Novel Keap1-Nrf2 Protein-Protein Interaction Inhibitor UBE-1099 Ameliorates Progressive Phenotype in Alport Syndrome Mouse Model
Kaseda, Shota, Sannomiya, Yuya, Horizono, Jun, Kuwazuru, Jun, Suico, Mary Ann, Ogi, Sayaka, Sasaki, Ryoko, Sunamoto, Hidetoshi, Fukiya, Hirohiko, Nishiyama, Hayato, Kamura, Misato, Niinou, Saki, Koyama, Yuimi, Nara, Futoshi, Shuto, Tsuyoshi, Onuma, Kazuhiro, Kai, Hirofumi
Published in Kidney360 (28.04.2022)
Published in Kidney360 (28.04.2022)
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Journal Article
Efficacy of Keap1-Nrf2 protein-protein interaction inhibitor for progressive phenotype in Alport syndrome mouse model
Shota Kaseda, Yuya Sannomiya, Jun Horizono, Jun Kuwazuru, Mary Ann Suico, Sayaka Ogi, Ryoko Sasaki, Hidetoshi Sunamoto, Hirohiko Fukiya, Hayato Nishiyama, Misato Kamura, Saki Niinou, Yuimi Koyama, Futoshi Nara, Tsuyoshi Shuto, Kazuhiro Onuma, Hirofumi Kai
Published in Japanese Journal of Pediatric Nephrology (15.11.2022)
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Published in Japanese Journal of Pediatric Nephrology (15.11.2022)
Journal Article
UBE-1099, a Novel Non-Covalent Keap1-Nrf2 Inhibitor, Protects Against Renal Ischemia-Reperfusion Injury via Nrf2 Activation: PO2508
Ogi, Sayaka, Sunamoto, Hidetoshi, Fukiya, Hirohiko, Nara, Futoshi, Onuma, Kazuhiro
Published in Journal of the American Society of Nephrology (01.10.2021)
Published in Journal of the American Society of Nephrology (01.10.2021)
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Journal Article
Novel Keap-Nrf2 Protein-Protein Interaction Inhibitor UBE-1099 Ameliorates the Severity of Experimental Alport Syndrome: PO1302
Kaseda, Shota, Suico, Mary Ann, Ogi, Sayaka, Sunamoto, Hidetoshi, Fukiya, Hirohiko, Nara, Futoshi, Shuto, Tsuyoshi, Onuma, Kazuhiro, Kai, Hirofumi
Published in Journal of the American Society of Nephrology (01.10.2021)
Published in Journal of the American Society of Nephrology (01.10.2021)
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Journal Article
Preclinical in vitro and in vivo study of UD-017, a novel highly selective and orally available CDK7 inhibitor, in a variety of cancers
Onuma, Kazuhiro, Aga, Yasuhiro, Ogi, Sayaka, Matsushita, Takashi, Sunamoto, Hidetoshi, Ogawa, Ayumi, Tokunaga, Yasunori, Ushiyama, Shigeru
Published in Journal of clinical oncology (20.05.2017)
Published in Journal of clinical oncology (20.05.2017)
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Abstract 4835: UD-017, a novel highly selective and orally active CDK7 inhibitor, shows a significant anticancer activity in patient-derived cancers
Matsushita, Takashi, Ogi, Sayaka, Onuma, Kazuhiro, Sunamoto, Hidetoshi, Ogawa, Ayumi, Hasegawa, Toru, Tokunaga, Yasunori, Aga, Yasuhiro, Ushiyama, Shigeru
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
Abstract 4837: Evaluation of anticancer activities of UD-017, a novel selective and orally available CDK7 inhibitor, in blood cancers
Aga, Yasuhiro, Ogi, Sayaka, Onuma, Kazuhiro, Sunamoto, Hidetoshi, Matsushita, Takashi, Ogawa, Ayumi, Hasegawa, toru, Kono, Shigeyuki, Iwase, Noriaki, Ushiyama, Shigeru
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Abstract LB-297: In vivo anti-tumor efficacy of UD-017, a novel highly selective & orally available CDK7 inhibitor, in colorectal cancer cells xenograft models
Aga, Yasuhiro, Ogi, Sayaka, Tokunaga, Yasunori, Ogawa, Ayumi, Onuma, Kazuhiro, Matsushita, Takashi, Sunamoto, Hidetoshi, Hasegawa, Toru, Ushiyama, Shigeru
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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Abstract LB-111: In vitro anti-cancer activity of UD-017, a novel potent & highly selective CDK7 reversible inhibitor
Matsushita, Takashi, Onuma, Kazuhiro, Sunamoto, Hidetoshi, Ogawa, Ayumi, Ogi, Sayaka, Hasegawa, Toru, Kono, Shigeyuki, Iwase, Noriaki, Aga, Yasuhiro, Ushiyama, Shigeru
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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Preclinical in vitro and in vivo evaluation of antitumor activity of UD-017, a novel selective and orally available CDK7 inhibitor, in colorectal cancer
