Preparation of 3,5-Methanobenzo[b]azepines: An sp3‑Rich Quinolone Isostere
Herter, Loïc, Perrin, Timothé, Fessard, Thomas, Salomé, Christophe
Published in Organic letters (25.08.2023)
Published in Organic letters (25.08.2023)
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Journal Article
Activating Pyrimidines by Pre-distortion for the General Synthesis of 7‑Aza-indazoles from 2‑Hydrazonylpyrimidines via Intramolecular Diels–Alder Reactions
Le Fouler, Vincent, Chen, Yu, Gandon, Vincent, Bizet, Vincent, Salomé, Christophe, Fessard, Thomas, Liu, Fang, Houk, K. N, Blanchard, Nicolas
Published in Journal of the American Chemical Society (09.10.2019)
Published in Journal of the American Chemical Society (09.10.2019)
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Journal Article
Domino Pd0‐Catalyzed C(sp3)–H Arylation/Electrocyclic Reactions via Benzazetidine Intermediates
Rocaboy, Ronan, Dailler, David, Zellweger, Florian, Neuburger, Markus, Salomé, Christophe, Clot, Eric, Baudoin, Olivier
Published in Angewandte Chemie International Edition (10.09.2018)
Published in Angewandte Chemie International Edition (10.09.2018)
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Journal Article
d-Glucose: An Efficient Reducing Agent for a Copper(II)-Mediated Arylation of Primary Amines in Water
Bollenbach, Maud, Wagner, Patrick, Aquino, Pedro G. V., Bourguignon, Jean-Jacques, Bihel, Frédéric, Salomé, Christophe, Schmitt, Martine
Published in ChemSusChem (23.11.2016)
Published in ChemSusChem (23.11.2016)
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Journal Article
Synthesis and Anticonvulsant Activities of (R)-N-(4′-Substituted)benzyl 2-Acetamido-3-methoxypropionamides
Salomé, Christophe, Salomé-Grosjean, Elise, Park, Ki Duk, Morieux, Pierre, Swendiman, Robert, DeMarco, Erica, Stables, James P, Kohn, Harold
Published in Journal of medicinal chemistry (11.02.2010)
Published in Journal of medicinal chemistry (11.02.2010)
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Journal Article
Efficient and Mild Ullmann‐Type N‐Arylation of Amides, Carbamates, and Azoles in Water
Bollenbach, Maud, Aquino, Pedro G. V., de Araújo‐Júnior, João Xavier, Bourguignon, Jean‐Jacques, Bihel, Frédéric, Salomé, Christophe, Wagner, Patrick, Schmitt, Martine
Published in Chemistry : a European journal (04.10.2017)
Published in Chemistry : a European journal (04.10.2017)
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Journal Article
Chemical Library Screening and Structure-Function Relationship Studies Identify Bisacodyl as a Potent and Selective Cytotoxic Agent Towards Quiescent Human Glioblastoma Tumor Stem-Like Cells
Zeniou, Maria, Fève, Marie, Mameri, Samir, Dong, Jihu, Salomé, Christophe, Chen, Wanyin, El-Habr, Elias A, Bousson, Fanny, Sy, Mohamadou, Obszynski, Julie, Boh, Alexandre, Villa, Pascal, Assad Kahn, Suzana, Didier, Bruno, Bagnard, Dominique, Junier, Marie-Pierre, Chneiweiss, Hervé, Haiech, Jacques, Hibert, Marcel, Kilhoffer, Marie-Claude
Published in PloS one (13.08.2015)
Published in PloS one (13.08.2015)
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Journal Article
Primary Amino Acid Derivatives: Compounds with Anticonvulsant and Neuropathic Pain Protection Activities
King, Amber M, Salomé, Christophe, Dinsmore, Jason, Salomé-Grosjean, Elise, De Ryck, Marc, Kaminski, Rafal, Valade, Anne, Kohn, Harold
Published in Journal of medicinal chemistry (14.07.2011)
Published in Journal of medicinal chemistry (14.07.2011)
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Journal Article
Primary Amino Acid Derivatives: Substitution of the 4′-N′-Benzylamide Site in (R)-N′-Benzyl 2-Amino-3-methylbutanamide, (R)-N′-Benzyl 2-Amino-3,3-dimethylbutanamide, and (R)-N′-Benzyl 2-Amino-3-methoxypropionamide Provides Potent Anticonvulsants with Pain-Attenuating Properties
King, Amber M, Salomé, Christophe, Salomé-Grosjean, Elise, De Ryck, Marc, Kaminski, Rafal, Valade, Anne, Stables, James P, Kohn, Harold
Published in Journal of medicinal chemistry (13.10.2011)
Published in Journal of medicinal chemistry (13.10.2011)
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Journal Article
Lacosamide Isothiocyanate-Based Agents: Novel Agents To Target and Identify Lacosamide Receptors
Park, Ki Duk, Morieux, Pierre, Salomé, Christophe, Cotten, Steven W, Reamtong, Onrapak, Eyers, Claire, Gaskell, Simon J, Stables, James P, Liu, Rihe, Kohn, Harold
Published in Journal of medicinal chemistry (12.11.2009)
Published in Journal of medicinal chemistry (12.11.2009)
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Journal Article
Development and Characterization of Novel Derivatives of the Antiepileptic Drug Lacosamide That Exhibit Far Greater Enhancement in Slow Inactivation of Voltage-Gated Sodium Channels
Wang, Yuying, Park, Ki Duk, Salomé, Christophe, Wilson, Sarah M, Stables, James P, Liu, Rihe, Khanna, Rajesh, Kohn, Harold
Published in ACS chemical neuroscience (16.02.2011)
Published in ACS chemical neuroscience (16.02.2011)
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Journal Article
Merging Structural Motifs of Functionalized Amino Acids and α-Aminoamides Results in Novel Anticonvulsant Compounds with Significant Effects on Slow and Fast Inactivation of Voltage-Gated Sodium Channels and in the Treatment of Neuropathic Pain
Wang, Yuying, Wilson, Sarah M, Brittain, Joel M, Ripsch, Matthew S, Salomé, Christophe, Park, Ki Duk, White, Fletcher A, Khanna, Rajesh, Kohn, Harold
Published in ACS chemical neuroscience (15.06.2011)
Published in ACS chemical neuroscience (15.06.2011)
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Journal Article
Identification of the Benzyloxyphenyl Pharmacophore: A Structural Unit That Promotes Sodium Channel Slow Inactivation
King, Amber M, Yang, Xiao-Fang, Wang, Yuying, Dustrude, Erik T, Barbosa, Cindy, Due, Michael R, Piekarz, Andrew D, Wilson, Sarah M, White, Fletcher A, Salomé, Christophe, Cummins, Theodore R, Khanna, Rajesh, Kohn, Harold
Published in ACS chemical neuroscience (19.12.2012)
Published in ACS chemical neuroscience (19.12.2012)
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Journal Article
Smart tools and orthogonal click-like reactions onto small unilamellar vesicles: Additional molecular data
Vittoria Spanedda, Maria, Salomé, Christophe, Hilbold, Benoît, Berner, Etienne, Heurtault, Béatrice, Fournel, Sylvie, Frisch, Benoît, Bourel-Bonnet, Line
Published in Data in brief (01.12.2015)
Published in Data in brief (01.12.2015)
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