Design, synthesis, mechanistic and histopathological studies of small-molecules of novel indole-2-carboxamides and pyrazino[1,2-a]indol-1(2H)-ones as potential anticancer agents effecting the reactive oxygen species production
Youssif, Bahaa G.M., Abdelrahman, Mostafa H., Abdelazeem, Ahmed H., abdelgawad, Mohamed A., Ibrahim, Hussein M., Salem, Ola I.A., Mohamed, Mamdouh F.A., Treambleau, Laurent, Bukhari, Syed Nasir Abbas
Published in European journal of medicinal chemistry (25.02.2018)
Published in European journal of medicinal chemistry (25.02.2018)
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Design, synthesis and antiproliferative evaluation of lipidated 1,3-diaryl propenones and their cyclized pyrimidine derivatives as tubulin polymerization inhibitors
Ali, Fatma Elzahraa, Salem, Ola I.A., El-Mokhtar, Mohamed A., Aboraia, Ahmed S., Abdel-Moty, Samia G., Abdel-Aal, Abu-Baker M.
Published in Results in Chemistry (01.12.2023)
Published in Results in Chemistry (01.12.2023)
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Novel class of benzimidazole-thiazole hybrids: The privileged scaffolds of potent anti-inflammatory activity with dual inhibition of cyclooxygenase and 15-lipoxygenase enzymes
Maghraby, Mohammed T.-E., Abou-Ghadir, Ola M.F., Abdel-Moty, Samia G., Ali, Asmaa Y., Salem, Ola I.A.
Published in Bioorganic & medicinal chemistry (01.04.2020)
Published in Bioorganic & medicinal chemistry (01.04.2020)
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Design, synthesis, and antiproliferative properties of new 1,2,3-triazole-carboximidamide derivatives as dual EGFR/VEGFR-2 inhibitors
Mahmoud, Mohamed A., Mohammed, Anber F., Salem, Ola I.A., Rabea, Safwat M., Youssif, Bahaa G.M.
Published in Journal of molecular structure (15.06.2023)
Published in Journal of molecular structure (15.06.2023)
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Novel fluoroquinolone hybrids as dual DNA gyrase and urease inhibitors with potential antibacterial activity: Design, synthesis, and biological evaluation
Abdel-Aziz, Salah A., Cirnski, Katarina, Herrmann, Jennifer, Abdel-Aal, Mohamed A.A., Youssif, Bahaa G.M., Salem, Ola I.A.
Published in Journal of molecular structure (05.01.2023)
Published in Journal of molecular structure (05.01.2023)
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Design and synthesis of novel 2,3-dihydropyrazino[1,2-a]indole-1,4-dione derivatives as antiproliferative EGFR and BRAF(V600E) dual inhibitors
Al-Wahaibi, Lamya H., Gouda, Ahmed M., Abou-Ghadir, Ola F., Salem, Ola I. A., Ali, Asmaa T., Farghaly, Hatem S., Abdelrahman, Mostafa H., Trembleau, Laurent, Abdu-Allah, Hajjaj H. M., Youssif, Bahaa G. M.
Published in Bioorganic chemistry (01.11.2020)
Published in Bioorganic chemistry (01.11.2020)
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Journal Article
New 1,3,4‐oxadiazoles linked with the 1,2,3‐triazole moiety as antiproliferative agents targeting the EGFR tyrosine kinase
Mahmoud, Mohamed A., Mohammed, Anber F., Salem, Ola I. A., Gomaa, Hesham A. M., Youssif, Bahaa G. M.
Published in Archiv der Pharmazie (Weinheim) (01.06.2022)
Published in Archiv der Pharmazie (Weinheim) (01.06.2022)
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Novel 1,2,4-triazole derivatives as apoptotic inducers targeting p53: Synthesis and antiproliferative activity
Gomaa, Hesham A.M., El-Sherief, Hany A.M., Hussein, Shaimaa, Gouda, Ahmed M., Salem, Ola I.A., Alharbi, Khalid Saad, Hayallah, Alaa M., Youssif, Bahaa G.M.
