Hydroxychloroquine for Treatment of SARS‐CoV‐2 Infection? Improving Our Confidence in a Model‐Based Approach to Dose Selection
Arnold, Samuel L.M., Buckner, Frederick
Published in Clinical and Translational Science (01.07.2020)
Published in Clinical and Translational Science (01.07.2020)
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Pharmacological inhibition of ALDH1A in mice decreases all-trans retinoic acid concentrations in a tissue specific manner
Arnold, Samuel L.M., Kent, Travis, Hogarth, Cathryn A., Griswold, Michael D., Amory, John K., Isoherranen, Nina
Published in Biochemical pharmacology (01.06.2015)
Published in Biochemical pharmacology (01.06.2015)
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In vitro activity, safety and in vivo efficacy of the novel bumped kinase inhibitor BKI-1748 in non-pregnant and pregnant mice experimentally infected with Neospora caninum tachyzoites and Toxoplasma gondii oocysts
Imhof, Dennis, Anghel, Nicoleta, Winzer, Pablo, Balmer, Vreni, Ramseier, Jessica, Hänggeli, Kai, Choi, Ryan, Hulverson, Matthew A., Whitman, Grant R., Arnold, Samuel L.M., Ojo, Kayode K., Van Voorhis, Wesley C., Doggett, J. Stone, Ortega-Mora, Luis M., Hemphill, Andrew
Published in International journal for parasitology -- drugs and drug resistance (01.08.2021)
Published in International journal for parasitology -- drugs and drug resistance (01.08.2021)
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Efficacy of the bumped kinase inhibitor BKI-1708 against the cyst-forming apicomplexan parasites Toxoplasma gondii and Neospora caninum in vitro and in experimentally infected mice
de Sousa, Maria Cristina Ferreira, Imhof, Dennis, Hänggeli, Kai Pascal Alexander, Choi, Ryan, Hulverson, Matthew A., Arnold, Samuel L.M., Van Voorhis, Wesley C., Fan, Erkang, Roberto, Sánchez-Sánchez, Ortega-Mora, Luis M., Hemphill, Andrew
Published in International journal for parasitology -- drugs and drug resistance (01.08.2024)
Published in International journal for parasitology -- drugs and drug resistance (01.08.2024)
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Clofazimine pharmacokinetics in HIV‐infected adults with diarrhea: Implications of diarrheal disease on absorption of orally administered therapeutics
Zhang, Cindy X., Conrad, Thomas M., Hermann, David, Gordon, Melita A., Houpt, Eric, Iroh Tam, Pui‐Ying, Jere, Khuzwayo C., Nedi, Wilfred, Operario, Darwin J., Phulusa, Jacob, Quinnan, Gerald V., Sawyer, Leigh A., Barrett, Lynn K., Thole, Herbert, Toto, Neema, Van Voorhis, Wesley C., Arnold, Samuel L. M.
Published in CPT: pharmacometrics and systems pharmacology (01.03.2024)
Published in CPT: pharmacometrics and systems pharmacology (01.03.2024)
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Pharmacologic inhibition of mTOR improves lapatinib sensitivity in HER2-overexpressing breast cancer cells with primary trastuzumab resistance
Gayle, Sylvia S, Arnold, Samuel L M, O'Regan, Ruth M, Nahta, Rita
Published in Anti-cancer agents in medicinal chemistry (01.02.2012)
Published in Anti-cancer agents in medicinal chemistry (01.02.2012)
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Endochin-like quinolones (ELQs) and bumped kinase inhibitors (BKIs): Synergistic and additive effects of combined treatments against Neospora caninum infection in vitro and in vivo
Anghel, Nicoleta, Imhof, Dennis, Winzer, Pablo, Balmer, Vreni, Ramseier, Jessica, Haenggeli, Kai, Choi, Ryan, Hulverson, Matthew A., Whitman, Grant R., Arnold, Samuel L.M., Ojo, Kayode K., Van Voorhis, Wesley C., Doggett, J. Stone, Ortega-Mora, Luis M., Hemphill, Andrew
Published in International journal for parasitology -- drugs and drug resistance (01.12.2021)
Published in International journal for parasitology -- drugs and drug resistance (01.12.2021)
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Repurposing Infectious Disease Hits as Anti-Cryptosporidium Leads
Hulverson, Matthew A, Choi, Ryan, McCloskey, Molly C, Whitman, Grant R, Ojo, Kayode K, Michaels, Samantha A, Somepalli, Mastanbabu, Love, Melissa S, McNamara, Case W, Rabago, Lesley M, Barrett, Lynn K, J. Verlinde, Christophe L. M, Arnold, Samuel L.M, Striepen, Boris, Jimenez-Alfaro, Dolores, Ballell, Lluis, Fernández, Elena, Greenwood, M. Nicole, las Heras, Laura de, Calderón, Felix, Van Voorhis, Wesley C
Published in ACS infectious diseases (14.05.2021)
Published in ACS infectious diseases (14.05.2021)
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CTLA-4 and PD-1 dual blockade induces SIV reactivation without control of rebound after antiretroviral therapy interruption
