Ultra-long-acting tunable biodegradable and removable controlled release implants for drug delivery
Benhabbour, S Rahima, Kovarova, Martina, Jones, Clinton, Copeland, Daijha J, Shrivastava, Roopali, Swanson, Michael D, Sykes, Craig, Ho, Phong T, Cottrell, Mackenzie L, Sridharan, Anush, Fix, Samantha M, Thayer, Orrin, Long, Julie M, Hazuda, Daria J, Dayton, Paul A, Mumper, Russell J, Kashuba, Angela D M, Victor Garcia, J
Published in Nature communications (20.09.2019)
Published in Nature communications (20.09.2019)
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Ultra-long-acting removable drug delivery system for HIV treatment and prevention
Kovarova, Martina, Benhabbour, S Rahima, Massud, Ivana, Spagnuolo, Rae Ann, Skinner, Brianna, Baker, Caroline E, Sykes, Craig, Mollan, Katie R, Kashuba, Angela D M, García-Lerma, J Gerardo, Mumper, Russell J, Garcia, J Victor
Published in Nature communications (08.10.2018)
Published in Nature communications (08.10.2018)
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Ultra-long-acting in-situ forming implants with cabotegravir protect female macaques against rectal SHIV infection
Young, Isabella C, Massud, Ivana, Cottrell, Mackenzie L, Shrivastava, Roopali, Maturavongsadit, Panita, Prasher, Alka, Wong-Sam, Andres, Dinh, Chuong, Edwards, Tiancheng, Mrotz, Victoria, Mitchell, James, Seixas, Josilene Nascimento, Pallerla, Aryani, Thorson, Allison, Schauer, Amanda, Sykes, Craig, De la Cruz, Gabriela, Montgomery, Stephanie A, Kashuba, Angela D M, Heneine, Walid, Dobard, Charles W, Kovarova, Martina, Garcia, J Victor, García-Lerma, J Gerardo, Benhabbour, S Rahima
Published in Nature communications (09.02.2023)
Published in Nature communications (09.02.2023)
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EFdA efficiently suppresses HIV replication in the male genital tract and prevents penile HIV acquisition
Kovarova, Martina, Wessel, Sarah E, Johnson, Claire E, Anderson, Shelby V, Cottrell, Mackenzie L, Sykes, Craig, Cohen, Myron S, Garcia, J Victor
Published in mBio (31.08.2023)
Published in mBio (31.08.2023)
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Author Correction: Ultra-long-acting in-situ forming implants with cabotegravir protect female macaques against rectal SHIV infection
Young, Isabella C, Massud, Ivana, Cottrell, Mackenzie L, Shrivastava, Roopali, Maturavongsadit, Panita, Prasher, Alka, Wong-Sam, Andres, Dinh, Chuong, Edwards, Tiancheng, Mrotz, Victoria, Mitchell, James, Seixas, Josilene Nascimento, Pallerla, Aryani, Thorson, Allison, Schauer, Amanda, Sykes, Craig, De la Cruz, Gabriela, Montgomery, Stephanie A, Kashuba, Angela D M, Heneine, Walid, Dobard, Charles W, Kovarova, Martina, Garcia, J Victor, Garcίa-Lerma, J Gerardo, Benhabbour, S Rahima
Published in Nature communications (05.02.2024)
Published in Nature communications (05.02.2024)
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Dolutegravir pharmacokinetics in the genital tract and colorectum of HIV-negative men after single and multiple dosing
Greener, Benjamin N, Patterson, Kristine B, Prince, Heather M A, Sykes, Craig S, Adams, Jessica L, Dumond, Julie B, Shaheen, Nicholas J, Madanick, Ryan D, Dellon, Evan S, Cohen, Myron S, Kashuba, Angela D M
Published in Journal of acquired immune deficiency syndromes (1999) (01.09.2013)
Published in Journal of acquired immune deficiency syndromes (1999) (01.09.2013)
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Pregnancy related hormones increase CYP3A mediated buprenorphine metabolism in human hepatocytes: a comparison to CYP3A substrates nifedipine and midazolam
Fashe, Muluneh M, Miner, Taryn A, Fallon, John K, Schauer, Amanda P, Sykes, Craig, Smith, Philip C, Lee, Craig R
Published in Frontiers in pharmacology (05.07.2023)
Published in Frontiers in pharmacology (05.07.2023)
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Validation of an LC–MS/MS assay to simultaneously monitor the intracellular active metabolites of tenofovir, emtricitabine, and lamivudine in dried blood spots
Schauer, Amanda P., Sykes, Craig, Cottrell, Mackenzie L., Prince, Heather, Kashuba, Angela D.M.
