Discovery and Selection of TMC114, a Next Generation HIV-1 Protease Inhibitor
Surleraux, Dominique L. N. G, Tahri, Abdellah, Verschueren, Wim G, Pille, Geert M. E, de Kock, Herman A, Jonckers, Tim H. M, Peeters, Anik, De Meyer, Sandra, Azijn, Hilde, Pauwels, Rudi, de Bethune, Marie-Pierre, King, Nancy M, Prabu-Jeyabalan, Moses, Schiffer, Celia A, Wigerinck, Piet B. T. P
Published in Journal of medicinal chemistry (24.03.2005)
Published in Journal of medicinal chemistry (24.03.2005)
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Journal Article
TMC114, a Novel Human Immunodeficiency Virus Type 1 Protease Inhibitor Active against Protease Inhibitor-Resistant Viruses, Including a Broad Range of Clinical Isolates
DE MEYER, Sandra, AZIJN, Hilde, SURLERAUX, Dominique, JOCHMANS, Dirk, TAHRI, Abdellah, PAUWELS, Rudi, WIGERINCK, Piet, DE BETHUNE, Marie-Pierre
Published in Antimicrobial Agents and Chemotherapy (01.06.2005)
Published in Antimicrobial Agents and Chemotherapy (01.06.2005)
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Design and Optimization of Tricyclic Phtalimide Analogues as Novel Inhibitors of HIV-1 Integrase
Verschueren, Wim G, Dierynck, Inge, Amssoms, Katie I. E, Hu, Lili, Boonants, Paul M. J. G, Pille, Geert M. E, Daeyaert, Frits F. D, Hertogs, Kurt, Surleraux, Dominique L. N. G, Wigerinck, Piet B. T. P
Published in Journal of medicinal chemistry (24.03.2005)
Published in Journal of medicinal chemistry (24.03.2005)
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Journal Article
Design of HIV-1 Protease Inhibitors Active on Multidrug-Resistant Virus
Surleraux, Dominique L. N. G, de Kock, Herman A, Verschueren, Wim G, Pille, Geert M. E, Maes, Louis J. R, Peeters, Anik, Vendeville, Sandrine, De Meyer, Sandra, Azijn, Hilde, Pauwels, Rudi, de Bethune, Marie-Pierre, King, Nancy M, Prabu-Jeyabalan, Moses, Schiffer, Celia A, Wigerinck, Piet B. T. P
Published in Journal of medicinal chemistry (24.03.2005)
Published in Journal of medicinal chemistry (24.03.2005)
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Journal Article
Structure-based design of a novel series of azetidine inhibitors of the hepatitis C virus NS3/4A serine protease
Parsy, Christophe, Alexandre, François-René, Brandt, Guillaume, Caillet, Catherine, Cappelle, Sylvie, Chaves, Dominique, Convard, Thierry, Derock, Michel, Gloux, Damien, Griffon, Yann, Lallos, Lisa, Leroy, Frédéric, Liuzzi, Michel, Loi, Anna-Giulia, Moulat, Laure, Musiu, Chiara, Rahali, Houcine, Roques, Virginie, Seifer, Maria, Standring, David, Surleraux, Dominique
Published in Bioorganic & medicinal chemistry letters (15.09.2014)
Published in Bioorganic & medicinal chemistry letters (15.09.2014)
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Journal Article
Binding-Site Identification and Genotypic Profiling of Hepatitis C Virus Polymerase Inhibitors
PAUWELS, Frederik, MOSTMANS, Wendy, SIMMEN, Kenneth A, QUIRYNEN, Ludo M. M, VAN DER HELM, Liesbet, BOUTTON, Carlo W, RUEFF, Anne-Stéphanie, CLEIREN, Erna, RABOISSON, Pierre, SURLERAUX, Dominique, NYANGUILE, Origène
Published in Journal of Virology (01.07.2007)
Published in Journal of Virology (01.07.2007)
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Evaluation of the anti-hepatitis C virus effect of novel potent, selective, and orally bioavailable JNK and VEGFR kinase inhibitors
