DNA‐damage inducible protein 1 is a conserved metacaspase substrate that is cleaved and further destabilized in yeast under specific metabolic conditions
Bouvier, León A., Niemirowicz, Gabriela T., Salas‐Sarduy, Emir, Cazzulo, Juan José, Alvarez, Vanina E.
Published in The FEBS journal (01.03.2018)
Published in The FEBS journal (01.03.2018)
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Journal Article
Enzyme Inhibitors from Gorgonians and Soft Corals
Córdova-Isaza, Andrea, Jiménez-Mármol, Sofía, Guerra, Yasel, Salas-Sarduy, Emir
Published in Marine drugs (31.01.2023)
Published in Marine drugs (31.01.2023)
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Journal Article
Three Decades of Targeting Falcipains to Develop Antiplasmodial Agents: What have we Learned and What can be Done Next?
González, Jorge Enrique Hernández, Salas-Sarduy, Emir, Alvarez, Lilian Hernández, Valiente, Pedro Alberto, Arni, Raghuvir Krishnaswamy, Pascutti, Pedro Geraldo
Published in Current medicinal chemistry (01.01.2024)
Published in Current medicinal chemistry (01.01.2024)
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Journal Article
The Trypanosoma cruzi Antigen and Epitope Atlas: antibody specificities in Chagas disease patients across the Americas
Ricci, Alejandro D, Bracco, Leonel, Salas-Sarduy, Emir, Ramsey, Janine M, Nolan, Melissa S, Lynn, M Katie, Altcheh, Jaime, Ballering, Griselda E, Torrico, Faustino, Kesper, Norival, Villar, Juan C, Marcipar, Iván S, Marco, Jorge D, Agüero, Fernán
Published in Nature communications (03.04.2023)
Published in Nature communications (03.04.2023)
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Journal Article
In silico identification of noncompetitive inhibitors targeting an uncharacterized allosteric site of falcipain-2
Hernández González, Jorge Enrique, Salas-Sarduy, Emir, Hernández Alvarez, Lilian, Barreto Gomes, Diego Enry, Pascutti, Pedro Geraldo, Oostenbrink, Chris, Leite, Vitor B. P.
Published in Journal of computer-aided molecular design (01.10.2021)
Published in Journal of computer-aided molecular design (01.10.2021)
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Journal Article
Potent and selective inhibitors for M32 metallocarboxypeptidases identified from high-throughput screening of anti-kinetoplastid chemical boxes
Salas-Sarduy, Emir, Landaburu, Lionel Urán, Carmona, Adriana K, Cazzulo, Juan José, Agüero, Fernán, Alvarez, Vanina E, Niemirowicz, Gabriela T
Published in PLoS neglected tropical diseases (01.07.2019)
Published in PLoS neglected tropical diseases (01.07.2019)
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Journal Article
Identification of Tight-Binding Plasmepsin II and Falcipain 2 Inhibitors in Aqueous Extracts of Marine Invertebrates by the Combination of Enzymatic and Interaction-Based Assays
Salas-Sarduy, Emir, Guerra, Yasel, Covaleda Cortés, Giovanni, Avilés, Francesc Xavier, Chávez Planes, María A
Published in Marine drugs (21.04.2017)
Published in Marine drugs (21.04.2017)
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Journal Article
Computer-aided design of bromelain and papain covalent immobilization
Cutiño-Avila, Bessy, Gil Pradas, Dayrom, Aragón Abreu, Carlos, Fernández Marrero, Yuniel, Hernández de la Torre, Martha, Salas Sarduy, Emir, Chávez Planes, María De los Ángeles, Guisán Seijas, José Manuel, Díaz Brito, Joaquín, Del Monte-Martínez, Alberto
Published in Revista Colombiana de biotecnologia (01.01.2014)
Published in Revista Colombiana de biotecnologia (01.01.2014)
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Journal Article
Design, synthesis and biological evaluation of novel thiosemicarbazones as cruzipain inhibitors
Jasinski, Gabriel, Salas-Sarduy, Emir, Vega, Daniel, Fabian, Lucas, Florencia Martini, M., Moglioni, Albertina G.
Published in European journal of medicinal chemistry (05.06.2023)
Published in European journal of medicinal chemistry (05.06.2023)
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Journal Article
Thiosemicarbazone derivatives: Evaluation as cruzipain inhibitors and molecular modeling study of complexes with cruzain
Jasinski, Gabriel, Salas-Sarduy, Emir, Vega, Daniel, Fabian, Lucas, Martini, María Florencia, Moglioni, Albertina G.
Published in Bioorganic & medicinal chemistry (01.05.2022)
Published in Bioorganic & medicinal chemistry (01.05.2022)
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Journal Article
Screening and Identification of Metacaspase Inhibitors: Evaluation of Inhibition Mechanism and Trypanocidal Activity
Pérez, Brian, Bouvier, León A, Cazzulo, Juan José, Agüero, Fernán, Salas-Sarduy, Emir, Alvarez, Vanina E
Published in Antimicrobial agents and chemotherapy (17.02.2021)
Published in Antimicrobial agents and chemotherapy (17.02.2021)
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Journal Article
Novel scaffolds for inhibition of Cruzipain identified from high-throughput screening of anti-kinetoplastid chemical boxes
Salas-Sarduy, Emir, Landaburu, Lionel Urán, Karpiak, Joel, Madauss, Kevin P, Cazzulo, Juan José, Agüero, Fernán, Alvarez, Vanina Eder
Published in Scientific reports (21.09.2017)
Published in Scientific reports (21.09.2017)
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Journal Article
Tetracycline Derivatives Inhibit Plasmodial Cysteine Protease Falcipain‑2 through Binding to a Distal Allosteric Site
Hernández González, Jorge Enrique, Alberca, Lucas N, Masforrol González, Yordanka, Reyes Acosta, Osvaldo, Talevi, Alan, Salas-Sarduy, Emir
Published in Journal of chemical information and modeling (10.01.2022)
Published in Journal of chemical information and modeling (10.01.2022)
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Journal Article
Author Correction: Novel scaffolds for inhibition of Cruzipain identified from high-throughput screening of anti-kinetoplastid chemical boxes
Salas-Sarduy, Emir, Landaburu, Lionel Urán, Karpiak, Joel, Madauss, Kevin P, Cazzulo, Juan José, Agüero, Fernán, Alvarez, Vanina Eder
Published in Scientific reports (04.06.2018)
Published in Scientific reports (04.06.2018)
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Journal Article
Intensity fading MALDI-TOF mass spectrometry and functional proteomics assignments to identify protease inhibitors in marine invertebrates
Covaleda, Giovanni, Trejo, Sebastian A., Salas-Sarduy, Emir, del Rivero, Maday Alonso, Chavez, Maria Angeles, Aviles, Francesc X.
Published in Journal of proteomics (08.08.2017)
Published in Journal of proteomics (08.08.2017)
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Journal Article
Identification of (4-(9H-fluoren-9-yl) piperazin-1-yl) methanone derivatives as falcipain 2 inhibitors active against Plasmodium falciparum cultures
Hernández-González, Jorge E., Salas-Sarduy, Emir, Hernández Ramírez, Luisa F., Pascual, María J., Álvarez, Diego E., Pabón, Adriana, Leite, Vitor B.P., Pascutti, Pedro G., Valiente, Pedro A.
Published in Biochimica et biophysica acta. General subjects (01.12.2018)
Published in Biochimica et biophysica acta. General subjects (01.12.2018)
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Journal Article