Striking Effect of Hydroxamic Acid Substitution on the Phosphodiesterase Type 4 (PDE4) and TNFα Inhibitory Activity of Two Series of Rolipram Analogues: Implications for a New Active Site Model of PDE4
Kleinman, Edward F, Campbell, Erin, Giordano, Lisa A, Cohan, Victoria L, Jenkinson, Teresa H, Cheng, John B, Shirley, John T, Pettipher, E. Roy, Salter, Eben D, Hibbs, Tessa A, DiCapua, Frank M, Bordner, John
Published in Journal of medicinal chemistry (29.01.1998)
Published in Journal of medicinal chemistry (29.01.1998)
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2‐Amino‐4‐methylpyridine as a potent inhibitor of inducible NO synthase activity in vitro and in vivo
Faraci, W. Stephen, Nagel, Arthur A., Verdries, Kimberly A., Vincent, Lawrence A., Xu, Hong, Nichols, Lois E., Labasi, Jeffrey M., Salter, Eben D., Pettipher, E. Roy
Published in British journal of pharmacology (01.11.1996)
Published in British journal of pharmacology (01.11.1996)
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Inhibition of leukotriene B4-receptor interaction suppresses eosinophil infiltration and disease pathology in a murine model of experimental allergic encephalomyelitis
Gladue, R P, Carroll, L A, Milici, A J, Scampoli, D N, Stukenbrok, H A, Pettipher, E R, Salter, E D, Contillo, L, Showell, H J
Published in The Journal of experimental medicine (01.04.1996)
Published in The Journal of experimental medicine (01.04.1996)
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The Preclinical Pharmacological Profile of the Potent and Selective Leukotriene B4 Antagonist CP-195543
Showell, H J, Conklyn, M J, Alpert, R, Hingorani, G P, Wright, K F, Smith, M A, Stam, E, Salter, E D, Scampoli, D N, Meltzer, S, Reiter, L A, Koch, K, Piscopio, A D, Cortina, S R, Lopez-Anaya, A, Pettipher, E R, Milici, A J, Griffiths, R J
Published in The Journal of pharmacology and experimental therapeutics (01.06.1998)
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Published in The Journal of pharmacology and experimental therapeutics (01.06.1998)
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The in vitro and in vivo pharmacologic activity of the potent and selective leukotriene B4 receptor antagonist CP-105696
Showell, H J, Pettipher, E R, Cheng, J B, Breslow, R, Conklyn, M J, Farrell, C A, Hingorani, G P, Salter, E D, Hackman, B C, Wimberly, D J
Published in The Journal of pharmacology and experimental therapeutics (01.04.1995)
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Published in The Journal of pharmacology and experimental therapeutics (01.04.1995)
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Specific inhibition of leukotriene B4 (LTB4)‐induced neutrophil emigration by 20‐hydroxy LTB4: implications for the regulation of inflammatory responses
Pettipher, E.R., Salter, E.D., Breslow, R., Raycroft, L., Showell, H.J.
Published in British journal of pharmacology (01.09.1993)
Published in British journal of pharmacology (01.09.1993)
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Biarylcarboxamide inhibitors of phosphodiesterase IV and tumor necrosis factor-α
Chambers, R.J., Marfat, A., Cheng, J.B., Cohan, V.L., Damon, D.B., Duplantier, A.J., Hibbs, T.A., Jenkinson, T.H., Johnson, K.L., Kraus, K.G., Pettipher, E.R., Salter, E.D., Shirley, J.T., Umland, J.P.
Published in Bioorganic & medicinal chemistry letters (18.03.1997)
Published in Bioorganic & medicinal chemistry letters (18.03.1997)
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A new chemical tool for exploring the role of the PDE4D isozyme in leukocyte function
Chambers, Robert J., Abrams, Kristin, Castleberry, Tessa A., Cheng, John B., Fisher, Douglas A., Kamath, Ajith V., Marfat, Anthony, Nettleton, David O., Pillar, Joann D., Salter, Eben D., Sheils, Alissa L., Shirley, John T., Turner, Claudia R., Umland, John P., Lam, Kelvin T.
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
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Inhibition of leukotriene B sub(4)-receptor interaction suppresses eosinophil infiltration and disease pathology in a murine model of experimental allergic encephalomyelitis
Gladue, R P, Carroll, LA, Milici, A J, Scampoli, D N, Stukenbrok, HA, Pettipher, E R, Salter, ED, Contillo, L, Showell, HJ
Published in The Journal of experimental medicine (01.01.1996)
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Published in The Journal of experimental medicine (01.01.1996)
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