Raboisson, Pierre, Lenz, Oliver, Lin, Tse-I, Surleraux, Dominique, Chakravarty, Sarvajit, Scholliers, Annick, Vermeiren, Katrien, Delouvroy, Frederic, Verbinnen, Thierry, Simmen, Kenneth
Published in Bioorganic & medicinal chemistry letters (01.04.2007)
Published in Bioorganic & medicinal chemistry letters (01.04.2007)
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Journal Article
Development of Novel Highly Specific FLT3 Targeted Inhibitors for Combination or Sequential Therapy of Acute Myeloid Leukemia
Sabir, Misbah, Hellesoy, Monica, Kivioja, Jarno, Engen, Caroline, Amiable, Claire, Popa, Mihaela, Guillon, Remi, Bruserud, Øystein, Heckman, Caroline A, McCormack, Emmet, Surleraux, Dominique, Gjertsen, Bjørn Tore
Published in Blood (08.12.2017)
Published in Blood (08.12.2017)
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단백질 키나아제 억제제로서의 퀴놀린 유도체
DEROO SABRINA, GUILLON REMI, AMIABLE CLAIRE, DIEUDONNE FRANCOIS XAVIER, LOUAT THIERRY, SURLERAUX DOMINIQUE
Year of Publication 24.05.2022
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Year of Publication 24.05.2022
Patent
The discovery of IDX21437: Design, synthesis and antiviral evaluation of 2′-α-chloro-2′-β-C-methyl branched uridine pronucleotides as potent liver-targeted HCV polymerase inhibitors
Alexandre, François-René, Badaroux, Eric, Bilello, John P., Bot, Stéphanie, Bouisset, Tony, Brandt, Guillaume, Cappelle, Sylvie, Chapron, Christopher, Chaves, Dominique, Convard, Thierry, Counor, Clément, Da Costa, Daniel, Dukhan, David, Gay, Marion, Gosselin, Gilles, Griffon, Jean-François, Gupta, Kusum, Hernandez-Santiago, Brenda, La Colla, Massimiliano, Lioure, Marie-Pierre, Milhau, Julien, Paparin, Jean-Laurent, Peyronnet, Jérôme, Parsy, Christophe, Pierra Rouvière, Claire, Rahali, Houcine, Rahali, Rachid, Salanson, Aurélien, Seifer, Maria, Serra, Ilaria, Standring, David, Surleraux, Dominique, Dousson, Cyril B.
Published in Bioorganic & medicinal chemistry letters (15.09.2017)
Published in Bioorganic & medicinal chemistry letters (15.09.2017)
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Journal Article
Discovery and structural diversity of the hepatitis C virus NS3/4A serine protease inhibitor series leading to clinical candidate IDX320
Parsy, Christophe C., Alexandre, François-René, Bidau, Valérie, Bonnaterre, Florence, Brandt, Guillaume, Caillet, Catherine, Cappelle, Sylvie, Chaves, Dominique, Convard, Thierry, Derock, Michel, Gloux, Damien, Griffon, Yann, Lallos, Lisa B., Leroy, Frederic, Liuzzi, Michel, Loi, Anna-Giulia, Moulat, Laure, Chiara, Musiu, Rahali, Houcine, Roques, Virginie, Rosinovsky, Elodie, Savin, Simon, Seifer, Maria, Standring, David, Surleraux, Dominique
Published in Bioorganic & medicinal chemistry letters (15.11.2015)
Published in Bioorganic & medicinal chemistry letters (15.11.2015)
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Journal Article
Discovery of benzophosphadiazine drug candidate IDX375: A novel hepatitis C allosteric NS5B RdRp inhibitor
Paparin, Jean-Laurent, Amador, Agnès, Badaroux, Eric, Bot, Stéphanie, Caillet, Catherine, Convard, Thierry, Da Costa, Daniel, Dukhan, David, Griffe, Ludovic, Griffon, Jean-François, LaColla, Massimiliano, Leroy, Frédéric, Liuzzi, Michel, Giulia Loi, Anna, McCarville, Joe, Mascia, Valeria, Milhau, Julien, Onidi, Loredana, Pierra, Claire, Rahali, Rachid, Rosinosky, Elodie, Sais, Efisio, Seifer, Maria, Surleraux, Dominique, Standring, David, Dousson, Cyril B.
