Synthesis and evaluation of coumarin derivatives as potential dual-action HIV-1 protease and reverse transcriptase inhibitors
Olomola, Temitope O., Klein, Rosalyn, Mautsa, Nicodemus, Sayed, Yasien, Kaye, Perry T.
Published in Bioorganic & medicinal chemistry (01.04.2013)
Published in Bioorganic & medicinal chemistry (01.04.2013)
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The crystal structure of the host-guest complex: N′-{5-[2-(2,6-dimethylphenoxy)acetamido]-4-hydroxy-1,6-diphenylhexan-2-yl}-3-methyl-2-(2-oxo-1,3-diazinan-1-yl)butanamide-diethyl ether (2/1)
Mokoto, Tebogo M. L., Lemmerer, Andreas, Sayed, Yasien, Smith, Mark G.
Published in Zeitschrift für Kristallographie. New crystal structures (25.04.2024)
Published in Zeitschrift für Kristallographie. New crystal structures (25.04.2024)
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Journal Article
The crystal structure of N′-{5-[2-(2,6-dimethylphenoxy) acetamido]-4-hydroxy-1,6-diphenylhexan-2-yl}-3-methyl-2-(2-oxo-1,3-diazinan-1-yl)butanamide hydrate
Mokoto, Tebogo M. L., Lemmerer, Andreas, Sayed, Yasien, Smith, Mark G.
Published in Zeitschrift für Kristallographie. New crystal structures (25.06.2024)
Published in Zeitschrift für Kristallographie. New crystal structures (25.06.2024)
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Structural studies of hemoglobin from two flightless birds, ostrich and turkey: insights into their differing oxygen-binding properties
Ramesh, Pandian, Sundaresan, Selvarajan Sigamani, Shobana, Nagaraj, Vinuchakkaravarthy, Thangaraj, Sivakumar, Kandasamy, Yasien, Sayed, Ponnuswamy, Mondikalipudur Nanjappa Gounder
Published in Acta crystallographica. Section D, Biological crystallography. (01.05.2021)
Published in Acta crystallographica. Section D, Biological crystallography. (01.05.2021)
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The Unusual Architecture of RNA-Dependent RNA Polymerase (RdRp)'s Catalytic Chamber Provides a Potential Strategy for Combination Therapy against COVID-19
Metwally, Kamel, Abo-Dya, Nader E, Alahmdi, Mohammed Issa, Albalawi, Maha Z, Yahya, Galal, Aljoundi, Aimen, Salifu, Elliasu Y, Elamin, Ghazi, Ibrahim, Mahmoud A A, Sayed, Yasien, Fanucchi, Sylvia, Soliman, Mahmoud E S
Published in Molecules (Basel, Switzerland) (01.03.2023)
Published in Molecules (Basel, Switzerland) (01.03.2023)
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Crystal structure of hemoglobin from mouse (Mus musculus) compared with those from other small animals and humans
Sundaresan, Selvarajan Sigamani, Ramesh, Pandian, Shobana, Nagaraj, Vinuchakkaravarthy, Thangaraj, Yasien, Sayed, Ponnuswamy, Mondikalipudur Nanjappa Gounder
Published in Acta crystallographica. Section F, Structural biology communications (01.04.2021)
Published in Acta crystallographica. Section F, Structural biology communications (01.04.2021)
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Understanding Drug Resistance of Wild-Type and L38HL Insertion Mutant of HIV-1 C Protease to Saquinavir
Venkatachalam, Sankaran, Murlidharan, Nisha, Krishnan, Sowmya R, Ramakrishnan, C, Setshedi, Mpho, Pandian, Ramesh, Barh, Debmalya, Tiwari, Sandeep, Azevedo, Vasco, Sayed, Yasien, Gromiha, M Michael
Published in Genes (01.02.2023)
Published in Genes (01.02.2023)
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V2-Directed Vaccine-like Antibodies from HIV-1 Infection Identify an Additional K169-Binding Light Chain Motif with Broad ADCC Activity