Published in Journal of pharmaceutical and biomedical analysis (05.02.2018)
Published in Journal of pharmaceutical and biomedical analysis (05.02.2018)
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Pregnancy-Related Hormones Increase UGT1A1-Mediated Labetalol Metabolism in Human Hepatocytes
Khatri, Raju, Fallon, John K, Sykes, Craig, Kulick, Natasha, Rementer, Rebecca J B, Miner, Taryn A, Schauer, Amanda P, Kashuba, Angela D M, Boggess, Kim A, Brouwer, Kim L R, Smith, Philip C, Lee, Craig R
Published in Frontiers in pharmacology (15.04.2021)
Published in Frontiers in pharmacology (15.04.2021)
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Next-Generation Contraceptive Intravaginal Ring: Comparison of Etonogestrel and Ethinyl Estradiol In Vitro and In Vivo Release from 3D-Printed Intravaginal Ring and NuvaRing
Young, Isabella C., Thorson, Allison L., Cottrell, Mackenzie L., Sykes, Craig, Schauer, Amanda P., Sellers, Rani S., Janusziewicz, Rima, Vincent, Kathleen L., Benhabbour, Soumya Rahima
Published in Pharmaceutics (02.08.2024)
Published in Pharmaceutics (02.08.2024)
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A multicompartment population PK model to predict tenofovir and emtricitabine mucosal tissue concentrations for HIV prevention
Leung, Erick, Cottrell, Mackenzie L., Sykes, Craig, White, Nicole, Kashuba, Angela D. M., Dumond, Julie B.
Published in CPT: pharmacometrics and systems pharmacology (01.12.2023)
Published in CPT: pharmacometrics and systems pharmacology (01.12.2023)
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Application of a Scavenger Receptor A1-Targeted Polymeric Prodrug Platform for Lymphatic Drug Delivery in HIV
Stevens, David M, Adiseshaiah, Pavan, Dasa, Siva S. K, Potter, Tim M, Skoczen, Sarah L, Snapp, Kelsie S, Cedrone, Edward, Patel, Nimit, Busman-Sahay, Kathleen, Rosen, Elias P, Sykes, Craig, Cottrell, Mackenzie, Dobrovolskaia, Marina A, Estes, Jacob D, Kashuba, Angela D. M, Stern, Stephan T
Published in Molecular pharmaceutics (05.10.2020)
Published in Molecular pharmaceutics (05.10.2020)
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Dose-Ranging Plasma and Genital Tissue Pharmacokinetics and Biodegradation of Ultra-Long-Acting Cabotegravir In Situ Forming Implant
Young, Isabella C, Thorson, Allison L, Shrivastava, Roopali, Sykes, Craig, Schauer, Amanda P, Cottrell, Mackenzie L, Kashuba, Angela D M, Benhabbour, Soumya Rahima
Published in Pharmaceutics (13.05.2023)
Published in Pharmaceutics (13.05.2023)
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Concentrations of Pro-Inflammatory Cytokines Are Not Associated with Senescence Marker p16INK4a or Predictive of Intracellular Emtricitabine/Tenofovir Metabolite and Endogenous Nucleotide Exposures in Adults with HIV Infection
Maas, Brian M, Francis, Owen, Mollan, Katie R, Lee, Cynthia, Cottrell, Mackenzie L, Prince, Heather M A, Sykes, Craig, Trezza, Christine, Torrice, Chad, White, Nicole, Malone, Stephanie, Hudgens, Michael G, Sharpless, Norman E, Dumond, Julie B
Published in PloS one (01.12.2016)
Published in PloS one (01.12.2016)
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Predicting Efavirenz Concentrations in the Brain Tissue of HIV‐Infected Individuals and Exploring their Relationship to Neurocognitive Impairment
Srinivas, Nithya, Joseph, Sarah Beth, Robertson, Kevin, Kincer, Laura P., Menezes, Prema, Adamson, Lourdes, Schauer, Amanda P., Blake, Kimberly H., White, Nicole, Sykes, Craig, Luciw, Paul, Eron, Joseph J., Forrest, Alan, Price, Richard W., Spudich, Serena, Swanstrom, Ronald, Kashuba, Angela D.M.
Published in Clinical and translational science (01.05.2019)
Published in Clinical and translational science (01.05.2019)
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Mucosal tissue pharmacokinetics of the integrase inhibitor raltegravir in a humanized mouse model: Implications for HIV pre-exposure prophylaxis
Veselinovic, Milena, Yang, Kuo-Hsiung, Sykes, Craig, Remling-Mulder, Leila, Kashuba, Angela D.M, Akkina, Ramesh
Published in Virology (New York, N.Y.) (01.02.2016)
Published in Virology (New York, N.Y.) (01.02.2016)
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A Translational Pharmacology Approach to Predicting Outcomes of Preexposure Prophylaxis Against HIV in Men and Women Using Tenofovir Disoproxil Fumarate With or Without Emtricitabine
Cottrell, Mackenzie L., Yang, Kuo H., Prince, Heather M. A., Sykes, Craig, White, Nicole, Malone, Stephanie, Dellon, Evan S., Madanick, Ryan D., Shaheen, Nicholas J., Hudgens, Michael G., Wulff, Jacob, Patterson, Kristine B., Nelson, Julie A. E., Kashuba, Angela D. M.
Published in The Journal of infectious diseases (01.07.2016)
Published in The Journal of infectious diseases (01.07.2016)
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