The Prodrug Approach: A Successful Tool for Improving Drug Solubility
Jornada, Daniela Hartmann, dos Santos Fernandes, Guilherme Felipe, Chiba, Diego Eidy, de Melo, Thais Regina Ferreira, dos Santos, Jean Leandro, Chung, Man Chin
Published in Molecules (29.12.2015)
Published in Molecules (29.12.2015)
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Book Review
Unraveling the Anticancer Effect of Curcumin and Resveratrol
Pavan, Aline Renata, Silva, Gabriel Dalio Bernardes da, Jornada, Daniela Hartmann, Chiba, Diego Eidy, Fernandes, Guilherme Felipe Dos Santos, Man Chin, Chung, Dos Santos, Jean Leandro
Published in Nutrients (10.11.2016)
Published in Nutrients (10.11.2016)
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Book Review
Resveratrol-nitric oxide donor hybrid effect on priapism in sickle cell and nitric oxide-deficient mouse
Pinheiro, Andressa Kely, Pereira, Dalila Andrade, Dos Santos, Jean Leandro, Calmasini, Fabiano Beraldi, Alexandre, Eduardo Costa, Reis, Leonardo Oliveira, Burnett, Arthur L, Costa, Fernando Ferreira, Silva, Fábio Henrique
Published in PloS one (02.06.2022)
Published in PloS one (02.06.2022)
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Design, synthesis and biological evaluation of N-oxide derivatives with potent in vivo antileishmanial activity
Clementino, Leandro da Costa, Fernandes, Guilherme Felipe Santos, Prokopczyk, Igor Muccilo, Laurindo, Wilquer Castro, Toyama, Danyelle, Motta, Bruno Pereira, Baviera, Amanda Martins, Henrique-Silva, Flávio, Santos, Jean Leandro Dos, Graminha, Marcia A S
Published in PloS one (01.11.2021)
Published in PloS one (01.11.2021)
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Optimization of Resveratrol Used as a Scaffold to Design Histone Deacetylase (HDAC-1 and HDAC-2) Inhibitors
Urias, Beatriz Silva, Pavan, Aline Renata, Albuquerque, Gabriela Ribeiro, Prokopczyk, Igor Muccilo, Alves, Tânia Mara Ferreira, de Melo, Thais Regina Ferreira, Sartori, Geraldo Rodrigues, da Silva, João Hermínio Martins, Chin, Chung Man, Santos, Jean Leandro Dos
Published in Pharmaceuticals (Basel, Switzerland) (01.10.2022)
Published in Pharmaceuticals (Basel, Switzerland) (01.10.2022)
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Journal Article
Current Advances in Antitubercular Drug Discovery: Potent Prototypes and New Targets
Dos Santos Fernandes, Guilherme Felipe, Jornada, Daniela Hartmann, de Souza, Paula Carolina, Chin, Chung Man, Pavan, Fernando Rogerio, Dos Santos, Jean Leandro
Published in Current medicinal chemistry (01.01.2015)
Published in Current medicinal chemistry (01.01.2015)
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Dietary Compound Resveratrol Is a Pan-BET Bromodomain Inhibitor
Dutra, Luiz Antonio, Heidenreich, David, Silva, Gabriel Dalio Bernardes da, Man Chin, Chung, Knapp, Stefan, Santos, Jean Leandro Dos
Published in Nutrients (27.10.2017)
Published in Nutrients (27.10.2017)
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Antiplatelet and antithrombotic activities of non-steroidal anti-inflammatory drugs containing an N-acyl hydrazone subunit
Chelucci, Rafael Consolin, Dutra, Luiz Antônio, Lopes Pires, Maria Elisa, de Melo, Thais Regina Ferreira, Bosquesi, Priscila Longhin, Chung, Man Chin, Dos Santos, Jean Leandro
Published in Molecules (Basel, Switzerland) (17.02.2014)
Published in Molecules (Basel, Switzerland) (17.02.2014)
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Anti-Inflammatory Drug Design Using a Molecular Hybridization Approach
Bosquesi, Priscila Longhin, Melo, Thais Regina Ferreira, Vizioli, Ednir Oliveira, Santos, Jean Leandro Dos, Chung, Man Chin
Published in Pharmaceuticals (27.10.2011)
Published in Pharmaceuticals (27.10.2011)
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Book Review
Synthesis and Preliminary Evaluation of N-Oxide Derivatives for the Prevention of Atherothrombotic Events
Rosseto, Leandro Augusto, Pires, Maria Elisa Lopes, Melchior, Aylime Castanho Bolognesi, Bosquesi, Priscila Longhin, Pavan, Aline Renata, Marcondes, Sisi, Chung, Man Chin, Santos, Jean Leandro Dos
Published in Molecules (Basel, Switzerland) (07.10.2015)
Published in Molecules (Basel, Switzerland) (07.10.2015)
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Pharmacological evaluation and preparation of nonsteroidal anti-inflammatory drugs containing an N-acyl hydrazone subunit
de Melo, Thais Regina Ferreira, Chelucci, Rafael Consolin, Pires, Maria Elisa Lopes, Dutra, Luiz Antonio, Barbieri, Karina Pereira, Bosquesi, Priscila Longhin, Trossini, Gustavo Henrique Goulart, Chung, Man Chin, dos Santos, Jean Leandro
Published in International journal of molecular sciences (04.04.2014)
Published in International journal of molecular sciences (04.04.2014)
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Advances in drug design based on the amino Acid approach: taurine analogues for the treatment of CNS diseases
Chung, Man Chin, Malatesta, Pedro, Bosquesi, Priscila Longhin, Yamasaki, Paulo Renato, Santos, Jean Leandro Dos, Vizioli, Ednir Oliveira
Published in Pharmaceuticals (23.10.2012)
Published in Pharmaceuticals (23.10.2012)
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Book Review
Endothelial dysfunction in Sickle Cell Disease: Strategies for the treatment
Pavan, Aline Renata, Terroni, Barbara, Dos Santos, Jean Leandro
Published in Nitric oxide (01.08.2024)
Published in Nitric oxide (01.08.2024)
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Journal Article
Recent advances in drug discovery against Mycobacterium tuberculosis: Metal-based complexes
Scarim, Cauê Benito, Lira de Farias, Renan, Vieira de Godoy Netto, Adelino, Chin, Chung Man, Leandro dos Santos, Jean, Pavan, Fernando Rogério
Published in European journal of medicinal chemistry (15.03.2021)
Published in European journal of medicinal chemistry (15.03.2021)
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Pharmacological evaluation and preliminary pharmacokinetics studies of a new diclofenac prodrug without gastric ulceration effect
Santos, Jean Leandro Dos, Moreira, Vanessa, Campos, Michel Leandro, Chelucci, Rafael Consolin, Barbieri, Karina Pereira, de Castro Souto, Pollyana Cristina Maggio, Matsubara, Márcio Hideki, Teixeira, Catarina, Bosquesi, Priscila Longhin, Peccinini, Rosângela Gonçalves, Chin, Chung Man
Published in International journal of molecular sciences (19.11.2012)
Published in International journal of molecular sciences (19.11.2012)
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