van Eeden, Charmaine, Wibmer, Constantinos Kurt, Scheepers, Cathrine, Richardson, Simone I., Nonyane, Molati, Lambson, Bronwen, Mkhize, Nonhlanhla N., Vijayakumar, Balakrishnan, Sheng, Zizhang, Stanfield-Oakley, Sherry, Bhiman, Jinal N., Bekker, Valerie, Hermanus, Tandile, Mabvakure, Batsirai, Ismail, Arshad, Moody, M. Anthony, Wiehe, Kevin, Garrett, Nigel, Karim, Salim Abdool, Dirr, Heini, Fernandes, Manuel A., Sayed, Yasien, Shapiro, Lawrence, Ferrari, Guido, Haynes, Barton F., Moore, Penny L., Morris, Lynn
Published in Cell reports (Cambridge) (11.12.2018)
Published in Cell reports (Cambridge) (11.12.2018)
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SARS-CoV-2 Spike Protein Unlikely to Bind to Integrins via the Arg-Gly-Asp (RGD) Motif of the Receptor Binding Domain: Evidence From Structural Analysis and Microscale Accelerated Molecular Dynamics
Othman, Houcemeddine, Messaoud, Haifa Ben, Khamessi, Oussema, Ben-Mabrouk, Hazem, Ghedira, Kais, Bharuthram, Avani, Treurnicht, Florette, Achilonu, Ikechukwu, Sayed, Yasien, Srairi-Abid, Najet
Published in Frontiers in molecular biosciences (14.02.2022)
Published in Frontiers in molecular biosciences (14.02.2022)
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Synthesis, Characterization and Biological Activity of Some Dithiourea Derivatives
Odame, Felix, Hosten, Eric, Krause, Jason, Isaacs, Michelle, Hoppe, Heinrich, Khanye, Setshaba D, Sayed, Yasien, Frost, Carminita, Lobb, Kevin, Tshentu, Zenixole
Published in Acta chimica Slovenica (01.09.2020)
Published in Acta chimica Slovenica (01.09.2020)
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Journal Article
Kinetic and thermodynamic characterisation of HIV-protease inhibitors against E35D↑G↑S mutant in the South African HIV-1 subtype C protease
Maseko, Sibusiso, Padayachee, Eden, Maphumulo, Siyabonga, Govender, Thavendran, Sayed, Yasien, Maguire, Glenn, Lin, Johnson, Naicker, Tricia, Baijnath, Sooraj, Gerhardus, Kruger Hendrik
Published in Journal of enzyme inhibition and medicinal chemistry (2019)
Published in Journal of enzyme inhibition and medicinal chemistry (2019)
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Journal Article
Active-Site Mutations in the South African Human Immunodeficiency Virus Type 1 Subtype C Protease Have a Significant Impact on Clinical Inhibitor Binding: Kinetic and Thermodynamic Study
MOSEBI, Salerwe, MORRIS, Lynn, DIRR, Heini W, SAYED, Yasien
Published in Journal of Virology (15.11.2008)
Published in Journal of Virology (15.11.2008)
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Journal Article
A Conserved N-capping Motif Contributes Significantly to the Stabilization and Dynamics of the C-terminal Region of Class Alpha Glutathione S-Transferases
Dirr, Heini W., Little, Tessa, Kuhnert, Diane C., Sayed, Yasien
Published in The Journal of biological chemistry (20.05.2005)
Published in The Journal of biological chemistry (20.05.2005)
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Journal Article
Obtaining high yield recombinant Enterococcus faecium nicotinate nucleotide adenylyltransferase for X-ray crystallography and biophysical studies
Jeje, Olamide, Pandian, Ramesh, Sayed, Yasien, Achilonu, Ikechukwu
Published in International journal of biological macromolecules (01.10.2023)
Published in International journal of biological macromolecules (01.10.2023)
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