Ligand-induced overexpression of a constitutively active β2-adrenergic receptor: Pharmacological creation of a phenotype in transgenic mice
Samama, Philippe, Bond, Richard A., Rockman, Howard A., Milano, Carmelo A., Lefkowitz, Robert J.
Published in Proceedings of the National Academy of Sciences - PNAS (07.01.1997)
Published in Proceedings of the National Academy of Sciences - PNAS (07.01.1997)
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Journal Article
A mutation-induced activated state of the β2-adrenergic receptor : extending the ternary complex model
SAMAMA, P, COTECCHIA, S, COSTA, T, LEFKOWITZ, R. J
Published in The Journal of biological chemistry (05.03.1993)
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Published in The Journal of biological chemistry (05.03.1993)
Journal Article
Cardiac Function in Mice Overexpressing the β-Adrenergic Receptor Kinase or a βARK Inhibitor
Koch, Walter J., Rockman, Howard A., Samama, Philippe, Hamilton, RaeAnn, Bond, Richard A., Milano, Carmelo A., Lefkowitz, Robert J.
Published in Science (American Association for the Advancement of Science) (02.06.1995)
Published in Science (American Association for the Advancement of Science) (02.06.1995)
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Journal Article
Negative antagonists promote as inactive conformation of the β2-adrenergic receptor
SAMAMA, P, GANG PEI, COSTA, T, COTECCHIA, S, LEFKOWITZ, R. J
Published in Molecular pharmacology (1994)
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Published in Molecular pharmacology (1994)
Journal Article
A Constitutively Active Mutant β2-Adrenergic Receptor is Constitutively Desensitized and Phosphorylated
Pei, Gang, Samama, Philippe, Lohse, Martin, Wang, Mei, Codina, Juan, Lefkowitz, Robert J.
Published in Proceedings of the National Academy of Sciences - PNAS (29.03.1994)
Published in Proceedings of the National Academy of Sciences - PNAS (29.03.1994)
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Journal Article
Conference Proceeding
Imidazolylpyrimidine based CXCR2 chemokine receptor antagonists
Ho, Koc-Kan, Auld, Douglas S., Bohnstedt, Adolph C., Conti, Paolo, Dokter, Wim, Erickson, Shawn, Feng, Daming, Inglese, Jim, Kingsbury, Celia, Kultgen, Steven G., Liu, Rong-Qiang, Masterson, Christopher M., Ohlmeyer, Michael, Rong, Yajing, Rooseboom, Martijn, Roughton, Andrew, Samama, Philippe, Smit, Martin-Jan, Son, Ellen, van der Louw, Jaap, Vogel, Gerard, Webb, Maria, Wijkmans, Jac, You, Ming
Published in Bioorganic & medicinal chemistry letters (15.05.2006)
Published in Bioorganic & medicinal chemistry letters (15.05.2006)
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Journal Article
Chemokine Receptor−Ligand Interactions Measured Using Time-Resolved Fluorescence
Inglese, James, Samama, Philippe, Patel, Sanjay, Burbaum, Jonathan, Stroke, Ilana L, Appell, Kenneth C
Published in Biochemistry (Easton) (24.02.1998)
Published in Biochemistry (Easton) (24.02.1998)
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Journal Article
Combinatorial gene expression using multiple episomal vectors
Horlick, Robert A., Schilling, Adriane E., Samama, Philippe, Swanson, Robert N., Fitzpatrick, V.Danial, Robbins, Alan K., Damaj, Bassam
Published in Gene (08.02.2000)
Published in Gene (08.02.2000)
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Journal Article
Development of a fluorescent ligand-binding assay using the AcroWell filter plate
Valenzano, K J, Miller, W, Kravitz, J N, Samama, P, Fitzpatrick, D, Seeley, K
Published in Journal of biomolecular screening (01.12.2000)
Published in Journal of biomolecular screening (01.12.2000)
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Journal Article
Ligand-induced overexpression of a constitutively active beta2-adrenergic receptor: pharmacological creation of a phenotype in transgenic mice
Samama, P, Bond, R A, Rockman, H A, Milano, C A, Lefkowitz, R J
Published in Proceedings of the National Academy of Sciences - PNAS (07.01.1997)
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Published in Proceedings of the National Academy of Sciences - PNAS (07.01.1997)
Journal Article
Ligand-Induced Overexpression of a Constitutively Active β 2-adrenergic Receptor: Pharmacological Creation of a Phenotype in Transgenic Mice
Samama, Philippe, Bond, Richard A., Rockman, Howard A., Milano, Carmelo A., Lefkowitz, Robert J.
Published in Proceedings of the National Academy of Sciences - PNAS (07.01.1997)
Published in Proceedings of the National Academy of Sciences - PNAS (07.01.1997)
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Journal Article
Cardiac function in mice overexpressing the Beta-adrenergic receptor kinase or a BataARK inhibitor. (Beta-adrenergic receptor kinase)
Koch, Walter J, Rockman, Howard A, Samama, Philippe, Hamilton, RaeAnn, Bond, Richard A, Milano, Carmelo A, Lefkowitz, Robert J
Published in Science (American Association for the Advancement of Science) (02.06.1995)
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Published in Science (American Association for the Advancement of Science) (02.06.1995)
Journal Article
Site-specific bioconjugates of chemokines and their use in assays
INGLESE; JAMES, SAMAMA; PHILIPPE, STROKE; ILANA L, BURBAUM; JONATHAN J, APPELL; KENNETH C
Year of Publication 05.12.2000
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Year of Publication 05.12.2000
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