Biochemical and Pharmacological Characterization of 2-(9-(2-Piperidinoethoxy)-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yloxymethyl)-4-(1-methylethyl)-6-methoxy-1,2-benzisothiazol-3(2H)-one-1,1-dioxide (SSR69071), a Novel, Orally Active Elastase Inhibitor
Kapui, Zoltan, Varga, Marton, Urban-Szabo, Katalin, Mikus, Endre, Szabo, Tibor, Szeredi, Judit, Batori, Sandor, Finance, Olivier, Aranyi, Peter
Published in The Journal of pharmacology and experimental therapeutics (01.05.2003)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2003)
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Evaluation of SSR161421, a novel orally active adenosine A3 receptor antagonist on pharmacology models
Mikus, Endre G., Szeredi, Judit, Boer, Kinga, Tímári, Géza, Finet, Michel, Aranyi, Péter, Galzin, Anne-Marie
Published in European journal of pharmacology (15.01.2013)
Published in European journal of pharmacology (15.01.2013)
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Interaction of SSR161421, a novel specific adenosine A3 receptor antagonist with adenosine A3 receptor agonists both in vitro and in vivo
Mikus, Endre G., Boér, Kinga, Timári, Géza, Urbán-Szabó, Katalin, Kapui, Zoltán, Szeredi, Judit, Gerber, Katalin, Szabó, Tibor, Bátori, Sándor, Finet, Michel, Arányi, Péter, Galzin, Anne-Marie
Published in European journal of pharmacology (15.01.2013)
Published in European journal of pharmacology (15.01.2013)
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Journal Article
Interaction of SSR161421, a novel specific adenosine A(3) receptor antagonist with adenosine A(3) receptor agonists both in vitro and in vivo
Mikus, Endre G, Boér, Kinga, Timári, Géza, Urbán-Szabó, Katalin, Kapui, Zoltán, Szeredi, Judit, Gerber, Katalin, Szabó, Tibor, Bátori, Sándor, Finet, Michel, Arányi, Péter, Galzin, Anne-Marie
Published in European journal of pharmacology (15.01.2013)
Published in European journal of pharmacology (15.01.2013)
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Journal Article
TRIAZOLO[1,5-A]QUINOLINES AS ADENOSINE A3 RECEPTOR LIGANDS
BOER KINGA, VARGANE SZEREDI JUDIT, SZLAVIK ZOLTAN, FINET MICHEL, TIMARI GEZA, URBAN SZABO KATALIN, SUSAN EDIT, KAPUI ZOLTAN, SZABO TIBOR, BATORI SANDOR, MIKUS ENDRE
Year of Publication 23.03.2010
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Year of Publication 23.03.2010
Patent
Biochemical and Pharmacological Characterization of 2-(9-(2-Piperidinoethoxy)-4-oxo-4 H -pyrido[1,2- a ]pyrimidin-2-yloxymethyl)-4-(1-methylethyl)-6-methoxy-1,2-benzisothiazol-3(2 H )-one-1,1-dioxide (SSR69071), a Novel, Orally Active Elastase Inhibitor
Kapui, Zoltán, Varga, Márton, Urban-Szabó, Katalin, Mikus, Endre, Szabó, Tibor, Szeredi, Judit, Bátori, Sándor, Finance, Olivier, Arányi, Péter
Published in The Journal of pharmacology and experimental therapeutics (01.05.2003)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2003)
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Journal Article
ΠΑΡΑΓΩΓΑ ΑΜΙΝΟΚΙΝΟΛΙΝΗΣ ΚΑΙ Η ΧΡΗΣΗ ΤΟΥΣ ΩΣ ΣΥΝΔΕΤΕΣ ΤΩΝ Α3 ΑΔΕΝΟΣΙΝΗΣ
BOER KINGA, VARGANE SZEREDI JUDIT, FINET MICHEL, TIMARI GEZA, GERBER KATALIN, KAPUI ZOLTAN, ARANYI PETER, BATORI SANDOR, MIKUS ENDRE, URBAN-SZABO KATALIN
Year of Publication 19.06.2013
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Year of Publication 19.06.2013
Patent
TRIAZOLO [1,5-A] QUINOLINES AS ADENOSINE A3 RECEPTOR LIGANDS
VARGANE SZEREDI, JUDIT, BOER, KINGA, FINET, MICHEL, URBAN SZABO, KATALIN, KAPUI, ZOLTAN, TIMARI, GEZA, MIKUS, ENDRE, SUSAN, EDIT, SZLAVIK, ZOLTAN, SZABO, TIBOR, BATORI, SANDOR
Year of Publication 15.05.2013
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Year of Publication 15.05.2013
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Compounds
Susan, Edit, Boer, Kinga, Kapui, Zoltan, Timari, Geza, Batori, Sandor, Szlavik, Zoltan, Mikus, Endre, Vargane Szeredi, Judit, Finet, Michel, Urban Szabo, Katalin, Szabo, Tibor
Year of Publication 25.12.2012
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Year of Publication 25.12.2012
Patent
Compounds
