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Discovery of (S) -2 -( (S) -2 -(3,5 -difluorophenyl ) -2-hydroxyacetamido ) -N-( (S,Z) -3 -methyl -4 -oxo -4,5 -dihydro -3H-benzo[d|[1,2 ]diazepin -5 -yl )propanamide (BMS -433796 ) : A γ-secretase inhibitor with Aβ lowering activity in a transgenic mouse model of Alzheimer's disease
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6-Hydroxybuspirone Is a Major Active Metabolite of Buspirone: Assessment of Pharmacokinetics and 5-Hydroxytryptamine 1A Receptor Occupancy in Rats
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Corrigendum to “Inhibitors of HIV-1 attachment. Part 2: An initial survey of indole substitution patterns” [Bioorg. Med. Chem. Lett. 19 (2009) 1977]
Meanwell, Nicholas A., Wallace, Owen B., Fang, Haiquan, Wang, Henry, Deshpande, Milind, Wang, Tao, Yin, Zhiwei, Zhang, Zhongxing, Pearce, Bradley C., James, Jennifer, Yeung, Kap-Sun, Qiu, Zhilei, Wright, J.J. Kim, Yang, Zheng, Zadjura, Lisa, Tweedie, Donald L., Yeola, Suresh, Zhao, Fang, Ranadive, Sunanda, Robinson, Brett A., Gong, Yi-Fei, Wang, Hwei-Gene Heidi, Spicer, Timothy P., Blair, Wade S., Shi, Pei-Yong, Colonno, Richard J., Lin, Pin-fang
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Published in Bioorganic & medicinal chemistry letters (15.02.2010)
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Discovery of (S)-2-((S)-2-(3,5-difluorophenyl)-2-hydroxyacetamido)-N-((S,Z)-3-methyl-4-oxo-4,5-dihydro-3H-benzo[d][1,2]diazepin-5-yl)propanamide (BMS-433796): a gamma-secretase inhibitor with Abeta lowering activity in a transgenic mouse model of Alzheimer's disease
Prasad, C V C, Zheng, Ming, Vig, Shikha, Bergstrom, Carl, Smith, David W, Gao, Qi, Yeola, Suresh, Polson, Craig T, Corsa, Jason A, Guss, Valerie L, Loo, Alice, Wang, Jian, Sleczka, Bogdan G, Dangler, Charles, Robertson, Barbara J, Hendrick, Joseph P, Roberts, Susan B, Barten, Donna M
Published in Bioorganic & medicinal chemistry letters (15.07.2007)
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Published in Bioorganic & medicinal chemistry letters (15.07.2007)
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Activities of the four optical isomers of 2',3'-dideoxy-3'-thiacytidine (BCH-189) against human immunodeficiency virus type 1 in human lymphocytes
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Published in Antimicrobial Agents and Chemotherapy (01.03.1992)
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MATTSON, Ronald J, DENHART, Derek J, PURANDARE, Ashok, TORTOLANI, David, YUFEN ZHAO, HUA YANG, YEOLA, Suresh, PALMER, Jane, TORRENTE, John, STARK, Arlene, JOHNSON, Graham, CATT, John D, DEE, Michael F, DESKUS, Jeffrey A, DITTA, Jonathan L, EPPERSON, James, KING, H. Dalton, AIMING GAO, POSS, Michael A
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
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Discovery of ( S)-2-(( S)-2-(3,5-difluorophenyl)-2-hydroxyacetamido)- N-(( S, Z)-3-methyl-4-oxo-4,5-dihydro-3 H-benzo[ d][1,2]diazepin-5-yl)propanamide (BMS-433796): A γ-secretase inhibitor with Aβ lowering activity in a transgenic mouse model of Alzheimer’s disease
Prasad, C.V.C., Zheng, Ming, Vig, Shikha, Bergstrom, Carl, Smith, David W., Gao, Qi, Yeola, Suresh, Polson, Craig T., Corsa, Jason A., Guss, Valerie L., Loo, Alice, Wang, Jian, Sleczka, Bogdan G., Dangler, Charles, Robertson, Barbara J., Hendrick, Joseph P., Roberts, Susan B., Barten, Donna M.
Published in Bioorganic & medicinal chemistry letters (2007)
Published in Bioorganic & medicinal chemistry letters (2007)
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In situ complexation directs the stereochemistry of N-glycosylation in the synthesis of oxathiolanyl and dioxolanyl nucleoside analogues
WOO-BAEG CHOI, WILSON, L. J, YEOLA, S, LIOTTA, D. C, SCHINAZI, R. F
Published in Journal of the American Chemical Society (01.11.1991)
Published in Journal of the American Chemical Society (01.11.1991)
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