Published in Bioorganic chemistry (01.12.2020)
Published in Bioorganic chemistry (01.12.2020)
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Journal Article
Design, synthesis, and apoptotic antiproliferative action of new 1,2,3-triazole/1,2,4-oxadiazole hybrids as dual EGFR/VEGFR-2 inhibitors
Mahmoud, Mohamed A., Mohammed, Anber F., Salem, Ola I. A., Almutairi, Tahani Mazyad, Braese, Stefan, Youssif, Bahaa G. M.
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2024)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2024)
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Journal Article
New 1,2,3-Triazole/1,2,4-triazole Hybrids as Aromatase Inhibitors: Design, Synthesis, and Apoptotic Antiproliferative Activity
Maghraby, Mohamed T-E, Mazyad Almutairi, Tahani, Bräse, Stefan, Salem, Ola I. A, Youssif, Bahaa G. M, Sheha, Mahmoud M
Published in Molecules (Basel, Switzerland) (01.10.2023)
Published in Molecules (Basel, Switzerland) (01.10.2023)
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New pyrimidine/thiazole hybrids endowed with analgesic, anti‐inflammatory, and lower cardiotoxic activities: Design, synthesis, and COX‐2/sEH dual inhibition
Abdel‐Aziz, Salah A., Taher, Ehab S., Lan, Ping, El‐Koussi, Nawal A., Salem, Ola I. A., Gomaa, Hesham A. M., Youssif, Bahaa G. M.
Published in Archiv der Pharmazie (Weinheim) (01.07.2022)
Published in Archiv der Pharmazie (Weinheim) (01.07.2022)
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Journal Article
Novel N-substituted 5-aminosalicylamides as dual inhibitors of cyclooxygenase and 5-lipoxygenase enzymes: Synthesis, biological evaluation and docking study
El-Nagar, Mohamed K.S., Abdu-Allah, Hajjaj H.M., Salem, Ola I.A., Kafafy, Abdel-Hamid N., Farghaly, Hanan S.M.
Published in Bioorganic chemistry (01.08.2018)
Published in Bioorganic chemistry (01.08.2018)
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Journal Article
Design and synthesis of novel 2,3-dihydropyrazino[1,2-a]indole-1,4-dione derivatives as antiproliferative EGFR and BRAFV600E dual inhibitors
Al-Wahaibi, Lamya H., Gouda, Ahmed M., Abou-Ghadir, Ola F., Salem, Ola I.A., Ali, Asmaa T., Farghaly, Hatem S., Abdelrahman, Mostafa H., Trembleau, Laurent, Abdu-Allah, Hajjaj H.M., Youssif, Bahaa G.M.
Published in Bioorganic chemistry (01.11.2020)
Published in Bioorganic chemistry (01.11.2020)
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Mineralogy and geochemistry of Gabal El-Ineigi Granite and associated fluorite veins, Central Eastern Desert, Egypt: application of fluid inclusions to fluorite genesis
Salem, I.A., Abdel-Moneum, A.A., Shazly, A.G., El-Shibiny, N.H.
Published in Journal of African earth sciences (1994) (2001)
Published in Journal of African earth sciences (1994) (2001)
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Novel 5α-Reductase Inhibitors: Synthesis, Structure−Activity Studies, and Pharmacokinetic Profile of Phenoxybenzoylphenyl Acetic Acids
Salem, Ola I. A, Frotscher, Martin, Scherer, Christiane, Neugebauer, Alexander, Biemel, Klaus, Streiber, Martina, Maas, Ruth, Hartmann, Rolf W
Published in Journal of medicinal chemistry (26.01.2006)
Published in Journal of medicinal chemistry (26.01.2006)
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Journal Article
6-Substituted 3,4-Dihydro-naphthalene-2-carboxylic Acids: Synthesis and Structure-Activity Studies in a Novel Class of Human 5 Reductase Inhibitors
Baston, Eckhard, Salem, Ola I.A., Hartmann, Rolf W.
Published in Journal of enzyme inhibition and medicinal chemistry (2002)
Published in Journal of enzyme inhibition and medicinal chemistry (2002)
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Journal Article
6-Substituted 3,4-Dihydro-naphthalene-2-carboxylic Acids: Synthesis and Structure-Activity Studies in a Novel Class of Human 5α Reductase Inhibitors
Baston, Eckhard, Salem, Ola I.A., Hartmann, Rolf W.
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2002)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2002)
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