Synthesis and anti-inflammatory activity of the major metabolites of imrecoxib
Feng, Zhiqiang, Chu, Fengming, Guo, Zongru, Sun, Piaoyang
Published in Bioorganic & medicinal chemistry letters (15.04.2009)
Published in Bioorganic & medicinal chemistry letters (15.04.2009)
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Brij-58, a potential injectable protein-stabilizer used in therapeutic protein formulation
Yue, Liyun, Yan, Zhen, Li, Hao, Liu, Xun, Sun, Piaoyang
Published in European journal of pharmaceutics and biopharmaceutics (01.01.2020)
Published in European journal of pharmaceutics and biopharmaceutics (01.01.2020)
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Randomized, Double-Blind, Placebo-Controlled Phase III Trial of Apatinib in Patients With Chemotherapy-Refractory Advanced or Metastatic Adenocarcinoma of the Stomach or Gastroesophageal Junction
Li, Jin, Qin, Shukui, Xu, Jianming, Xiong, Jianping, Wu, Changping, Bai, Yuxian, Liu, Wei, Tong, Jiandong, Liu, Yunpeng, Xu, Ruihua, Wang, Zhehai, Wang, Qiong, Ouyang, Xuenong, Yang, Yan, Ba, Yi, Liang, Jun, Lin, Xiaoyan, Luo, Deyun, Zheng, Rongsheng, Wang, Xin, Sun, Guoping, Wang, Liwei, Zheng, Leizhen, Guo, Hong, Wu, Jingbo, Xu, Nong, Yang, Jianwei, Zhang, Honggang, Cheng, Ying, Wang, Ningju, Chen, Lei, Fan, Zhining, Sun, Piaoyang, Yu, Hao
Published in Journal of clinical oncology (01.05.2016)
Published in Journal of clinical oncology (01.05.2016)
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Design and Synthesis of 7-Oxabicyclo[2.2.1]heptane-2,3-dicarboxylic Acid Derivatives as PP5 Inhibitors To Reverse Temozolomide Resistance in Glioblastoma Multiforme
Li, Zekun, Guo, Mochen, Gu, Mingxiao, Cai, Zhongtian, Wu, Qiuyu, Yu, Jia, Tang, Meilun, He, Chenxi, Wang, Yuxuan, Sun, Piaoyang, You, Qidong, Wang, Lei
Published in Journal of medicinal chemistry (12.09.2024)
Published in Journal of medicinal chemistry (12.09.2024)
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Journal Article
Design and Synthesis of 7-Oxabicyclo2.2.1heptane-2,3-dicarboxylic Acid Derivatives as PP5 Inhibitors To Reverse Temozolomide Resistance in Glioblastoma Multiforme
Li, Zekun, Guo, Mochen, Gu, Mingxiao, Cai, Zhongtian, Wu, Qiuyu, Yu, Jia, Tang, Meilun, He, Chenxi, Wang, Yuxuan, Sun, Piaoyang, You, Qidong, Wang, Lei
Published in Journal of medicinal chemistry (12.09.2024)
Published in Journal of medicinal chemistry (12.09.2024)
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Evaluating supersaturation in vitro and predicting its performance in vivo with Biphasic gastrointestinal Simulator: A case study of a BCS IIB drug
Gan, Yanxiong, Zhang, Xue, Xu, Dengqiu, Zhang, Hongjuan, Baak, Jan P., Luo, Lin, Xia, Yulong, Wang, Jie, Ke, Xue, Sun, Piaoyang
Published in International journal of pharmaceutics (30.03.2020)
Published in International journal of pharmaceutics (30.03.2020)
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Discovery of novel orally bioavailable GPR40 agonists
Lu, Hejun, Fei, Hongbo, Yang, Fanglong, Zheng, Suxin, Hu, Qiyue, Zhang, Lei, Yuan, Jijun, Feng, Jun, Sun, Piaoyang, Dong, Qing
Published in Bioorganic & medicinal chemistry letters (15.05.2013)
Published in Bioorganic & medicinal chemistry letters (15.05.2013)
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Journal Article
Synthesis and biological evaluation of cyclopentyl-triazolol-pyrimidine (CPTP) based P2Y12 antagonists
Tu, Wangyang, Fan, Jiang, Zhang, Haitang, Xu, Guoji, Liu, Zhiwei, Qu, Jian, Yang, Fanglong, Zhang, Lei, Luan, Tianyu, Yuan, Jijun, Gong, Aishen, Feng, Jun, Sun, Piaoyang, Dong, Qing
Published in Bioorganic & medicinal chemistry letters (01.01.2014)
Published in Bioorganic & medicinal chemistry letters (01.01.2014)
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Journal Article
Synthesis and biological evaluation of cyclopentyl-triazolol-pyrimidine (CPTP) based P2Y(12) antagonists
Tu, Wangyang, Fan, Jiang, Zhang, Haitang, Xu, Guoji, Liu, Zhiwei, Qu, Jian, Yang, Fanglong, Zhang, Lei, Luan, Tianyu, Yuan, Jijun, Gong, Aishen, Feng, Jun, Sun, Piaoyang, Dong, Qing
Published in Bioorganic & medicinal chemistry letters (01.01.2014)
Published in Bioorganic & medicinal chemistry letters (01.01.2014)
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Journal Article
LAG-3 항체, 이의 항원-결합 단편 및 이의 약학적 용도
HU QIYUE, TAO WEIKANG, CAO ZHUOXIAO, FU YAYUAN, ZHANG LIANSHAN, SUN PIAOYANG
Year of Publication 05.03.2019
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Year of Publication 05.03.2019
Patent
Structure-based design and synthesis of bicyclic fused-pyridines as MEK inhibitors
Lu, Hejun, Tu, Wangyang, Fei, Hongbo, Xu, Guoji, Hu, Qiyue, Zhang, Lei, Lin, Bing, Yuan, Jijun, Yin, Junzhao, Gong, Aishen, Wan, Mimi, Wang, Dan, Zhu, Xiaoyan, Feng, Jun, Wang, Qian, Sun, Piaoyang
Published in Bioorganic & medicinal chemistry letters (01.06.2014)
Published in Bioorganic & medicinal chemistry letters (01.06.2014)
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Journal Article
항체-약물 접합체를 제조하는 방법
TAO WEIKANG, LIU YUPENG, ZHANG XIAOFEI, SHI RUIJUN, LIANG ZHI, ZHANG LIANSHAN, ZHONG JIN, LIU XUN, SUN PIAOYANG
Year of Publication 02.12.2019
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Year of Publication 02.12.2019
Patent
안정한 항-PD-1 항체 약학적 제조물 및 의료에서의 그의 적용
FANG YAN, TAO WEIKANG, YAN ZHEN, WANG PINGPING, LI JIE, ZHANG LIANSHAN, SUN PIAOYANG
Year of Publication 24.05.2018
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Year of Publication 24.05.2018
Patent
JAK Crystal Form of JAK Kinase inhibitor Bisulfate and a preparation method therefor
ZHANG QUANLIANG, CHEN YONGJIANG, WU GUAILI, SUN PIAOYANG, SHEN LINGJIA
Year of Publication 07.07.2017
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Year of Publication 07.07.2017
Patent