Tirzepatide is an imbalanced and biased dual GIP and GLP-1 receptor agonist
Willard, Francis S, Douros, Jonathan D, Gabe, Maria Bn, Showalter, Aaron D, Wainscott, David B, Suter, Todd M, Capozzi, Megan E, van der Velden, Wijnand Jc, Stutsman, Cynthia, Cardona, Guemalli R, Urva, Shweta, Emmerson, Paul J, Holst, Jens J, D'Alessio, David A, Coghlan, Matthew P, Rosenkilde, Mette M, Campbell, Jonathan E, Sloop, Kyle W
Published in JCI insight (03.09.2020)
Published in JCI insight (03.09.2020)
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Structural determinants of dual incretin receptor agonism by tirzepatide
Sun, Bingfa, Willard, Francis S, Feng, Dan, Alsina-Fernandez, Jorge, Chen, Qi, Vieth, Michal, Ho, Joseph D, Showalter, Aaron D, Stutsman, Cynthia, Ding, Liyun, Suter, Todd M, Dunbar, James D, Carpenter, John W, Mohammed, Faiz Ahmad, Aihara, Eitaro, Brown, Robert A, Bueno, Ana B, Emmerson, Paul J, Moyers, Julie S, Kobilka, Tong Sun, Coghlan, Matthew P, Kobilka, Brian K, Sloop, Kyle W
Published in Proceedings of the National Academy of Sciences - PNAS (29.03.2022)
Published in Proceedings of the National Academy of Sciences - PNAS (29.03.2022)
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A Novel Nociceptin Receptor Antagonist LY2940094 Inhibits Excessive Feeding Behavior in Rodents: A Possible Mechanism for the Treatment of Binge Eating Disorder
Statnick, Michael A, Chen, Yanyun, Ansonoff, Michael, Witkin, Jeffrey M, Rorick-Kehn, Linda, Suter, Todd M, Song, Min, Hu, Charlie, Lafuente, Celia, Jiménez, Alma, Benito, Ana, Diaz, Nuria, Martínez-Grau, Maria Angeles, Toledo, Miguel A, Pintar, John E
Published in The Journal of pharmacology and experimental therapeutics (01.02.2016)
Published in The Journal of pharmacology and experimental therapeutics (01.02.2016)
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Regulation of Endogenous (Male) Rodent GLP-1 Secretion and Human Islet Insulin Secretion by Antagonism of Somatostatin Receptor 5
Farb, Thomas B, Adeva, Marta, Beauchamp, Thomas J, Cabrera, Over, Coates, David A, Meredith, Tamika DeShea, Droz, Brian A, Efanov, Alexander, Ficorilli, James V, Gackenheimer, Susan L, Martinez-Grau, Maria A, Molero, Victoriano, Ruano, Gema, Statnick, Michael A, Suter, Todd M, Syed, Samreen K, Toledo, Miguel A, Willard, Francis S, Zhou, Xin, Bokvist, Krister B, Barrett, David G
Published in Endocrinology (Philadelphia) (01.11.2017)
Published in Endocrinology (Philadelphia) (01.11.2017)
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An Allosteric Potentiator of the Dopamine D1 Receptor Increases Locomotor Activity in Human D1 Knock-In Mice without Causing Stereotypy or Tachyphylaxis
Svensson, Kjell A, Heinz, Beverly A, Schaus, John M, Beck, James P, Hao, Junliang, Krushinski, Joseph H, Reinhard, Matthew R, Cohen, Michael P, Hellman, Sarah L, Getman, Brian G, Wang, Xushan, Menezes, Michelle M, Maren, Deanna L, Falcone, Julie F, Anderson, Wesley H, Wright, Rebecca A, Morin, S Michelle, Knopp, Kelly L, Adams, Benjamin L, Rogovoy, Borys, Okun, Ilya, Suter, Todd M, Statnick, Michael A, Gehlert, Donald R, Nelson, David L, Lucaites, Virginia L, Emkey, Renee, DeLapp, Neil W, Wiernicki, Todd R, Cramer, Jeffrey W, Yang, Charles R, Bruns, Robert F
Published in The Journal of pharmacology and experimental therapeutics (01.01.2017)
Published in The Journal of pharmacology and experimental therapeutics (01.01.2017)
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Journal Article
Pharmacological characterization of the cannabinoid CB1 receptor PET ligand ortholog, [3H]MePPEP
SUTER, Todd M, CHESTERFIELD, Amy K, CHUN BAO, SCHAUS, John M, KRUSHINSKI, Joseph H, STATNICK, Michael A, FELDER, Christian C
Published in European journal of pharmacology (15.12.2010)
Published in European journal of pharmacology (15.12.2010)
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Journal Article
Structure activity relationship studies of carboxamido-biaryl ethers as opioid receptor antagonists (OpRAs). Part 2
Takeuchi, Kumiko, Holloway, William G., Mitch, Charles H., Quimby, Steven J., McKinzie, Jamie H., Suter, Todd M., Statnick, Michael A., Surface, Peggy L., Emmerson, Paul J., Thomas, Elizabeth M., Siegel, Miles G.
