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Published in Journal of medicinal chemistry (11.11.2010)
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Folate–Vinca Alkaloid Conjugates for Cancer Therapy: A Structure–Activity Relationship
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Published in Bioconjugate chemistry (19.03.2014)
Published in Bioconjugate chemistry (19.03.2014)
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Design and regioselective synthesis of a new generation of targeted chemotherapeutics. Part 1: EC145, a folic acid conjugate of desacetylvinblastine monohydrazide
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Published in Bioorganic & medicinal chemistry letters (01.10.2006)
Published in Bioorganic & medicinal chemistry letters (01.10.2006)
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Antiinflammatory Activity of a Novel Folic Acid Targeted Conjugate of the mTOR Inhibitor Everolimus
Lu, Yingjuan, Parker, Nikki, Kleindl, Paul J, Cross, Vicky A, Wollak, Kristin, Westrick, Elaine, Stinnette, Torian W, Gehrke, Mark A, Wang, Kevin, Santhapuram, Hari Krishna R, You, Fei, Hahn, Spencer J, Vaughn, Jeremy F, Klein, Patrick J, Vlahov, Iontcho R, Low, Philip S, Leamon, Christopher P
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Published in Molecular medicine (Cambridge, Mass.) (08.07.2015)
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An Assembly Concept for the Consecutive Introduction of Unsymmetrical Disulfide Bonds: Synthesis of a Releasable Multidrug Conjugate of Folic Acid
Vlahov, Iontcho R, Santhapuram, Hari Krishna R, Wang, Yu, Kleindl, Paul J, You, Fei, Howard, Stephen J, Westrick, Elaine, Reddy, Joseph A, Leamon, Christopher P
Published in Journal of organic chemistry (03.08.2007)
Published in Journal of organic chemistry (03.08.2007)
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Design and synthesis of a folate-receptor targeted diazepine-ring-opened pyrrolobenzodiazepine prodrug conjugate
Vlahov, Iontcho R., Qi, Longwu, Santhapuram, Hari Krishna R., Felten, Albert, Parham, Garth L., Zou, Ning, Wang, Kevin, You, Fei, Vaughn, Jeremy F., Hahn, Spencer J., Klein, Hanna F., Kleindl, Paul J., Reddy, Joe, Reno, Dan, Nicoson, Jeff, Leamon, Christopher P.
Published in Bioorganic & medicinal chemistry letters (01.04.2020)
Published in Bioorganic & medicinal chemistry letters (01.04.2020)
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Pre-clinical studies of EC2629, a highly potent folate- receptor-targeted DNA crosslinking agent
Reddy, Joseph A., Nelson, Melissa, Dircksen, Christina, Vetzel, Marilynn, Johnson, Theresa, Cross, Vicky, Westrick, Elaine, Qi, LongWu, Hahn, Spencer, Santhapuram, Hari Krishna, Parham, Garth, Wang, Kevin, Vaughn, Jeremy F., Felten, Albert, Pugh, Michael, Lu, June, Klein, Patrick, Vlahov, Iontcho R., Leamon, Christopher P.
Published in Scientific reports (29.07.2020)
Published in Scientific reports (29.07.2020)
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Carbohydrate-Based Synthetic Approach to Control Toxicity Profiles of Folate−Drug Conjugates
Vlahov, Iontcho R, Santhapuram, Hari Krishna R, You, Fei, Wang, Yu, Kleindl, Paul J, Hahn, Spencer J, Vaughn, Jeremy F, Reno, Daniel S, Leamon, Christopher P
Published in Journal of organic chemistry (04.06.2010)
Published in Journal of organic chemistry (04.06.2010)
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Regioselective synthesis of folate receptor-targeted agents derived from epothilone analogs and folic acid
Vlahov, Iontcho R., Vite, Gregory D., Kleindl, Paul J., Wang, Yu, Santhapuram, Hari Krishna R., You, Fei, Howard, Stephen J., Kim, Soong-Hoon, Lee, Francis F.Y., Leamon, Christopher P.
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
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Design and regioselective synthesis of a new generation of targeted therapeutics. Part 3: Folate conjugates of aminopterin hydrazide for the treatment of inflammation
Vlahov, Iontcho R., You, Fei, Santhapuram, Hari Krishna R., Wang, Yu, Vaughn, Jeremy F., Hahn, Spencer J., Kleindl, Paul J., Fan, Mingjin, Leamon, Christopher P.
Published in Bioorganic & medicinal chemistry letters (15.02.2011)
Published in Bioorganic & medicinal chemistry letters (15.02.2011)
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Year of Publication 21.12.2023
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Year of Publication 21.12.2023
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Tumor targeting using 67Ga-DOTA-Bz-folate — investigations of methods to improve the tissue distribution of radiofolates
Müller, Cristina, Vlahov, Iontcho R., Santhapuram, Hari Krishna R., Leamon, Christopher P., Schibli, Roger
Published in Nuclear medicine and biology (01.07.2011)
Published in Nuclear medicine and biology (01.07.2011)
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Strategy to Prevent Drug-Related Hypersensitivity in Folate-Targeted Hapten Immunotherapy of Cancer
Lu, Yingjuan, Klein, Patrick J., Westrick, Elaine, Xu, Le-Cun, Santhapuram, Hari Krishna R., Bloomfield, Alicia, Howard, Stephen J., Vlahov, Iontcho R., Ellis, P. Ron, Low, Philip S., Leamon, Christopher P.
Published in The AAPS journal (01.09.2009)
Published in The AAPS journal (01.09.2009)
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PROCESSES FOR PREPARING TUBULYSINS
STANFORD KATHERYN MARIE, SANTHAPURAM HARI KRISHNA R, VLAHOV IONTCHO RADOSLAVOV, YOU FEI, GROANING MICHAEL, KLEINDL PAUL JOSEPH, WANG YU, XU LE CUN, RITTER ALLEN, LEAMON CHRISTOPHER PAUL
Year of Publication 30.08.2013
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Year of Publication 30.08.2013
Patent
Preclinical Antitumor Activity of a Novel Folate-Targeted Dual Drug Conjugate
Leamon, Christopher P, Reddy, Joseph A, Vlahov, Iontcho R, Westrick, Elaine, Dawson, Alicia, Dorton, Ryan, Vetzel, Marilynn, Santhapuram, Hari Krishna, Wang, Yu
Published in Molecular pharmaceutics (01.09.2007)
Published in Molecular pharmaceutics (01.09.2007)
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Abstract 3259: An efficient total synthesis of Tubulysin B
Vlahov, Iontcho R., Groaning, Michael, Kleindl, Paul, Santhapuram, Hari Krishna R., You, Fei, Wang, Yu, Xu, Lecun, Stanford, Katheryn, Ritter, Allen, Leamon, Christopher P.
Published in Cancer research (Chicago, Ill.) (15.04.2011)
Published in Cancer research (Chicago, Ill.) (15.04.2011)
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Tumor targeting using67 Ga-DOTA-Bz-folate — investigations of methods to improve the tissue distribution of radiofolates
Müller, Cristina, Vlahov, Iontcho R, Santhapuram, Hari Krishna R, Leamon, Christopher P, Schibli, Roger
Published in Nuclear medicine and biology (2011)
Published in Nuclear medicine and biology (2011)
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