The discovery and development of rivaroxaban, an oral, direct factor Xa inhibitor
Perzborn, Elisabeth, Roehrig, Susanne, Straub, Alexander, Kubitza, Dagmar, Misselwitz, Frank
Published in Nature reviews. Drug discovery (01.01.2011)
Published in Nature reviews. Drug discovery (01.01.2011)
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Journal Article
Pharmacological profile of asundexian, a novel, orally bioavailable inhibitor of factor XIa
Heitmeier, Stefan, Visser, Mayken, Tersteegen, Adrian, Dietze‐Torres, Julia, Glunz, Julia, Gerdes, Christoph, Laux, Volker, Stampfuss, Jan, Roehrig, Susanne
Published in Journal of thrombosis and haemostasis (01.06.2022)
Published in Journal of thrombosis and haemostasis (01.06.2022)
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Journal Article
Rivaroxaban: A New Oral Factor Xa Inhibitor
Perzborn, Elisabeth, Roehrig, Susanne, Straub, Alexander, Kubitza, Dagmar, Mueck, Wolfgang, Laux, Volker
Published in Arteriosclerosis, thrombosis, and vascular biology (01.03.2010)
Published in Arteriosclerosis, thrombosis, and vascular biology (01.03.2010)
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Journal Article
Discovery of the Novel Antithrombotic Agent 5-Chloro-N-({(5S)-2-oxo-3- [4-(3-oxomorpholin-4-yl)phenyl]-1,3-oxazolidin-5-yl}methyl)thiophene- 2-carboxamide (BAY 59-7939): An Oral, Direct Factor Xa Inhibitor
Roehrig, Susanne, Straub, Alexander, Pohlmann, Jens, Lampe, Thomas, Pernerstorfer, Josef, Schlemmer, Karl-Heinz, Reinemer, Peter, Perzborn, Elisabeth
Published in Journal of medicinal chemistry (22.09.2005)
Published in Journal of medicinal chemistry (22.09.2005)
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Journal Article
Entering the era of non-basic p1 site groups: discovery of Xarelto (Rivaroxaban)
Straub, Alexander, Roehrig, Susanne, Hillisch, Alexander
Published in Current topics in medicinal chemistry (01.02.2010)
Published in Current topics in medicinal chemistry (01.02.2010)
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Journal Article
Design, Synthesis, and Pharmacological Characterization of a Neutral, Non-Prodrug Thrombin Inhibitor with Good Oral Pharmacokinetics
Hillisch, Alexander, Gericke, Kersten M, Allerheiligen, Swen, Roehrig, Susanne, Schaefer, Martina, Tersteegen, Adrian, Schulz, Simone, Lienau, Philip, Gnoth, Mark, Puetter, Vera, Hillig, Roman C, Heitmeier, Stefan
Published in Journal of medicinal chemistry (12.11.2020)
Published in Journal of medicinal chemistry (12.11.2020)
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Journal Article
Design and Preclinical Characterization Program toward Asundexian (BAY 2433334), an Oral Factor XIa Inhibitor for the Prevention and Treatment of Thromboembolic Disorders
Roehrig, Susanne, Ackerstaff, Jens, Jiménez Núñez, Eloísa, Teller, Henrik, Ellerbrock, Pascal, Meier, Katharina, Heitmeier, Stefan, Tersteegen, Adrian, Stampfuss, Jan, Lang, Dieter, Schlemmer, Karl-Heinz, Schaefer, Martina, Gericke, Kersten M., Kinzel, Tom, Meibom, Daniel, Schmidt, Martina, Gerdes, Christoph, Follmann, Markus, Hillisch, Alexander
Published in Journal of medicinal chemistry (14.09.2023)
Published in Journal of medicinal chemistry (14.09.2023)
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Journal Article
Cover Picture: Oral, Direct Thrombin and Factor Xa Inhibitors: The Replacement for Warfarin, Leeches, and Pig Intestines? (Angew. Chem. Int. Ed. 20/2011)
Straub, Alexander, Roehrig, Susanne, Hillisch, Alexander
Published in Angewandte Chemie (International ed.) (09.05.2011)
Published in Angewandte Chemie (International ed.) (09.05.2011)
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Journal Article
Cover Picture: Oral, Direct Thrombin and FactorXa Inhibitors: The Replacement for Warfarin, Leeches, and Pig Intestines? (Angew. Chem. Int. Ed. 20/2011)
Straub, Alexander, Roehrig, Susanne, Hillisch, Alexander
Published in Angewandte Chemie International Edition (09.05.2011)
Published in Angewandte Chemie International Edition (09.05.2011)
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Journal Article
Orale, direkte Thrombin‐ und Faktor‐Xa‐Hemmer: Kommt die Ablösung für Warfarin, Blutegel und Schweinedärme?
Straub, Alexander, Roehrig, Susanne, Hillisch, Alexander
Published in Angewandte Chemie (09.05.2011)
Published in Angewandte Chemie (09.05.2011)
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Journal Article
SUBSTITUTED OXOPYRIDINE DERIVATIVES AND USE THEREOF IN THE TREATMENT OF CARDIOVASCULAR DISORDERS
CHRISTOPH GERDES, HENRIK TELLER, ADRIAN TERSTEEGEN, ANJA BUCHMUELLER, MARTINA SCHAEFER, ELOISA JIMENEZ NUNEZ, TOM KINZEL, KARL-HEINZ SCHLEMMER, JUERGEN KLAR, MARTINA VICTORIA SCHMIDT, JULIA STRASSBURGER, STEFAN HEITMEIER, SUSANNE ROEHRIG, ALEXANDER HILLISCH, HARTMUT SCHIROK
Year of Publication 26.04.2018
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Year of Publication 26.04.2018
Patent
Synthesis and transformations of d-glucuronic and l-iduronic acid glycals
Schell, Peter, Orgueira, Hernan A, Roehrig, Susanne, Seeberger, Peter H
Published in Tetrahedron letters (04.06.2001)
Published in Tetrahedron letters (04.06.2001)
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Journal Article
Orale, direkte Thrombin- und Faktor-Xa-Hemmer: Kommt die Ablösung für Warfarin, Blutegel und Schweinedärme?
Straub, Alexander, Roehrig, Susanne, Hillisch, Alexander
Published in Angewandte Chemie (09.05.2011)
Published in Angewandte Chemie (09.05.2011)
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Journal Article
SUBSTITUTED OXOPYRIDINE DERIVATIVES
TERSTEEGEN, Adrian, MEIBOM, Daniel, JIMENEZ NUNEZ, Eloisa, HILLISCH, Alexander, HEITMEIER, Stefan, ELLERBROCK, Pascal, STAMPFUSS, Jan, ACKERSTAFF, Jens, ROEHRIG, Susanne, MEIER, Katharina, LANG, Dieter
Year of Publication 26.01.2023
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Year of Publication 26.01.2023
Patent
Substituted oxopyridine derivatives
Heitmeier, Stefan, Stampfuss, Jan, Roehrig, Susanne, Tersteegen, Adrian, Ackerstaff, Jens, Meibom, Daniel, Jimenez Nunez, Eloisa, Ellerbrock, Pascal, Lang, Dieter, Hillisch, Alexander, Meier, Katharina
Year of Publication 23.11.2021
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Year of Publication 23.11.2021
Patent