BOER KINGA, VARGANE SZEREDI JUDIT, SZLAVIK ZOLTAN, FINET MICHEL, TIMARI GEZA, URBAN SZABO KATALIN, SUSAN EDIT, KAPUI ZOLTAN, SZABO TIBOR, BATORI SANDOR, MIKUS ENDRE
Year of Publication 25.12.2012
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Year of Publication 25.12.2012
Patent
TRIAZOLO [1,5-a]QUINOLINES AS ADENOSINE A3 RECEPTOR LIGANDS
VARGANE SZEREDI, JUDIT, BOER, KINGA, FINET, MICHEL, URBAN SZABO, KATALIN, KAPUI, ZOLTAN, TIMARI, GEZA, MIKUS, ENDRE, SUSAN, EDIT, SZLAVIK, ZOLTAN, SZABO, TIBOR, BATORI, SANDOR
Year of Publication 27.08.2012
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Year of Publication 27.08.2012
Patent
Triazolo [1, 5-a] quinolines as adenosine A3 receptor ligands
VARGANE SZEREDI, JUDIT, BOER, KINGA, FINET, MICHEL, URBAN SZABO, KATALIN, KAPUI, ZOLTAN, TIMARI, GEZA, MIKUS, ENDRE, SUSAN, EDIT, SZLAVIK, ZOLTAN, SZABO, TIBOR, BATORI, SANDOR
Year of Publication 05.07.2012
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Year of Publication 05.07.2012
Patent
TRIAZOLO [1, 5-A] QUINOLINES AS ADENOSINE A3 RECEPTOR LIGANDS
SZABÓ, Tibor, KAPUI, Zoltán, SZLÁVIK, Zoltán, FINET, Michel, BOÉR, Kinga, MIKUS, Endre, SUSÁN, Edit, VARGÁNÉ SZEREDI, Judit, URBÁN SZABÓ, Katalin, BÁTORI, Sándor, TÍMÁRI, Géza
Year of Publication 20.06.2012
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Year of Publication 20.06.2012
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TRIAZOLO [1, 5-A] QUINOLINES AS ADENOSINE A3 RECEPTOR LIGANDS
VARGANE SZEREDI, JUDIT, BOER, KINGA, FINET, MICHEL, URBAN SZABO, KATALIN, KAPUI, ZOLTAN, TIMARI, GEZA, MIKUS, ENDRE, SUSAN, EDIT, SZLAVIK, ZOLTAN, SZABO, TIBOR, BATORI, SANDOR
Year of Publication 30.03.2012
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Year of Publication 30.03.2012
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AMINOQUINOLINE DERIVATIVES AND THEIR USE AS ADENOSINE A3 LIGANDS
GERBER, KATALIN, VARGANE SZEREDI, JUDIT, BOER, KINGA, FINET, MICHEL, ARANYI, PETER, KAPUI, ZOLTAN, TIMARI, GEZA, MIKUS, ENDRE, URBAN-SZABO, KATALIN, BATORI, SANDOR
Year of Publication 21.02.2012
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Year of Publication 21.02.2012
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Aminoquinoline derivatives and their use as adenosine A3 ligands
Aranyi, Peter, Batori, Sandor, Timari, Geza, Boer, Kinga, Kapui, Zoltan, Mikus, Endre, Urban-Szabo, Katalin, Gerber, Katalin, Vargane Szeredi, Judit, Finet, Michel
Year of Publication 06.12.2011
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Year of Publication 06.12.2011
Patent
Aminoquinoline derivatives and their use as adenosine A3 ligands
BOER KINGA, VARGANE SZEREDI JUDIT, FINET MICHEL, TIMARI GEZA, GERBER KATALIN, KAPUI ZOLTAN, ARANYI PETER, BATORI SANDOR, MIKUS ENDRE, URBAN-SZABO KATALIN
Year of Publication 06.12.2011
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Year of Publication 06.12.2011
Patent
TRIAZOLO [1, 5-A]QUINOLINES AS ADENOSINE A3 RECEPTOR LIGANDS
KAPUI, Zoltán, SZLÁVIK, Zoltán, SZABÓ, Tibor, FINET, Michel, BOÉR, Kinga, TIMÁRI, Géza, MIKUS, Endre, SUSÁN, Edit, VARGÁNÉ SZEREDI, Judit, BÁTORI, Sándor, URBÁN SZABÓ, Katalin
Year of Publication 31.08.2011
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Year of Publication 31.08.2011
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TRIAZOLO ?á1, 5-A?åQUINOLINES AS ADENOSINE A3 RECEPTOR LIGANDS
BOER KINGA, VARGANE SZEREDI JUDIT, SZLAVIK ZOLTAN, FINET MICHEL, TIMARI GEZA, URBAN SZABO KATALIN, SUSAN EDIT, KAPUI ZOLTAN, SZABO TIBOR, BATORI SANDOR, MIKUS ENDRE
Year of Publication 30.06.2011
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Year of Publication 30.06.2011
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Triazolo-[1,5A]-chinoliner som adenosin-A3-receptor ligander
VARGANE SZEREDI, JUDIT, BOER, KINGA, FINET, MICHEL, URBAN SZABO, KATALIN, KAPUI, ZOLTAN, MIKUS, ENDRE, TIMARI, GEZA, SUSAN, EDIT, SZLAVIK, ZOLTAN, SZABO, TIBOR, BATORI, SANDOR
Year of Publication 27.06.2011
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Year of Publication 27.06.2011
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