Discovery of a Potent, Selective Protein Tyrosine Phosphatase 1B Inhibitor Using a Linked-Fragment Strategy
Szczepankiewicz, Bruce G, Liu, Gang, Hajduk, Philip J, Abad-Zapatero, Cele, Pei, Zhonghua, Xin, Zhili, Lubben, Thomas H, Trevillyan, James M, Stashko, Michael A, Ballaron, Stephen J, Liang, Heng, Huang, Flora, Hutchins, Charles W, Fesik, Stephen W, Jirousek, Michael R
Published in Journal of the American Chemical Society (09.04.2003)
Published in Journal of the American Chemical Society (09.04.2003)
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Journal Article
Discovery of piperidine-aryl urea-based stearoyl-CoA desaturase 1 inhibitors
Xin, Zhili, Zhao, Hongyu, Serby, Michael D., Liu, Bo, Liu, Mei, Szczepankiewicz, Bruce G., Nelson, Lissa T.J., Smith, Harriet T., Suhar, Tom S., Janis, Rich S., Cao, Ning, Camp, Heidi S., Collins, Christine A., Sham, Hing L., Surowy, Teresa K., Liu, Gang
Published in Bioorganic & medicinal chemistry (01.08.2008)
Published in Bioorganic & medicinal chemistry (01.08.2008)
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Journal Article
Discovery of Potent, Highly Selective, and Orally Bioavailable Pyridine Carboxamide c-Jun NH2-Terminal Kinase Inhibitors
Zhao, Hongyu, Serby, Michael D, Xin, Zhili, Szczepankiewicz, Bruce G, Liu, Mei, Kosogof, Christi, Liu, Bo, Nelson, Lissa T. J, Johnson, Eric F, Wang, Sanyi, Pederson, Terry, Gum, Rebecca J, Clampit, Jill E, Haasch, Deanna L, Abad-Zapatero, Cele, Fry, Elizabeth H, Rondinone, Cristina, Trevillyan, James M, Sham, Hing L, Liu, Gang
Published in Journal of medicinal chemistry (27.07.2006)
Published in Journal of medicinal chemistry (27.07.2006)
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Journal Article
Synthesis of Purines and Other Fused Imidazoles from Acyclic Amidines and Guanidines
Szczepankiewicz, Bruce G, Rohde, Jeffrey J, Kurukulasuriya, Ravi
Published in Organic letters (28.04.2005)
Published in Organic letters (28.04.2005)
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Journal Article
Identification of a monoacid-Based, cell permeable, selective inhibitor of protein tyrosine phosphatase 1B
Xin, Zhili, Liu, Gang, Abad-Zapatero, Cele, Pei, Zhonghua, Szczepankiewicz, Bruce G., Li, Xiaofeng, Zhang, Tianyuan, Hutchins, Charles W., Hajduk, Philip J., Ballaron, Stephen J., Stashko, Michael A., Lubben, Thomas H., Trevillyan, James M., Jirousek, Michael R.
Published in Bioorganic & medicinal chemistry letters (17.11.2003)
Published in Bioorganic & medicinal chemistry letters (17.11.2003)
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Journal Article
Xanthine mimetics as potent dipeptidyl peptidase IV inhibitors
Kurukulasuriya, Ravi, Rohde, Jeffrey J., Szczepankiewicz, Bruce G., Basha, Fatima, Lai, Chunqui, Jae, Hwan-Soo, Winn, Martin, Stewart, Kent D., Longenecker, Kenton L., Lubben, Thomas W., Ballaron, Stephen J., Sham, Hing L., von Geldern, Thomas W.
Published in Bioorganic & medicinal chemistry letters (15.12.2006)
Published in Bioorganic & medicinal chemistry letters (15.12.2006)
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Journal Article
Pyrrolidine-3-carboxylic Acids as Endothelin Antagonists. 4. Side Chain Conformational Restriction Leads to ETB Selectivity
von Geldern, Thomas W, Tasker, Andrew S, Sorensen, Bryan K, Winn, Martin, Szczepankiewicz, Bruce G, Dixon, Douglas B, Chiou, William J, Wang, Liming, Wessale, Jerry L, Adler, Andy, Marsh, Kennan C, Nguyen, Bach, Opgenorth, Terry J
Published in Journal of medicinal chemistry (09.09.1999)
Published in Journal of medicinal chemistry (09.09.1999)
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Journal Article
The Synthesis of Bromomethyltrifluoroborates through Continuous Flow Chemistry
Broom, Toby, Hughes, Mark, Szczepankiewicz, Bruce G., Ace, Karl, Hagger, Ben, Lacking, Gary, Chima, Ranjit, Marchbank, Graeme, Alford, Gareth, Evans, Paul, Cunningham, Christopher, Roberts, John C., Perni, Robert B., Berry, Malcolm, Rutter, Andrew, Watson, Simon A.
