Rapid identification of a novel phosphodiesterase 7B tracer for receptor occupancy studies using LC─MS/MS
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Published in Neurochemistry international (01.07.2020)
Published in Neurochemistry international (01.07.2020)
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Design and Synthesis of Novel and Selective Glycine Transporter‑1 (GlyT1) Inhibitors with Memory Enhancing Properties
Santora, Vincent J, Almos, Theresa A, Barido, Richard, Basinger, Jillian, Bellows, Chris L, Bookser, Brett C, Breitenbucher, J. Guy, Broadbent, Nicola J, Cabebe, Clifford, Chai, Chih-Kun, Chen, Mi, Chow, Stephine, Chung, De Michael, Crickard, Lindsay, Danks, Anne M, Freestone, Graeme C, Gitnick, Dany, Gupta, Varsha, Hoffmaster, Christine, Hudson, Andrew R, Kaplan, Alan P, Kennedy, Michael R, Lee, Dong, Limberis, James, Ly, Kiev, Mak, Chi Ching, Masatsugu, Brittany, Morse, Andrew C, Na, Jim, Neul, David, Nikpur, John, Peters, Marco, Petroski, Robert E, Renick, Joel, Sebring, Kristen, Sevidal, Samantha, Tabatabaei, Ali, Wen, Jenny, Yan, Yingzhuo, Yoder, Zachary W, Zook, Douglas
Published in Journal of medicinal chemistry (26.07.2018)
Published in Journal of medicinal chemistry (26.07.2018)
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Azetidine-based selective glycine transporter-1 (GlyT1) inhibitors with memory enhancing properties
Hudson, Andrew R., Santora, Vincent J., Petroski, Robert E., Almos, Theresa A., Anderson, Gary, Barido, Richard, Basinger, Jillian, Bellows, Chris L., Bookser, Brett C., Broadbent, Nicola J., Cabebe, Clifford, Chai, Chih-Kun, Chen, Mi, Chow, Stephine, Chung, De Michael, Heger, Lindsay, Danks, Anne M., Freestone, Graeme C., Gitnick, Dany, Gupta, Varsha, Hoffmaster, Christine, Kaplan, Alan P., Kennedy, Michael R., Lee, Dong, Limberis, James, Ly, Kiev, Mak, Chi Ching, Masatsugu, Brittany, Morse, Andrew C., Na, Jim, Neul, David, Nikpur, John, Renick, Joel, Sebring, Kristen, Sevidal, Samantha, Tabatabaei, Ali, Wen, Jenny, Xia, Shouzhen, Yan, Yingzhuo, Yoder, Zachary W., Zook, Douglas, Peters, Marco, Breitenbucher, J. Guy
Published in Bioorganic & medicinal chemistry letters (15.07.2020)
Published in Bioorganic & medicinal chemistry letters (15.07.2020)
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Structure-activity relationships of 3,4-dihydro-1H-quinazolin-2-one derivatives as potential CDK5 inhibitors
RZASA, Robert M, KALLER, Matthew R, XIAOLING XIONG, WENGE ZHONG, NORMAN, Mark H, GANG LIU, MAGAL, Ella, NGUYEN, Thomas T, OSSLUND, Timothy D, POWERS, David, SANTORA, Vincent J, VISWANADHAN, Vellarkad N, WANG, Hui-Ling
Published in Bioorganic & medicinal chemistry (15.10.2007)
Published in Bioorganic & medicinal chemistry (15.10.2007)
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A new family of H3 receptor antagonists based on the natural product Conessine
SANTORA, Vincent J, COVEL, Jonathan A, WEBB, Robert R, SAGE, Carleton, REN, Albert, PEREIRA, Guilherme, KNUDSEN, Jens, EDWARDS, Jeffrey E, SUAREZ, Marissa, FRAZER, John, THOMSEN, William, HAUSER, Erin, HAYASHI, Rena, WHELAN, Kevin, GROTTICK, Andrew J, HOFILENA, Brian J, IBARRA, Jason B, PULLEY, Michelle D, WEINHOUSE, Michael I, SENGUPTA, Dipanjan, DUFFIELD, Jonathan J, SEMPLE, Graeme
Published in Bioorganic & medicinal chemistry letters (15.02.2008)
Published in Bioorganic & medicinal chemistry letters (15.02.2008)
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Identification of biaryl sulfone derivatives as antagonists of the histamine H3 receptor: Discovery of (R)-1-(2-(4′-(3-methoxypropylsulfonyl)biphenyl-4-yl)ethyl)-2-methylpyrrolidine (APD916)
Semple, Graeme, Santora, Vincent J., Smith, Jeffrey M., Covel, Jonathan A., Hayashi, Rena, Gallardo, Charlemagne, Ibarra, Jason B., Schultz, Jeffrey A., Park, Douglas M., Estrada, Scott A., Hofilena, Brian J., Smith, Brian M., Ren, Albert, Suarez, Marissa, Frazer, John, Edwards, Jeffrey E., Hart, Ryan, Hauser, Erin K., Lorea, Jodie, Grottick, Andrew J.
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
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Design and Evaluation of Novel Biphenyl Sulfonamide Derivatives with Potent Histamine H(3) Receptor Inverse Agonist Activity
Covel, Jonathan A., Santora, Vincent J., Smith, Jeffrey M., Hayashi, Rena, Gallardo, Charlemagne, Weinhouse, Michael I., Ibarra, Jason B., Schultz, Jeffrey A., Park, Douglas M., Estrada, Scott A., Hofilena, Brian J., Pulley, Michelle D., Smith, Brian M., Ren, Albert, Suarez, Marissa, Frazer, John, Edwards, Jeffrey, Hauser, Erin K., Lorca, Jodie, Semple, Graeme, Grottick, Andrew J.