Published in Bioorganic & medicinal chemistry letters (15.12.2007)
Published in Bioorganic & medicinal chemistry letters (15.12.2007)
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Journal Article
Structure–activity relationship studies of carboxamido-biaryl ethers as opioid receptor antagonists (OpRAs). Part 1
Takeuchi, Kumiko, Holloway, William G., McKinzie, Jamie H., Suter, Todd M., Statnick, Michael A., Surface, Peggy L., Emmerson, Paul J., Thomas, Elizabeth M., Siegel, Miles G., Matt, James E., Wolfe, Chad N., Mitch, Charles H.
Published in Bioorganic & medicinal chemistry letters (01.10.2007)
Published in Bioorganic & medicinal chemistry letters (01.10.2007)
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Journal Article
Na +-dependent high affinity binding of [ 3H]LY515300, a 3,4-dimethyl-4-(3-hydroxyphenyl)piperidine opioid receptor inverse agonist
Statnick, Michael A., Suter, Todd M., Gackenheimer, Susan L., Emmerson, Paul J., Quimby, Steve J., Gehlert, Donald R., Wheeler, William J., Mitch, Charles H.
Published in European journal of pharmacology (15.12.2003)
Published in European journal of pharmacology (15.12.2003)
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Journal Article
Decreased Expression Of apM1 in Omental and Subcutaneous Adipose Tissue of HumansWith Type 2 Diabetes
Statnick, Michael A., Beavers, Lisa S., Conner, Laura J., Corominola, Helena, Johnson, Dwayne, Hammond, Craig D., Rafaeloff-Phail, Ronit, Seng, Thomas, Suter, Todd M., Sluka, James P., Ravussin, Eric, Gadski, Robert A., Caro, Jose F.
Published in Journal of diabetes research (01.01.2000)
Published in Journal of diabetes research (01.01.2000)
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Journal Article
Antagonism of opioid receptors reduces body fat in obese rats by decreasing food intake and stimulating lipid utilization
Statnick, Michael A., Tinsley, Frank C., Eastwood, Brian J., Suter, Todd M., Mitch, Charles H., Heiman, Mark L.
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.06.2003)
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.06.2003)
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Journal Article
Pharmacological characterization of the cannabinoid CB 1 receptor PET ligand ortholog, [ 3H]MePPEP
Suter, Todd M., Chesterfield, Amy K., Bao, Chun, Schaus, John M., Krushinski, Joseph H., Statnick, Michael A., Felder, Christian C.
Published in European journal of pharmacology (2010)
Published in European journal of pharmacology (2010)
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Journal Article
Peptides that Regulate Food Intake: Antagonism of opioid receptors reduces body fat in obese rats by decreasing food intake and stimulating lipid utilization
Statnick, Michael A, Tinsley, Frank C, Eastwood, Brian J, Suter, Todd M, Mitch, Charles H, Heiman, Mark L
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.06.2003)
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.06.2003)
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Journal Article
Decreased expression of apM1 in omental and subcutaneous adipose tissue of humans with type 2 diabetes
Statnick, M A, Beavers, L S, Conner, L J, Corominola, H, Johnson, D, Hammond, C D, Rafaeloff-Phail, R, Seng, T, Suter, T M, Sluka, J P, Ravussin, E, Gadski, R A, Caro, J F
Published in International journal of experimental diabetes research (2000)
Published in International journal of experimental diabetes research (2000)
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Journal Article
Antagonism of opioid receptors reduces body fat in obese rats by decreasing food intake and stimulating lipid utilization
Michael A Statnick, Frank C Tinsley, Eastwood, Brian J, Suter, Todd M
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.06.2003)
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Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.06.2003)
Journal Article
Antagonism of opioid receptors reduces body fat in obese rats by decreasing food intake and stimulating lipid utilization : Peptides that regulate food intake
STATNICK, Michael A, TINSLEY, Frank C, EASTWOOD, Brian J, SUTER, Todd M, MITCH, Charles H, HEIMAN, Mark L
Published in American journal of physiology. Regulatory, integrative and comparative physiology (2003)
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Published in American journal of physiology. Regulatory, integrative and comparative physiology (2003)
Journal Article
Isolation of a gene encoding a novel spectinomycin phosphotransferase from Legionella pneumophila
SUTER, T. M, VISWANATHAN, V. K, CIANCIOTTO, N. P
Published in Antimicrobial Agents and Chemotherapy (01.06.1997)
Published in Antimicrobial Agents and Chemotherapy (01.06.1997)
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