs

Comparison of the Water Diuretic Activity of KappaReceptor Agonists and a Vasopressin Receptor Antagonist in Dogs

by David P. Brooks, Maurizio Valente, Giuseppe Petrone, P. Dennis Depalma, Massimo Sbacchi, Geoffrey D. Clarke
Published in The Journal of pharmacology and experimental therapeutics (01.03.1997)

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Selective .kappa.-Opioid Agonists: Synthesis and Structure-Activity Relationships of Piperidines Incorporating an Oxo-Containing Acyl Group

Selective .kappa.-Opioid Agonists: Synthesis and Structure-Activity Relationships of Piperidines Incorporating an Oxo-Containing Acyl Group

by Giardina, Giuseppe, Clarke, Geoffrey D, Dondio, Giulio, Petrone, Giuseppe, Sbacchi, Massimo, Vecchietti, Vittorio
Published in Journal of medicinal chemistry (14.10.1994)

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Comparison of the water diuretic activity of kappa receptor agonists and a vasopressin receptor antagonist in dogs

Comparison of the water diuretic activity of kappa receptor agonists and a vasopressin receptor antagonist in dogs

by Brooks, D P, Valente, M, Petrone, G, Depalma, P D, Sbacchi, M, Clarke, G D
Published in The Journal of pharmacology and experimental therapeutics (01.03.1997)

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Characterization of opioid binding sites in rat spinal cord

Characterization of opioid binding sites in rat spinal cord

by Petrillo, P, Kowalski, J, Sbacchi, M, Tavani, A
Published in Journal of receptor research (1992)

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Substituted 1-(aminomethyl)-2-(arylacetyl)-1,2,3,4-tetrahydroisoquinolines: a novel class of very potent antinociceptive agents with varying degrees of selectivity for .kappa. and .mu. opioid receptors

Substituted 1-(aminomethyl)-2-(arylacetyl)-1,2,3,4-tetrahydroisoquinolines: a novel class of very potent antinociceptive agents with varying degrees of selectivity for .kappa. and .mu. opioid receptors

by Vecchietti, Vittorio, Clarke, Geoffrey D, Colle, Roberto, Dondio, Giulio, Giardina, Giuseppe, Petrone, Giuseppe, Sbacchi, Massimo
Published in Journal of medicinal chemistry (01.08.1992)

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Enantiospecificity of kappa receptors: comparison of racemic compounds and active enantiomers in two novel series of kappa agonist analgesics

Enantiospecificity of kappa receptors: comparison of racemic compounds and active enantiomers in two novel series of kappa agonist analgesics

by Colle, R, Clarke, G D, Dondio, G, Giardina, G, Petrone, G, Sbacchi, M, Vecchietti, V
Published in Chirality (New York, N.Y.) (1992)

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Regional variations in binding capacities at mu-, delta- and kappa-opioid sites in membrane suspensions from rabbit brain

Regional variations in binding capacities at mu-, delta- and kappa-opioid sites in membrane suspensions from rabbit brain

by Petrillo, P, La Regina, A, Sbacchi, M, Tavani, A, Robson, L E, Kosterlitz, H W
Published in European journal of pharmacology (18.07.1989)

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