Published in Journal of medicinal chemistry (24.09.2009)
Published in Journal of medicinal chemistry (24.09.2009)
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Journal Article
Design and Evaluation of Novel Biphenyl Sulfonamide Derivatives with Potent Histamine H3 Receptor Inverse Agonist Activity
Covel, Jonathan A., Santora, Vincent J., Smith, Jeffrey M., Hayashi, Rena, Gallardo, Charlemagne, Weinhouse, Michael I., Ibarra, Jason B., Schultz, Jeffrey A., Park, Douglas M., Estrada, Scott A., Hofilena, Brian J., Pulley, Michelle D., Smith, Brian M., Ren, Albert, Suarez, Marissa, Frazer, John, Edwards, Jeffrey, Hauser, Erin K., Lorea, Jodie, Semple, Graeme, Grottick, Andrew J.
Published in Journal of medicinal chemistry (24.09.2009)
Published in Journal of medicinal chemistry (24.09.2009)
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Novel H3 receptor antagonists with improved pharmacokinetic profiles
SANTORA, Vincent J, COVEL, Jonathan A, EDWARDS, Jeffrey E, SUAREZ, Marissa, FRAZER, John, THOMSEN, William, HAUSER, Erin, LOREA, Jodie, GROTTICK, Andrew J, HAYASHI, Rena, HOFILENA, Brian J, IBARRA, Jason B, PULLEY, Michelle D, WEINHOUSE, Michael I, SEMPLE, Graeme, REN, Albert, PEREIRA, Guilherme
Published in Bioorganic & medicinal chemistry letters (15.07.2008)
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Structure−Activity Relationships of a Series of Pyrrolo[3,2-d]pyrimidine Derivatives and Related Compounds as Neuropeptide Y5 Receptor Antagonists
Norman, Mark H, Chen, Ning, Chen, Zhidong, Fotsch, Christopher, Hale, Clarence, Han, Nianhe, Hurt, Ray, Jenkins, Tracy, Kincaid, John, Liu, Longbin, Lu, Yuelie, Moreno, Ofir, Santora, Vincent J, Sonnenberg, Jennifer D, Karbon, William
Published in Journal of medicinal chemistry (02.11.2000)
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Cyclobutenone-Based Syntheses of Polyquinanes and Bicyclo[6.3.0]undecanes by Tandem Anionic Oxy-Cope Reactions. Total Synthesis of (±)-Precapnelladiene
MacDougall, James M, Santora, Vincent J, Verma, Sharad K, Turnbull, Philip, Hernandez, Cameron R, Moore, Harold W
Published in Journal of organic chemistry (02.10.1998)
Published in Journal of organic chemistry (02.10.1998)
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Complexation of benzamidinium by a new family of artificial receptors
Bell, Thomas W, Santora, Vincent J
Published in Journal of the American Chemical Society (01.10.1992)
Published in Journal of the American Chemical Society (01.10.1992)
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WONG ALICE R, CZABANIUK LARA C, WU YONGWEI, RESCOURIO GWENAELLA, SANTORA VINCENT, HOUZE JONATHAN B, WHITE RYAN D, HOPPER TIMOTHY, WANG HAOXUAN
Year of Publication 13.02.2023
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Year of Publication 13.02.2023
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골수성 세포 2 작용제 상에서 발현되는 유발 수용체로서의 헤테로고리 화합물 및 사용 방법
MANCUSO JOHN, WU YONGWEI, RESCOURIO GWENAELLA, PANTELEEV JANE, WHITE RYAN D, HOPPER TIMOTHY, BOS MAXENCE, WONG ALICE R, CZABANIUK LARA C, SANTORA VINCENT, HOUZE JONATHAN B, FRANZONI IVAN, WANG HAOXUAN
Year of Publication 09.02.2023
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Year of Publication 09.02.2023
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Discovery and evaluation of dual CDK1 and CDK2 inhibitors
PAYTON, Marc, CHUNG, Grace, ASKEW, Ben, TASKER, Andrew, RADINSKY, Robert, KENDALL, Richard, COATS, Steve, YAKOWEC, Peter, WONG, Andrew, POWERS, Dave, LING XIONG, ZHANG, Nancy, LEAL, Juan, BUSH, Tammy L, SANTORA, Vincent
Published in Cancer research (Chicago, Ill.) (15.04.2006)
Published in Cancer research (Chicago, Ill.) (15.04.2006)
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Tandem Oxy-Cope-Transannular Ring Closure Route to Polyquinanes
Santora, Vincent J, Moore, Harold W
Published in Journal of the American Chemical Society (01.08.1995)
Published in Journal of the American Chemical Society (01.08.1995)
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A new family of H 3 receptor antagonists based on the natural product Conessine
Santora, Vincent J., Covel, Jonathan A., Hayashi, Rena, Hofilena, Brian J., Ibarra, Jason B., Pulley, Michelle D., Weinhouse, Michael I., Sengupta, Dipanjan, Duffield, Jonathan J., Semple, Graeme, Webb, Robert R., Sage, Carleton, Ren, Albert, Pereira, Guilherme, Knudsen, Jens, Edwards, Jeffrey E., Suarez, Marissa, Frazer, John, Thomsen, William, Hauser, Erin, Whelan, Kevin, Grottick, Andrew J.
Published in Bioorganic & medicinal chemistry letters (15.02.2008)
Published in Bioorganic & medicinal chemistry letters (15.02.2008)
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