Ogi, Sayaka, Aga, Yasuhiro, Onuma, Kazuhiro, Sunamoto, Hidetoshi, Matsushita, Takashi, Ogawa, Ayumi, Hasegawa, Tohru, Kono, Shigeyuki, Iwase, Noriaki, Tokunaga, Yasunori, Ushiyama, Shigeru
Published in Journal of clinical oncology (20.05.2017)
Published in Journal of clinical oncology (20.05.2017)
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糸球体障害を呈する慢性腎臓病モデルマウスに対するKeap1-Nrf2タンパク質間相互作用阻害薬の有効性
加世田, 将大, 三宮, 裕也, 堀園, 潤, 桑水流, 淳, Ann, Suico Mary, 小木, 彩矢佳, 佐々木, 亮子, 砂本, 秀利, 吹屋, 洋彦, 西山, 勇人, 嘉村, 美里, 奈良, 太, 首藤, 剛, 大沼, 和弘, 甲斐, 広文
Published in 日本薬理学会年会要旨集 (2022)
Published in 日本薬理学会年会要旨集 (2022)
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치환 디히드로피롤로피라졸 유도체
AGA YASUHIRO, KONO SHIGEYUKI, IWASE NORIAKI, OKUDO MAKOTO, OGI SAYAKA, KOJIMA MASAHIRO, MATSUSHITA TAKASHI, SUNAMOTO HIDETOSHI, ONUMA KAZUHIRO, USHIYAMA SHIGERU, SHIRAISHI YUSUKE, UMEZAKI SATOSHI, KIMURA TOMIO
Year of Publication 21.02.2018
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Year of Publication 21.02.2018
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SUBSTITUTED DIHYDROPYRROLOPYRAZOLE DERIVATIVE
UMEZAKI Satoshi, OKUDO Makoto, SUNAMOTO Hidetoshi, SHIRAISHI Yusuke, KIMURA Tomio, IWASE Noriaki, KONO Shigeyuki, MATSUSHITA Takashi, ONUMA Kazuhiro, USHIYAMA Shigeru, OGI Sayaka, AGA Yasuhiro, KOJIMA Masahiro
Year of Publication 22.12.2016
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Year of Publication 22.12.2016
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SUBSTITUTED DIHYDROPYRROLOPYRAZOLE COMPOUND
AGA YASUHIRO, KONO SHIGEYUKI, IWASE NORIAKI, OGI SAYAKA, KOJIMA MASAHIRO, MATSUSHITA TAKASHI, SUNAMOTO HIDETOSHI, ONUMA KAZUHIRO, TANAKA MASAYUKI, USHIYAMA SHIGERU, SHIRAISHI YUSUKE, NISHIYAMA HAYATO, MATOYAMA MASAAKI, UMEZAKI SATOSHI, KIMURA TOMIO
Year of Publication 05.07.2017
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Year of Publication 05.07.2017
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SUBSTITUTED DIHYDROPYRROLOPYRAZOLE COMPOUND
AGA YASUHIRO, KONO SHIGEYUKI, IWASE NORIAKI, OGI SAYAKA, KOJIMA MASAHIRO, MATSUSHITA TAKASHI, SUNAMOTO HIDETOSHI, ONUMA KAZUHIRO, TANAKA MASAYUKI, USHIYAMA SHIGERU, SHIRAISHI YUSUKE, NISHIYAMA HAYATO, MATOYAMA MASAAKI, UMEZAKI SATOSHI, KIMURA TOMIO
Year of Publication 06.05.2016
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Year of Publication 06.05.2016
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NOVEL INDAZOLE DERIVATIVE OR SALT THEREOF AND PRODUCTION INTERMEDIATE THEREOF, AND ANTIOXIDANT USING SAME, AND USE OF INDAZOLE DERIVATIVE OR SALT THEREOF
HAGIHARA MASAHIKO, FUJIMOTO TOMOKAZU, TAKAMA AKIRA, KOMORI KEN ICHI, KIDO KAZUTAKA, SUNAMOTO HIDETOSHI, MATSUGI TAKESHI, NISHIDA HIROSHI, TSUZAKI YASUNORI
Year of Publication 01.11.2013
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Year of Publication 01.11.2013
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SUBSTITUTED PYRIDINE COMPOUND
KIKUCHI OSAMU, IWASE NORIAKI, ITO KOJI, TAKATA KATSUNORI, SUNAMOTO HIDETOSHI, TERASAKA NAOKI, SHIMA AKIKO, NAMIKI HIDENORI, HAGIHARA MASAHIKO, TSUBOIKE KAZUNARI, NAKAMURA TSUYOSHI, SETOGUCHI HIROYUKI, YONEDA KENJI
Year of Publication 21.08.2013
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Year of Publication 21.08.2013
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NOVEL INDAZOLE DERIVATIVE OR SALT THEREOF, MANUFACTURING INTERMEDIATE THEREFOR, ANTIOXIDANT USING SAME, AND USE FOR AN INDAZOLE DERIVATIVE OR SALT THEREOF
HAGIHARA, MASAHIKO, MATSUGI, TAKESHI, SUNAMOTO, HIDETOSHI, TAKAMA, AKIRA, FUJIMOTO, TOMOKAZU, KOMORI, KEN-ICHI, TSUZAKI, YASUNORI, KIDO, KAZUTAKA, NISHIDA, HIROSHI
Year of Publication 01.12.2011
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Year of Publication 01.12.2011
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SUBSTITUTED PYRIDINE COMPOUND
TAKATA, KATSUNORI, YONEDA, KENJI, SETOGUCHI, HIROYUKI, NAMIKI, HIDENORI, SHIMA, AKIKO, KIKUCHI, OSAMU, NAKAMURA, TSUYOSHI, HAGIHARA, MASAHIKO, IWASE, NORIAKI, SUNAMOTO, HIDETOSHI, TERASAKA, NAOKI, TSUBOIKE, KAZUNARI, ITO, KOJI
Year of Publication 12.01.2012
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Year of Publication 12.01.2012
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