Harper, Justin, Gordon, Shari, Chan, Chi Ngai, Wang, Hong, Lindemuth, Emily, Galardi, Cristin, Falcinelli, Shane D, Raines, Samuel L M, Read, Jenna L, Nguyen, Kevin, McGary, Colleen S, Nekorchuk, Michael, Busman-Sahay, Kathleen, Schawalder, James, King, Colin, Pino, Maria, Micci, Luca, Cervasi, Barbara, Jean, Sherrie, Sanderson, Andrew, Johns, Brian, Koblansky, A Alicia, Amrine-Madsen, Heather, Lifson, Jeffrey, Margolis, David M, Silvestri, Guido, Bar, Katharine J, Favre, David, Estes, Jacob D, Paiardini, Mirko
Published in Nature medicine (01.04.2020)
Published in Nature medicine (01.04.2020)
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An Early Treatment With BKI-1748 Exhibits Full Protection Against Abortion and Congenital Infection in Sheep Experimentally Infected With Toxoplasma gondii
Sánchez-Sánchez, Roberto, Imhof, Dennis, Hecker, Yanina P, Ferre, Ignacio, Re, Michela, Moreno-Gonzalo, Javier, Blanco-Murcia, Javier, Mejías-López, Elena, Hulverson, Matthew A, Choi, Ryan, Arnold, Samuel L M, Ojo, Kayode K, Barrett, Lynn K, Hemphill, Andrew, Van Voorhis, Wesley C, Ortega-Mora, Luis Miguel
Published in The Journal of infectious diseases (14.02.2024)
Published in The Journal of infectious diseases (14.02.2024)
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Stable Latent HIV Infection and Low-level Viremia Despite Treatment With the Broadly Neutralizing Antibody VRC07-523LS and the Latency Reversal Agent Vorinostat
Gay, Cynthia L, James, Katherine S, Tuyishime, Marina, Falcinelli, Shane D, Joseph, Sarah B, Moeser, Matthew J, Allard, Brigitte, Kirchherr, Jennifer L, Clohosey, Matthew, Raines, Samuel L M, Montefiori, David C, Shen, Xiaoying, Gorelick, Robert J, Gama, Lucio, McDermott, Adrian B, Koup, Richard A, Mascola, John R, Floris-Moore, Michelle, Kuruc, JoAnn D, Ferrari, Guido, Eron, Joseph J, Archin, Nancie M, Margolis, David M
Published in The Journal of infectious diseases (02.03.2022)
Published in The Journal of infectious diseases (02.03.2022)
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The Effects of Human Immunodeficiency Virus Type 1 (HIV-1) Antigen-Expanded Specific T-Cell Therapy and Vorinostat on Persistent HIV-1 Infection in People With HIV on Antiretroviral Therapy
Gay, Cynthia L, Hanley, Patrick J, Falcinelli, Shane D, Kuruc, JoAnn D, Pedersen, Susan M, Kirchherr, Jennifer, Raines, Samuel L M, Motta, Cecilia M, Lazarski, Chris, Chansky, Pamela, Tanna, Jay, Shibli, Abeer, Datar, Anushree, McCann, Chase D, Sili, Uluhan, Ke, Ruian, Eron, Joseph J, Archin, Nancie, Goonetilleke, Nilu, Bollard, Catherine M, Margolis, David M
Published in The Journal of infectious diseases (14.03.2024)
Published in The Journal of infectious diseases (14.03.2024)
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Pharmacokinetics and Pharmacodynamics of Clofazimine for Treatment of Cryptosporidiosis
Zhang, Cindy X, Love, Melissa S, McNamara, Case W, Chi, Victor, Woods, Ashley K, Joseph, Sean, Schaefer, Deborah A, Betzer, Dana P, Riggs, Michael W, Iroh Tam, Pui-Ying, Van Voorhis, Wesley C, Arnold, Samuel L M
Published in Antimicrobial agents and chemotherapy (18.01.2022)
Published in Antimicrobial agents and chemotherapy (18.01.2022)
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Development of 5‑Aminopyrazole-4-carboxamide-based Bumped-Kinase Inhibitors for Cryptosporidiosis Therapy
Huang, Wenlin, Hulverson, Matthew A, Choi, Ryan, Arnold, Samuel L. M, Zhang, Zhongsheng, McCloskey, Molly C, Whitman, Grant R, Hackman, Robert C, Rivas, Kasey L, Barrett, Lynn K, Ojo, Kayode K, Van Voorhis, Wesley C, Fan, Erkang
Published in Journal of medicinal chemistry (28.03.2019)
Published in Journal of medicinal chemistry (28.03.2019)
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Bumped Kinase Inhibitors as therapy for apicomplexan parasitic diseases: lessons learned
Choi, Ryan, Hulverson, Matthew A., Huang, Wenlin, Vidadala, Rama S.R., Whitman, Grant R., Barrett, Lynn K., Schaefer, Deborah A., Betzer, Dana P., Riggs, Michael W., Doggett, J. Stone, Hemphill, Andrew, Ortega-Mora, Luis Miguel, McCloskey, Molly C., Arnold, Samuel L.M., Hackman, Robert C., Marsh, Kennan C., Lynch, James J., Freiberg, Gail M., Leroy, Bruce E., Kempf, Dale J., Choy, Robert K.M., de Hostos, Eugenio L., Maly, Dustin J., Fan, Erkang, Ojo, Kayode K., Van Voorhis, Wesley C.
Published in International journal for parasitology (01.05.2020)
Published in International journal for parasitology (01.05.2020)
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Altered Expression of Small Heterodimer Partner Governs Cytochrome P450 (CYP) 2D6 Induction during Pregnancy in CYP2D6-humanized Mice
Koh, Kwi Hye, Pan, Xian, Shen, Hong-Wu, Arnold, Samuel L.M., Yu, Ai-Ming, Gonzalez, Frank J., Isoherranen, Nina, Jeong, Hyunyoung
Published in The Journal of biological chemistry (07.02.2014)
Published in The Journal of biological chemistry (07.02.2014)
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