Published in Organic process research & development (21.11.2014)
Published in Organic process research & development (21.11.2014)
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Journal Article
Aminopyridine-Based c-Jun N-Terminal Kinase Inhibitors with Cellular Activity and Minimal Cross-Kinase Activity
Szczepankiewicz, Bruce G, Kosogof, Christi, Nelson, Lissa T. J, Liu, Gang, Liu, Bo, Zhao, Hongyu, Serby, Michael D, Xin, Zhili, Liu, Mei, Gum, Rebecca J, Haasch, Deanna L, Wang, Sanyi, Clampit, Jill E, Johnson, Eric F, Lubben, Thomas H, Stashko, Michael A, Olejniczak, Edward T, Sun, Chaohong, Dorwin, Sarah A, Haskins, Kristi, Abad-Zapatero, Cele, Fry, Elizabeth H, Hutchins, Charles W, Sham, Hing L, Rondinone, Cristina M, Trevillyan, James M
Published in Journal of medicinal chemistry (15.06.2006)
Published in Journal of medicinal chemistry (15.06.2006)
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Journal Article
Selective Protein Tyrosine Phosphatase 1B Inhibitors: Targeting the Second Phosphotyrosine Binding Site with Non-Carboxylic Acid-Containing Ligands
Liu, Gang, Xin, Zhili, Liang, Heng, Abad-Zapatero, Cele, Hajduk, Philip J, Janowick, David A, Szczepankiewicz, Bruce G, Pei, Zhonghua, Hutchins, Charles W, Ballaron, Stephen J, Stashko, Michael A, Lubben, Thomas H, Berg, Cathy E, Rondinone, Cristina M, Trevillyan, James M, Jirousek, Michael R
Published in Journal of medicinal chemistry (31.07.2003)
Published in Journal of medicinal chemistry (31.07.2003)
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Journal Article
Isoxazole carboxylic acids as protein tyrosine phosphatase 1B (PTP1B) inhibitors
Zhao, Hongyu, Liu, Gang, Xin, Zhili, Serby, Michael D., Pei, Zhonghua, Szczepankiewicz, Bruce G., Hajduk, Philip J., Abad-Zapatero, Cele, Hutchins, Charles W., Lubben, Thomas H., Ballaron, Stephen J., Haasch, Deanna L., Kaszubska, Wiweka, Rondinone, Cristina M., Trevillyan, James M., Jirousek, Michael R.
Published in Bioorganic & medicinal chemistry letters (15.11.2004)
Published in Bioorganic & medicinal chemistry letters (15.11.2004)
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Journal Article
Inhibition of Protein Tyrosine Phosphatase 1B as a Potential Treatment of Diabetes and Obesity
Pei, Zhonghua, Liu, Gang, Lubben, Thomas H, Szczepankiewicz, Bruce G
Published in Current pharmaceutical design (01.01.2004)
Published in Current pharmaceutical design (01.01.2004)
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Journal Article
Discovery and Pharmacological Evaluation of Growth Hormone Secretagogue Receptor Antagonists
Xin, Zhili, Serby, Michael D, Zhao, Hongyu, Kosogof, Christi, Szczepankiewicz, Bruce G, Liu, Mei, Hutchins, Charles W, Sarris, Kathy A, Hoff, Ethan D, Falls, H. Douglas, Lin, Chun W, Ogiela, Christopher A, Collins, Christine A, Brune, Michael E, Bush, Eugene N, Droz, Brian A, Fey, Thomas A, Knourek-Segel, Victoria E, Shapiro, Robin, Jacobson, Peer B, Beno, David W. A, Turner, Teresa M, Sham, Hing L, Liu, Gang
Published in Journal of medicinal chemistry (27.07.2006)
Published in Journal of medicinal chemistry (27.07.2006)
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Journal Article
2,4-Diaminopyrimidine Derivatives as Potent Growth Hormone Secretagogue Receptor Antagonists
Serby, Michael D., Zhao, Hongyu, Szczepankiewicz, Bruce G., Kosogof, Christi, Xin, Zhili, Liu, Bo, Liu, Mei, Nelson, Lissa T. J., Kaszubska, Wiweka, Falls, H. Douglas, Schaefer, Verlyn, Bush, Eugene N., Shapiro, Robin, Droz, Brian A., Knourek-Segel, Victoria E., Fey, Thomas A., Brune, Michael E., Beno, David W. A., Turner, Theresa M., Collins, Christine A., Jacobson, Peer B., Sham, Hing L., Liu, Gang
Published in Journal of medicinal chemistry (20.04.2006)
Published in Journal of medicinal chemistry (20.04.2006)
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Journal Article
Aminopyridine carboxamides as c-Jun N-terminal kinase inhibitors: Targeting the gatekeeper residue and beyond
Liu, Gang, Zhao, Hongyu, Liu, Bo, Xin, Zhili, Liu, Mei, Kosogof, Christi, Szczepankiewicz, Bruce G., Wang, Sanyi, Clampit, Jill E., Gum, Rebecca J., Haasch, Deanna L., Trevillyan, James M., Sham, Hing L.
Published in Bioorganic & medicinal chemistry letters (15.11.2006)
Published in Bioorganic & medicinal chemistry letters (15.11.2006)
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Journal Article
Potent, selective inhibitors of protein tyrosine phosphatase 1B
Xin, Zhili, Oost, Thorsten K, Abad-Zapatero, Cele, Hajduk, Philip J, Pei, Zhonghua, Szczepankiewicz, Bruce G, Hutchins, Charles W, Ballaron, Steve J, Stashko, Mike A, Lubben, Tom, Trevillyan, James M, Jirousek, Mike R, Liu, Gang
Published in Bioorganic & medicinal chemistry letters (02.06.2003)
Published in Bioorganic & medicinal chemistry letters (02.06.2003)
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Journal Article
New Antimitotic Agents with Activity in Multi-Drug-Resistant Cell Lines and in Vivo Efficacy in Murine Tumor Models
Szczepankiewicz, Bruce G, Liu, Gang, Jae, Hwan-Soo, Tasker, Andrew S, Gunawardana, Indrani W, von Geldern, Thomas W, Gwaltney, Stephen L, Wu-Wong, J. Ruth, Gehrke, Laura, Chiou, William J, Credo, R. Bruce, Alder, Jeffery D, Nukkala, Michael A, Zielinski, Nicolette A, Jarvis, Ken, Mollison, Karl W, Frost, David J, Bauch, Joy L, Hui, Yu Hua, Claiborne, Akiyo K, Li, Qun, Rosenberg, Saul H
Published in Journal of medicinal chemistry (06.12.2001)
Published in Journal of medicinal chemistry (06.12.2001)
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