Published in Bioorganic & medicinal chemistry letters (01.06.2017)
Published in Bioorganic & medicinal chemistry letters (01.06.2017)
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Journal Article
Synthesis of potent and broad genotypically active NS5B HCV non-nucleoside inhibitors binding to the thumb domain allosteric site 2 of the viral polymerase
Pierra Rouvière, Claire, Amador, Agnès, Badaroux, Eric, Convard, Thierry, Da Costa, Daniel, Dukhan, David, Griffe, Ludovic, Griffon, Jean-François, LaColla, Massimiliano, Leroy, Frédéric, Liuzzi, Michel, Loi, Anna Giulia, McCarville, Joe, Mascia, Valeria, Milhau, Julien, Onidi, Loredana, Paparin, Jean-Laurent, Rahali, Rachid, Sais, Efisio, Seifer, Maria, Surleraux, Dominique, Standring, David, Dousson, Cyril
Published in Bioorganic & medicinal chemistry letters (15.09.2016)
Published in Bioorganic & medicinal chemistry letters (15.09.2016)
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Journal Article
Corrigendum to “Synthesis of unnatural 3′-phospha-2′-deoxyfuranose nucleoside analogues” [Tetrahedron Lett. 55 (2014) 6328–6330]
Dayde, Bénédicte, Pierra, Claire, Gosselin, Gilles, Surleraux, Dominique, Da Costa, Daniel, Ilagouma, Amadou Tidjani, Volle, Jean-Noël, Virieux, David, Pirat, Jean-Luc
Published in Tetrahedron letters (08.04.2015)
Published in Tetrahedron letters (08.04.2015)
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Journal Article
Synthesis and antiviral evaluation of a novel series of homoserine-based inhibitors of the hepatitis C virus NS3/4A serine protease
Alexandre, François-René, Brandt, Guillaume, Caillet, Catherine, Chaves, Dominique, Convard, Thierry, Derock, Michel, Gloux, Damien, Griffon, Yann, Lallos, Lisa, Leroy, Frédéric, Liuzzi, Michel, Loi, Anna-Giulia, Moulat, Laure, Musiu, Chiara, Parsy, Christophe, Rahali, Houcine, Roques, Virginie, Seifer, Maria, Standring, David, Surleraux, Dominique
Published in Bioorganic & medicinal chemistry letters (15.09.2015)
Published in Bioorganic & medicinal chemistry letters (15.09.2015)
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Journal Article
Synthesis of Unnatural Phosphonosugar Analogues
Dayde, Bénédicte, Pierra, Claire, Gosselin, Gilles, Surleraux, Dominique, Ilagouma, Amadou Tidjani, Laborde, Coralie, Volle, Jean-Noel, Virieux, David, Pirat, Jean-Luc
Published in European journal of organic chemistry (01.02.2014)
Published in European journal of organic chemistry (01.02.2014)
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Journal Article
Corrigendum to “Synthesis of unnatural 2- and 3-deoxyfuranose analogues” [Tetrahedron Lett. 55 (2014) 3706–3708]
Dayde, Bénédicte, Pierra, Claire, Gosselin, Gilles, Surleraux, Dominique, Da Costa, Daniel, Ilagouma, Amadou Tidjani, Van der Lee, Arie, Volle, Jean-Noël, Virieux, David, Pirat, Jean-Luc
Published in Tetrahedron letters (01.04.2015)
Published in Tetrahedron letters (01.04.2015)
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Journal Article